(Q33926024)

English

Development of a novel high-throughput screen and identification of small-molecule inhibitors of the Gα-RGS17 protein-protein interaction using AlphaScreen

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

Development of a novel high-throughput screen and identification of small-molecule inhibitors of the Gα-RGS17 protein-protein interaction using AlphaScreen (English)

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

protein-protein interaction

1 reference

based on heuristic

inferred from title

author name string

Duncan I Mackie

1

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

David L Roman

2

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

publication date

16 June 2011

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

Journal of Biomolecular Screening

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

16

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

8

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

869-877

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

Thinking outside of the "RGS box": new approaches to therapeutic targeting of regulators of G protein signaling.

1 reference

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5 July 2018

Cancer statistics, 2010

1 reference

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5 July 2018

Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins

1 reference

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5 July 2018

Identification of ligands targeting RGS proteins high-throughput screening and therapeutic potential

1 reference

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5 July 2018

Regulation of immune function by G protein-coupled receptors, trimeric G proteins, and RGS proteins.

1 reference

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5 July 2018

Regulators of G protein signaling proteins as central components of G protein-coupled receptor signaling complexes

1 reference

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5 July 2018

Polyplexed flow cytometry protein interaction assay: a novel high-throughput screening paradigm for RGS protein inhibitors

1 reference

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Stimulatory heterotrimeric G protein augments gamma ray-induced apoptosis by up-regulation of Bak expression via CREB and AP-1 in H1299 human lung cancer cells

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Fine mapping of chromosome 6q23-25 region in familial lung cancer families reveals RGS17 as a likely candidate gene

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RGS17, an overexpressed gene in human lung and prostate cancer, induces tumor cell proliferation through the cyclic AMP-PKA-CREB pathway

1 reference

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An AlphaScreen-based high-throughput screen to identify inhibitors of Hsp90-cochaperone interaction

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Regulator of G-protein signalling expression and function in ovarian cancer cell lines.

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Novel peptide ligands of RGS4 from a focused one-bead, one-compound library

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Generation of antigen-specific CTL responses using RGS1 mRNA transfected dendritic cells

1 reference

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Regulator of G-protein signalling 2 mRNA is differentially expressed in mammary epithelial subpopulations and over-expressed in the majority of breast cancers

1 reference

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Identification and characterization of T-cell epitopes deduced from RGS5, a novel broadly expressed tumor antigen

1 reference

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Overexpressed Raf-1 and phosphorylated cyclic adenosine 3'-5'-monophosphatate response element-binding protein are early markers for lung adenocarcinoma

1 reference

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5 July 2018

G-protein-coupled receptors and cancer.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5525514

5 July 2018

Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5525514

5 July 2018

Screening in a spirit haunted world

1 reference

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5 July 2018

Structure and dynamics of PKA signaling proteins

1 reference

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5 July 2018

Dynamics of signaling by PKA.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5525514

5 July 2018

RGS17/RGSZ2, a novel regulator of Gi/o, Gz, and Gq signaling

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5525514

5 July 2018

Selective expression of regulators of G-protein signaling (RGS) in the human central nervous system

1 reference

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Regulators of G protein signaling (RGS proteins): novel central nervous system drug targets

1 reference

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Seven-transmembrane receptors

1 reference

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Regulators of G-protein signalling as new central nervous system drug targets.

1 reference

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Role of the PKA-regulated transcription factor CREB in development and tumorigenesis of endocrine tissues.

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Cyclic adenosine monophosphate-dependent phosphorylation of mammalian mitochondrial proteins: enzyme and substrate characterization and functional role.

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1 reference

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1 reference

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1 reference

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Yeast-based screening for inhibitors of RGS proteins.

1 reference

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21 January 2018

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10.1177/1087057111410427

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

30 July 2017

ResearchGate publication ID

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