(Q33525920)

27 July 2017

A miniaturized screen for inhibitors of Jumonji histone demethylases (English)

1 reference

27 July 2017

Christopher J. Schofield

8

1 reference

27 July 2017

Nathan R Rose

2

0 references

Ajit Jadhav

object named as

Ajit Jadhav

5

0 references

Anton Simeonov

9

object named as

Anton Simeonov

1 reference

27 July 2017

7

Udo Oppermann

1 reference

27 July 2017

Masaaki Sakurai

1

1 reference

27 July 2017

Lena Schultz

3

1 reference

27 July 2017

Amy M Quinn

4

1 reference

27 July 2017

Stanley S Ng

6

1 reference

27 July 2017

8 October 2009

1 reference

27 July 2017

1 reference

27 July 2017

6

1 reference

27 July 2017

2

1 reference

27 July 2017

357-364

1 reference

Identification and characterization of inhibitors of human apurinic/apyrimidinic endonuclease APE1

27 July 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Synthesis and activity of N-oxalylglycine and its derivatives as Jumonji C-domain-containing histone lysine demethylase inhibitors.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Structural basis for G9a-like protein lysine methyltransferase inhibition by BIX-01294

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Prolyl 4-hydroxylases, key enzymes in the synthesis of collagens and regulation of the response to hypoxia, and their roles as treatment targets

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

A robotic platform for quantitative high-throughput screening

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Kinetic characterization and identification of a novel inhibitor of hypoxia-inducible factor prolyl hydroxylase 2 using a time-resolved fluorescence resonance energy transfer-based assay technology

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Inhibitor scaffolds for 2-oxoglutarate-dependent histone lysine demethylases

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Compound Management for Quantitative High-Throughput Screening

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Erasing the methyl mark: histone demethylases at the center of cellular differentiation and disease

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Baicalein induces functional hypoxia-inducible factor-1alpha and angiogenesis

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Expanding chemical biology of 2-oxoglutarate oxygenases

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

High-throughput screening assays for the identification of chemical probes

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Crystal structures of histone demethylase JMJD2A reveal basis for substrate specificity

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Regulation of histone methylation by demethylimination and demethylation

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Discovery and development of SAHA as an anticancer agent

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Reversal of H3K9me2 by a small-molecule inhibitor for the G9a histone methyltransferase

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Cooperative demethylation by JMJD2C and LSD1 promotes androgen receptor-dependent gene expression

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Structural and mechanistic studies on the inhibition of the hypoxia-inducible transcription factor hydroxylases by tricarboxylic acid cycle intermediates

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Quantitative high-throughput screening: a titration-based approach that efficiently identifies biological activities in large chemical libraries

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Structural studies on 2-oxoglutarate oxygenases and related double-stranded beta-helix fold proteins

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Hypoxia-inducible factor-1 activation by (-)-epicatechin gallate: potential adverse effects of cancer chemoprevention with high-dose green tea extracts

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

FeII/alpha-ketoglutarate-dependent hydroxylases and related enzymes

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

GROWTH RETARDANTS: Effects on Gibberellin Biosynthesis and Other Metabolic Pathways

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Kinase inhibitors: not just for kinases anymore

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

The dietary flavonoid quercetin modulates HIF-1 alpha activity in endothelial cells

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Inhibition of prolyl hydroxylation and procollagen processing in chick-embryo calvaria by a derivative of pyridine-2,4-dicarboxylate. Characterization of the diethyl ester as a proinhibitor

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Inhibition of lysyl hydroxylase by catechol analogs

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3401096

Evidence for hydrogen abstraction from C1 of taurine by the high-spin Fe(IV) intermediate detected during oxygen activation by taurine:alpha-ketoglutarate dioxygenase (TauD).

21 June 2018

1 reference

Selective inhibition of factor inhibiting hypoxia-inducible factor

21 January 2018

1 reference

The selectivity and inhibition of AlkB.

21 January 2018

1 reference

Iron-mediated cleavage of C-C bonds in vicinal tricarbonyl compounds in water

21 January 2018

1 reference

Interactions of flavonoids with iron and copper ions: a mechanism for their antioxidant activity.

21 January 2018

1 reference

Baicalein suppresses hypoxia-induced HIF-1alpha protein accumulation and activation through inhibition of reactive oxygen species and PI 3-kinase/Akt pathway in BV2 murine microglial cells

21 January 2018

1 reference

Flavonoids induce HIF-1alpha but impair its nuclear accumulation and activity

21 January 2018

1 reference

Novel drugs and the response to hypoxia: HIF stabilizers and prolyl hydroxylase

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20094655

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Aminosuberoyl hydroxamic acids (ASHAs): a potent new class of HDAC inhibitors

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20094655

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

A Spectrophotometric Method for Determining the Oxidative Deamination of Methylamine by the Amine Oxidases

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20094655

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1039/B912993F

1 reference

27 July 2017

1 reference

27 July 2017

1 reference