(Q28486239)

English

Tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide and N-benzyl-6',7'-dihydrospiro[piperidine-4,4'-thieno[3,2-c]pyran] analogues with bactericidal efficacy against Mycobacterium tuberculosis targeting MmpL3

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Tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide and N-benzyl-6',7'-dihydrospiro[piperidine-4,4'-thieno[3,2-c]pyran] analogues with bactericidal efficacy against Mycobacterium tuberculosis targeting MmpL3 (English)

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Mycobacterium tuberculosis

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Iñigo Angulo-Barturen

22

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Nicholas J. Loman

14

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Carlos Alemparte

object named as

Carlos Alemparte

4

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object named as

Lluís Ballell

26

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object named as

Mark J Pallen

15

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object named as

Gurdyal S Besra

25

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author name string

Modesto J Remuiñán

1

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Esther Pérez-Herrán

2

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Joaquín Rullás

3

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María Martínez-Hoyos

5

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David J Dow

6

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Johnson Afari

7

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Nalini Mehta

8

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Jorge Esquivias

9

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Elena Jiménez

10

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Fátima Ortega-Muro

11

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María Teresa Fraile-Gabaldón

12

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Vickey L Spivey

13

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Chrystala Constantinidou

16

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Douglas J Minick

17

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Mónica Cacho

18

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María José Rebollo-López

19

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Carolina González

20

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Verónica Sousa

21

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Alfonso Mendoza-Losana

23

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David Barros

24

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Nicholas Cammack

27

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language of work or name

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publication date

2013

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8

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4

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e60933

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copyright license

Creative Commons Attribution 4.0 International

17 April 2013

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April 2022 Public Data File from Crossref

copyright status

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Inhibition of mycolic acid transport across the Mycobacterium tuberculosis plasma membrane

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

19 March 2017

The population dynamics and control of tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

19 March 2017

Benzothiazinones kill Mycobacterium tuberculosis by blocking arabinan synthesis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

19 March 2017

PA-824 kills nonreplicating Mycobacterium tuberculosis by intracellular NO release

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

19 March 2017

A small-molecule nitroimidazopyran drug candidate for the treatment of tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

19 March 2017

Deciphering the biology of Mycobacterium tuberculosis from the complete genome sequence

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

19 March 2017

Drugs for bad bugs: confronting the challenges of antibacterial discovery

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

7 April 2017

A diarylquinoline drug active on the ATP synthase of Mycobacterium tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

7 April 2017

Fueling open-source drug discovery: 177 small-molecule leads against tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

Identification of novel inhibitors of M. tuberculosis growth using whole cell based high-throughput screening.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

SQ109 targets MmpL3, a membrane transporter of trehalose monomycolate involved in mycolic acid donation to the cell wall core of Mycobacterium tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

MmpL3 is the cellular target of the antitubercular pyrrole derivative BM212

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

The challenge of new drug discovery for tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

A chemical genetic screen in Mycobacterium tuberculosis identifies carbon-source-dependent growth inhibitors devoid of in vivo efficacy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

Getting physical in drug discovery: a contemporary perspective on solubility and hydrophobicity

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

Fast standardized therapeutic-efficacy assay for drug discovery against tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

Antituberculosis activity of the molecular libraries screening center network library

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

Identification of a new antitubercular drug candidate, SQ109, from a combinatorial library of 1,2-ethylenediamines

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

Mechanisms of inhibitory and regulatory effects of methylenedioxyphenyl compounds on cytochrome P450-dependent drug oxidation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

29 September 2017

MmpL genes are associated with mycolic acid metabolism in mycobacteria and corynebacteria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3629081

2 June 2018

Antimycobacterial Agents. Novel Diarylpyrrole Derivatives of BM212 Endowed with High Activity toward Mycobacterium tuberculosis and Low Cytotoxicity

1 reference

https://pubmed.ncbi.nlm.nih.gov/23613759

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Multidrug- and extensively drug-resistant tuberculosis: an emerging threat

1 reference

https://pubmed.ncbi.nlm.nih.gov/23613759

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1371/JOURNAL.PONE.0060933

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

2013PLoSO...860933R

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OpenCitations bibliographic resource ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

PMC publication ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

PubMed publication ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

ResearchGate publication ID

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