(Q33522652)

27 July 2017

title

Chelator fragment libraries for targeting metalloproteinases. (English)

1 reference

27 July 2017

Jennifer A Jacobsen

3

0 references

Seth M Cohen

object named as

Seth M Cohen

7

0 references

author name string

Arpita Agrawal

1

1 reference

27 July 2017

Sherida L Johnson

2

1 reference

27 July 2017

Melissa T Miller

4

1 reference

27 July 2017

Li-Hsing Chen

5

1 reference

27 July 2017

Maurizio Pellecchia

6

1 reference

27 July 2017

publication date

1 February 2010

1 reference

27 July 2017

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27 July 2017

volume

5

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27 July 2017

issue

2

1 reference

27 July 2017

page(s)

195-199

1 reference

Identification and characterization of small molecule inhibitors of a class I histone deacetylase from Plasmodium falciparum

27 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Thioamide hydroxypyrothiones supersede amide hydroxypyrothiones in potency against anthrax lethal factor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Recent developments in fragment-based drug discovery

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Zinc-binding groups modulate selective inhibition of MMPs

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

A high-throughput screening approach to anthrax lethal factor inhibition

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

The design of inhibitors for medicinally relevant metalloproteins

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

A library of novel hydroxamic acids targeting the metallo-protease family: design, parallel synthesis and screening

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Structure- and fragment-based approaches to protease inhibition

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Matrix metalloproteinase inhibitors as prospective agents for the prevention and treatment of cardiovascular and neoplastic diseases

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Anthrax lethal factor protease inhibitors: synthesis, SAR, and structure-based 3D QSAR studies.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Heterocyclic zinc-binding groups for use in next-generation matrix metalloproteinase inhibitors: potency, toxicity, and reactivity

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Efficient synthetic inhibitors of anthrax lethal factor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Ligand efficiency: a useful metric for lead selection

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Identification of small molecule inhibitors of anthrax lethal factor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Synthesis of 7200 small molecules based on a substructural analysis of the histone deacetylase inhibitors trichostatin and trapoxin

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Drug-like properties and the causes of poor solubility and poor permeability

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Solid-phase synthesis of an arylsulfone hydroxamate library

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Fragment-based drug design: how big is too big?

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Evaluation and binding-mode prediction of thiopyrone-based inhibitors of anthrax lethal factor

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

A new role for old ligands: discerning chelators for zinc metalloproteinases

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

New beginnings for matrix metalloproteinase inhibitors: identification of high-affinity zinc-binding groups

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2825879

Novel small-molecule inhibitors of anthrax lethal factor identified by high-throughput screening

31 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20058293

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identification of novel anthrax lethal factor inhibitors generated by combinatorial Pictet-Spengler reaction followed by screening in situ

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20058293

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1002/CMDC.200900516

1 reference

27 July 2017

1 reference

27 July 2017

1 reference