(Q33211921)

24 July 2017

title

Disulfide trapping to localize small-molecule agonists and antagonists for a G protein-coupled receptor (English)

1 reference

G protein-coupled receptor

24 July 2017

main subject

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author name string

Elizabeth Buck

series ordinal

1

1 reference

24 July 2017

James A Wells

series ordinal

2

1 reference

24 July 2017

language of work or name

English

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publication date

14 February 2005

1 reference

Proceedings of the National Academy of Sciences of the United States of America

24 July 2017

published in

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24 July 2017

volume

102

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24 July 2017

issue

8

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24 July 2017

page(s)

2719-2724

1 reference

Tethering: fragment-based drug discovery

24 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Small-molecule inhibitors of protein-protein interactions: progressing towards the dream

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Peptide-binding G protein-coupled receptors: new opportunities for drug design

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

An activation switch in the ligand binding pocket of the C5a receptor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Site-directed ligand discovery

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Crystal structure of rhodopsin: A G protein-coupled receptor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Uncovering molecular mechanisms involved in activation of G protein-coupled receptors

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Conversion of agonist site to metal-ion chelator site in the beta(2)-adrenergic receptor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

C5a receptor activation. Genetic identification of critical residues in four transmembrane helices

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Molecular tinkering of G protein-coupled receptors: an evolutionary success

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

G protein-coupled receptors. II. Mechanism of agonist activation

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Mechanism of activation and inactivation of opsin: role of Glu113 and Lys296

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Low-molecular-weight peptidic and cyclic antagonists of the receptor for the complement factor C5a.

21 June 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.0500016102

Site-specific disulfide capture of agonist and antagonist peptides on the C5a receptor

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.0500016102

The amino terminus of the human C5a receptor is required for high affinity C5a binding and for receptor activation by C5a but not C5a analogs

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Active site-directed inactivation of constitutively active mutants of rhodopsin.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=549436

Partial agonism through a zinc-Ion switch constructed between transmembrane domains III and VII in the tachykinin NK(1) receptor

31 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/15710877

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.0500016102

1 reference

24 July 2017

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1 reference

24 July 2017

1 reference