(Q33525153)

27 July 2017

title

A high-throughput 1,536-well luminescence assay for glutathione S-transferase activity (English)

1 reference

27 July 2017

Erika L Abel

7

0 references

Adam Yasgar

object named as

Adam Yasgar

1

0 references

Anton Simeonov

10

object named as

Anton Simeonov

1 reference

27 July 2017

John Shultz

2

1 reference

27 July 2017

Wenhui Zhou

3

1 reference

27 July 2017

Hui Wang

4

1 reference

27 July 2017

Fen Huang

5

1 reference

27 July 2017

Nancy Murphy

6

1 reference

27 July 2017

John DiGiovanni

8

1 reference

27 July 2017

James Inglese

9

1 reference

27 July 2017

publication date

1 April 2010

1 reference

Assay and Drug Development Technologies

27 July 2017

published in

1 reference

27 July 2017

volume

8

1 reference

27 July 2017

issue

2

1 reference

27 July 2017

page(s)

200-211

1 reference

ADDME--Avoiding Drug Development Mistakes Early: central nervous system drug discovery perspective

27 July 2017

cites work

1 reference

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Characterization of a new fluorogenic substrate for microsomal glutathione transferase 1.

21 June 2018

1 reference

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A basis for reduced chemical library inhibition of firefly luciferase obtained from directed evolution

21 June 2018

1 reference

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An updating meta-analysis of the GSTM1, GSTT1, and GSTP1 polymorphisms and prostate cancer: a HuGE review

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

A robotic platform for quantitative high-throughput screening

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Compound Management for Quantitative High-Throughput Screening

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Characterization of chemical libraries for luciferase inhibitory activity

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Toxicology. Transforming environmental health protection

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Reporting data from high-throughput screening of small-molecule libraries

21 June 2018

1 reference

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Why drugs fail--a study on side effects in new chemical entities.

21 June 2018

1 reference

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7-Nitro-2,1,3-benzoxadiazole derivatives, a new class of suicide inhibitors for glutathione S-transferases. Mechanism of action of potential anticancer drugs

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

21 June 2018

Glutathione transferases

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

NIH Molecular Libraries Initiative

21 June 2018

1 reference

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Characterization of bromosulphophthalein binding to human glutathione S-transferase A1-1: thermodynamics and inhibition kinetics

21 June 2018

1 reference

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Drug research: myths, hype and reality

21 June 2018

1 reference

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Cancer drugs, genetic variation and the glutathione-S-transferase gene family

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

The catalytic Tyr-9 of glutathione S-transferase A1-1 controls the dynamics of the C terminus

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Concise review of the glutathione S-transferases and their significance to toxicology

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Human glutathione transferase A4-4: an alpha class enzyme with high catalytic efficiency in the conjugation of 4-hydroxynonenal and other genotoxic products of lipid peroxidation

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Glutathione-associated enzymes in anticancer drug resistance.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

The isoenzymes of glutathione transferase

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Naphthyl- and quinolylluciferin: green and red light emitting firefly luciferin analogues

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

The inhibition of glutathione S-transferases: Mechanisms, toxic consequences and therapeutic benefits

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Differential gene expression in epidermis of mice sensitive and resistant to phorbol ester skin tumor promotion

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Characterization of atrazine biotransformation by human and murine glutathione S-transferases

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Biotransformation of methyl parathion by glutathione S-transferases

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Mechanism of the glutathione transferase-catalyzed conversion of antitumor 2-crotonyloxymethyl-2-cycloalkenones to GSH adducts

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Novel class of bivalent glutathione S-transferase inhibitors

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

The polymorphic human glutathione transferase T1-1, the most efficient glutathione transferase in the denitrosation and inactivation of the anticancer drug 1,3-bis(2-chloroethyl)-1-nitrosourea

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Estimation of genomic complexity, heterologous expression, and enzymatic characterization of mouse glutathione S-transferase mGSTA4-4 (GST 5.7).

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2864799

Electrophilic aromatic substituted luciferins as bioluminescent probes for glutathione S-transferase assays

31 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20085484

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Active site architecture of polymorphic forms of human glutathione S-transferase P1-1 accounts for their enantioselectivity and disparate activity in the glutathione conjugation of 7beta,8alpha-dihydroxy-9alpha,10alpha-ox y-7,8,9,10-tetrahydrobenzo(

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20085484

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1089/ADT.2009.0248

1 reference

27 July 2017

1 reference

27 July 2017

1 reference