(Q33323622)

English

Substituted pyrazolo[3,4-b]pyridines as potent A1 adenosine antagonists: synthesis, biological evaluation, and development of an A1 bovine receptor model

scientific article

In more languages

Statements

scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

Substituted pyrazolo[3,4-b]pyridines as potent A1 adenosine antagonists: synthesis, biological evaluation, and development of an A1 bovine receptor model (English)

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

Maria Letizia Trincavelli

11

object named as

Maria Letizia Trincavelli

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

Adriano Martinelli

object named as

Adriano Martinelli

13

0 references

Fabrizio Manetti

object named as

Fabrizio Manetti

9

0 references

Tiziano Tuccinardi

object named as

Tiziano Tuccinardi

1

0 references

Claudia Martini

object named as

Claudia Martini

12

0 references

Silvia Schenone

2

object named as

Silvia Schenone

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

4

object named as

Chiara Brullo

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

Alessandra Tania Zizzari

7

object named as

Alessandra Tania Zizzari

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

10

object named as

Osele Ciampi

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

Francesco Bondavalli

3

object named as

Francesco Bondavalli

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

6

object named as

Luisa Mosti

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

Cristina Tintori

8

object named as

Cristina Tintori

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

14

object named as

Maurizio Botta

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

author name string

Olga Bruno

5

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

publication date

1 June 2008

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

3

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

6

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

898-913

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

Adenosine, an endogenous distress signal, modulates tissue damage and repair

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Adenosine receptors as therapeutic targets

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Animal models for the study of adenosine receptor function.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Progress in the pursuit of therapeutic adenosine receptor antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Potent adenosine A1 and A2A receptors antagonists: recent developments.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Pharmacology and therapeutic applications of A1 adenosine receptor ligands

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Adenosine receptor antagonists for cognitive dysfunction: a review of animal studies

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Expression levels of adenosine receptors in hippocampus and frontal cortex in argyrophilic grain disease

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Adenosine in the airways: implications and applications

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

2-(Benzimidazol-2-yl)quinoxalines: a novel class of selective antagonists at human A(1) and A(3) adenosine receptors designed by 3D database searching

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Tricyclic imidazoline derivatives as potent and selective adenosine A1 receptor antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and pharmacology of pyrido[2,3-d]pyrimidinediones bearing polar substituents as adenosine receptor antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

2,6,8-trisubstituted 1-deazapurines as adenosine receptor antagonists.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Potent and orally bioavailable 8-bicyclo[2.2.2]octylxanthines as adenosine A1 receptor antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and preliminary evaluation of new 1- and 3-[1-(2-hydroxy-3-phenoxypropyl)]xanthines from 2-amino-2-oxazolines as potential A1 and A2A adenosine receptor antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and biological data of 4-amino-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl esters, a new series of A1-adenosine receptor (A1AR) ligands.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis, molecular modeling studies, and pharmacological activity of selective A(1) receptor antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and 3D QSAR of new pyrazolo[3,4-b]pyridines: potent and selective inhibitors of A1 adenosine receptors

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Novel, highly potent adenosine deaminase inhibitors containing the pyrazolo[3,4-d]pyrimidine ring system. Synthesis, structure-activity relationships, and molecular modeling studies.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Chiral azole derivatives. 4. Enantiomers of bifonazole and related antifungal agents: synthesis, configuration assignment, and biological evaluation

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Functional role of internal water molecules in rhodopsin revealed by X-ray crystallography.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

An overview of recent developments in GPCR modelling: methods and validation

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Modeling of loops in protein structures

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

PROCHECK: a program to check the stereochemical quality of protein structures

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Modeling the adenosine receptors: comparison of the binding domains of A2A agonists and antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Molecular modeling of adenosine receptors: new results and trends.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Development and validation of a genetic algorithm for flexible docking

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Study on affinity profile toward native human and bovine adenosine receptors of a series of 1,8-naphthyridine derivatives

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Synthesis and Structure−Activity Relationships of a New Set of 2-Arylpyrazolo[3,4-c]quinoline Derivatives as Adenosine Receptor Antagonists

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Influence of the molecular structure of N6-(omega-aminoalkyl)adenosines on adenosine receptor affinity and intrinsic activity

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: a new class of selective A1 adenosine receptor antagonists.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as new potent and selective human A3 adenosine receptor antagonists. synthesis, pharmacological evaluation, and ligand-receptor modeling studies

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

The Protein Data Bank

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

ExPASy: The proteomics server for in-depth protein knowledge and analysis

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

CLUSTAL W: improving the sensitivity of progressive multiple sequence alignment through sequence weighting, position-specific gap penalties and weight matrix choice

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Serine and alanine mutagenesis of the nine native cysteine residues of the human A(1) adenosine receptor

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Particle mesh Ewald: An N⋅log(N) method for Ewald sums in large systems

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700355

7 January 2021

based on heuristic

inferred from DOI database lookup

Identifiers

10.1002/CMDC.200700355

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

25 July 2017

ResearchGate publication ID

0 references

Sitelinks

Wikipedia(0 entries)

Wikibooks(0 entries)

Wikinews(0 entries)

Wikiquote(0 entries)

Wikisource(0 entries)

Wikiversity(0 entries)

Wikivoyage(0 entries)

Wiktionary(0 entries)

Multilingual sites(0 entries)

Retrieved from "https://www.wikidata.org/w/index.php?title=Q33323622&oldid=1784615648"