(Q33952708)

30 July 2017

A comparative study of fragment screening methods on the p38α kinase: new methods, new insights (English)

1 reference

30 July 2017

Scott J Pollack

1

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30 July 2017

Kim S Beyer

2

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30 July 2017

Christopher Lock

3

1 reference

30 July 2017

Ilka Müller

4

1 reference

30 July 2017

David Sheppard

5

1 reference

30 July 2017

Mike Lipkin

6

1 reference

30 July 2017

David Hardick

7

1 reference

30 July 2017

Peter Blurton

8

1 reference

30 July 2017

Philip M Leonard

9

1 reference

30 July 2017

Paul A Hubbard

10

1 reference

30 July 2017

Daniel Todd

11

1 reference

30 July 2017

Christine M Richardson

12

1 reference

30 July 2017

Thomas Ahrens

13

1 reference

30 July 2017

Manuel Baader

14

1 reference

30 July 2017

Doris O Hafenbradl

15

1 reference

30 July 2017

Kate Hilyard

16

1 reference

30 July 2017

Roland W Bürli

17

1 reference

30 July 2017

6 July 2011

1 reference

Journal of Computer - Aided Molecular Design

30 July 2017

1 reference

30 July 2017

25

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30 July 2017

677-687

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30 July 2017

7

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https://scigraph.springernature.com/pub.10.1007/s10822-011-9454-9

30 July 2017

0 references

cites work

Discovery and characterization of non-ATP site inhibitors of the mitogen activated protein (MAP) kinases

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Features and development of Coot

5 July 2018

1 reference

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p38α MAP Kinase C-Terminal Domain Binding Pocket Characterized by Crystallographic and Computational Analyses

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3155752

Phasercrystallographic software

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3155752

Recent developments in fragment-based drug discovery

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3155752

Fragment-based activity space: smaller is better

5 July 2018

1 reference

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A novel lipid binding site formed by the MAP kinase insert in p38 alpha

5 July 2018

1 reference

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Scaling and assessment of data quality

5 July 2018

1 reference

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The integration of macromolecular diffraction data

5 July 2018

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Refinement of macromolecular structures by the maximum-likelihood method

5 July 2018

1 reference

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The CCP4 suite: programs for protein crystallography

5 July 2018

1 reference

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Ligand efficiency: a useful metric for lead selection

5 July 2018

1 reference

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A ‘Rule of Three’ for fragment-based lead discovery?

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3155752

Structure validation by Calpha geometry: phi,psi and Cbeta deviation

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3155752

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3155752

The structure of mitogen-activated protein kinase p38 at 2.1-A resolution

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3155752

A protein kinase involved in the regulation of inflammatory cytokine biosynthesis

5 July 2018

1 reference

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A fluorescence lifetime-based assay for serine and threonine kinases that is suitable for high-throughput screening

5 July 2018

1 reference

Crossref

https://api.crossref.org/works/10.1007%2FS10822-011-9454-9

9-Aminoacridine peptide derivatives as versatile reporter systems for use in fluorescence lifetime assays

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1007%2FS10822-011-9454-9

Fragment-based screening by biochemical assays: Systematic feasibility studies with trypsin and MMP12.

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1007%2FS10822-011-9454-9

10.1007/S10822-011-9454-9

21 January 2018

Identifiers

DOI

1 reference

journals/jcamd/PollackBLMSLHBLHTRABHHB11

30 July 2017

1 reference

DBLP Dataset 2021-01-02

28 January 2021

1 reference

30 July 2017

1 reference