(Q32020825)

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Antagonists of the human CCR5 receptor as anti-HIV-1 agents. part 1: discovery and initial structure-activity relationships for 1 -amino-2-phenyl-4-(piperidin-1-yl)butanes

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Europe PubMed Central

5 July 2017

Antagonists of the human CCR5 receptor as anti-HIV-1 agents. part 1: discovery and initial structure-activity relationships for 1 -amino-2-phenyl-4-(piperidin-1-yl)butanes (English)

1 reference

Europe PubMed Central

5 July 2017

author name string

Dorn CP

1

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5 July 2017

Finke PE

2

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Europe PubMed Central

5 July 2017

Oates B

3

1 reference

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5 July 2017

Budhu RJ

4

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5 July 2017

Mills SG

5

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5 July 2017

MacCoss M

6

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5 July 2017

Malkowitz L

7

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5 July 2017

Springer MS

8

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Europe PubMed Central

5 July 2017

Daugherty BL

9

1 reference

Europe PubMed Central

5 July 2017

Gould SL

10

1 reference

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5 July 2017

DeMartino JA

11

1 reference

Europe PubMed Central

5 July 2017

Siciliano SJ

12

1 reference

Europe PubMed Central

5 July 2017

Carella A

13

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Europe PubMed Central

5 July 2017

Carver G

14

1 reference

Europe PubMed Central

5 July 2017

Holmes K

15

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5 July 2017

Danzeisen R

16

1 reference

Europe PubMed Central

5 July 2017

Hazuda D

17

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5 July 2017

Kessler J

18

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5 July 2017

Lineberger J

19

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5 July 2017

Miller M

20

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5 July 2017

Schleif WA

21

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5 July 2017

Emini EA

22

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5 July 2017

language of work or name

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publication date

1 January 2001

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5 July 2017

Bioorganic & Medicinal Chemistry Letters

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5 July 2017

11

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5 July 2017

2

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5 July 2017

259-264

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5 July 2017

HIV-1 entry - an expanding portal for drug discovery

1 reference

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The T4 gene encodes the AIDS virus receptor and is expressed in the immune system and the brain

1 reference

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7 January 2021

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Host factors and the pathogenesis of HIV-induced disease

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

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Identification of RANTES, MIP-1 alpha, and MIP-1 beta as the major HIV-suppressive factors produced by CD8+ T cells

1 reference

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7 January 2021

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The beta-chemokine receptors CCR3 and CCR5 facilitate infection by primary HIV-1 isolates

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

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A dual-tropic primary HIV-1 isolate that uses fusin and the beta-chemokine receptors CKR-5, CKR-3, and CKR-2b as fusion cofactors

1 reference

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HIV-1 entry into CD4+ cells is mediated by the chemokine receptor CC-CKR-5

1 reference

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7 January 2021

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Identification of a major co-receptor for primary isolates of HIV-1

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

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CC CKR5: a RANTES, MIP-1alpha, MIP-1beta receptor as a fusion cofactor for macrophage-tropic HIV-1

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

HIV-1 Entry Cofactor: Functional cDNA Cloning of a Seven-Transmembrane, G Protein-Coupled Receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Relative resistance to HIV-1 infection of CD4 lymphocytes from persons who remain uninfected despite multiple high-risk sexual exposure

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Homozygous defect in HIV-1 coreceptor accounts for resistance of some multiply-exposed individuals to HIV-1 infection

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

The role of viral phenotype and CCR-5 gene defects in HIV-1 transmission and disease progression

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Chemokine receptors and HIV-1: an attractive pair?

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Coreceptors--Implications for HIV Pathogenesis and Therapy

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Host factors in the pathogenesis of HIV disease

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Human chemokines: an update

1 reference

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7 January 2021

based on heuristic

inferred from DOI database lookup

CC-chemokine receptor 5 polymorphism and age of onset in familial multiple sclerosis. Multiple Sclerosis Genetics Group

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

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CCR5 Δ32, matrix metalloproteinase-9 and disease activity in multiple sclerosis

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Chemokine receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Discovery of novel, potent, and selective small-molecule CCR5 antagonists as anti-HIV-1 agents: synthesis and biological evaluation of anilide derivatives with a quaternary ammonium moiety

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

In vivo emergence of HIV-1 variants resistant to multiple protease inhibitors

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Reductive Amination of Aldehydes and Ketones with Sodium Triacetoxyborohydride. Studies on Direct and Indirect Reductive Amination Procedures(1).

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 2: structure-activity relationships for substituted 2-Aryl-1-[N-(methyl)-N-(phenylsulfonyl)amino]-4-(piperidin-1-yl)butanes

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

A critical site in the core of the CCR5 chemokine receptor required for binding and infectivity of human immunodeficiency virus type 1.

1 reference

https://api.crossref.org/works/10.1016%2FS0960-894X%2800%2900637-5

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1016/S0960-894X(00)00637-5

1 reference

Europe PubMed Central

5 July 2017

1 reference

Europe PubMed Central

5 July 2017

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