(Q33764147)

29 July 2017

title

Ex vivo activity of histone deacetylase inhibitors against multidrug-resistant clinical isolates of Plasmodium falciparum and P. vivax (English)

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29 July 2017

main subject

Plasmodium falciparum

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Plasmodium vivax

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multiple drug resistance

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Kathy T Andrews

10

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David P. Fairlie

object named as

David P Fairlie

series ordinal

7

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Enny Kenangalem

series ordinal

5

object named as

Enny Kenangalem

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29 July 2017

9

Nicholas M Anstey

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29 July 2017

8

Emiliana Tjitra

1 reference

29 July 2017

11

Ric N Price

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29 July 2017

2

Ferryanto Chalfein

1 reference

29 July 2017

6

Kim A Piera

1 reference

29 July 2017

3

Pak Prayoga

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29 July 2017

4

Frans Wabiser

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29 July 2017

1

Jutta Marfurt

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29 July 2017

language of work or name

English

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publication date

6 December 2010

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Antimicrobial Agents and Chemotherapy

29 July 2017

published in

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29 July 2017

volume

55

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29 July 2017

issue

3

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29 July 2017

page(s)

961-966

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Artemisinin combination therapy for vivax malaria

29 July 2017

cites work

1 reference

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14 July 2018

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Histone deacetylases play a major role in the transcriptional regulation of the Plasmodium falciparum life cycle

14 July 2018

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Transcriptional profiling of growth perturbations of the human malaria parasite Plasmodium falciparum

14 July 2018

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Antimalarial and antileishmanial activities of histone deacetylase inhibitors with triazole-linked cap group

14 July 2018

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14 July 2018

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14 July 2018

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14 July 2018

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Histone deacetylase inhibitors induce a very broad, pleiotropic anticancer drug resistance phenotype in acute myeloid leukemia cells by modulation of multiple ABC transporter genes

14 July 2018

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14 July 2018

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Identification and characterization of small molecule inhibitors of a class I histone deacetylase from Plasmodium falciparum

14 July 2018

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Role of known molecular markers of resistance in the antimalarial potency of piperaquine and dihydroartemisinin in vitro

14 July 2018

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Amplification of pvmdr1 associated with multidrug-resistant Plasmodium vivax

14 July 2018

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Synthesis, antimalarial activity, and intracellular targets of MEFAS, a new hybrid compound derived from mefloquine and artesunate

14 July 2018

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Malaria morbidity in Papua Indonesia, an area with multidrug resistant Plasmodium vivax and Plasmodium falciparum

14 July 2018

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Antimalarial activity of phenylthiazolyl-bearing hydroxamate-based histone deacetylase inhibitors

14 July 2018

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Multidrug-resistant Plasmodium vivax associated with severe and fatal malaria: a prospective study in Papua, Indonesia

14 July 2018

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Plasmodium vivax and mixed infections are associated with severe malaria in children: a prospective cohort study from Papua New Guinea

14 July 2018

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Plasmodium vivax trophozoites insensitive to chloroquine

14 July 2018

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The potential use of methotrexate in the treatment of falciparum malaria: in vitro assays against sensitive and multidrug-resistant falciparum strains.

14 July 2018

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14 July 2018

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Determinants of in vitro drug susceptibility testing of Plasmodium vivax

14 July 2018

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Demographic risk factors for severe and fatal vivax and falciparum malaria among hospital admissions in northeastern Indonesian Papua

14 July 2018

1 reference

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Chloroquine resistant Plasmodium vivax: in vitro characterisation and association with molecular polymorphisms

14 July 2018

1 reference

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Histone deacetylase inhibitors: molecular mechanisms of action

14 July 2018

1 reference

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HATs and HDACs: from structure, function and regulation to novel strategies for therapy and prevention

14 July 2018

1 reference

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The histone deacetylase inhibitors suberoylanilide hydroxamic (Vorinostat) and valproic acid induce irreversible and MDR1-independent resistance in human colon cancer cells

14 July 2018

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Design, synthesis, potency, and cytoselectivity of anticancer agents derived by parallel synthesis from alpha-aminosuberic acid.

14 July 2018

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Therapeutic response of multidrug-resistant Plasmodium falciparum and P. vivax to chloroquine and sulfadoxine-pyrimethamine in southern Papua, Indonesia

14 July 2018

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Plasmodium vivax: in vitro susceptibility of blood stages to synthetic trioxolane compounds and the diamidine DB75.

14 July 2018

1 reference

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In vitro metabolism of ferroquine (SSR97193) in animal and human hepatic models and antimalarial activity of major metabolites on Plasmodium falciparum.

14 July 2018

1 reference

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In vitro assessment of methylene blue on chloroquine-sensitive and -resistant Plasmodium falciparum strains reveals synergistic action with artemisinins

14 July 2018

1 reference

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Multiple drug resistance genes in malaria -- from epistasis to epidemiology

14 July 2018

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Phase I study of an oral histone deacetylase inhibitor, suberoylanilide hydroxamic acid, in patients with advanced cancer

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Chemoresistance to depsipeptide FK228 [(E)-(1S,4S,10S,21R)-7-[(Z)-ethylidene]-4,21-diisopropyl-2-oxa-12,13-dithia-5,8,20,23-tetraazabicyclo[8,7,6]-tricos-16-ene-3,6,9,22-pentanone] is mediated by reversible MDR1 induction in human cancer cell lines

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Telomeric heterochromatin propagation and histone acetylation control mutually exclusive expression of antigenic variation genes in malaria parasites

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

The global distribution and population at risk of malaria: past, present, and future

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Phase I clinical trial of histone deacetylase inhibitor: suberoylanilide hydroxamic acid administered intravenously.

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Very high risk of therapeutic failure with chloroquine for uncomplicated Plasmodium falciparum and P. vivax malaria in Indonesian Papua

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Simple in vitro assay for determining the sensitivity of Plasmodium vivax isolates from fresh human blood to antimalarials in areas where P. vivax is endemic

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

The pfmdr1 gene is associated with a multidrug-resistant phenotype in Plasmodium falciparum from the western border of Thailand.

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Molecular cloning and nuclear localization of a histone deacetylase homologue in Plasmodium falciparum

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

The removal of leucocytes from malaria infected blood

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Histone deacetylase inhibitor apicidin-mediated drug resistance: involvement of P-glycoprotein

14 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Heterochromatin silencing and locus repositioning linked to regulation of virulence genes in Plasmodium falciparum

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Evidence for different mechanisms of chloroquine resistance in 2 Plasmodium species that cause human malaria.

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

Anti-malarial effect of histone deacetylation inhibitors and mammalian tumour cytodifferentiating agents

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3067106

30 October 2018

Identifiers

DOI

10.1128/AAC.01220-10

1 reference

29 July 2017

1 reference

29 July 2017

1 reference