(Q34012132)

30 July 2017

title

Small molecule chemokine mimetics suggest a molecular basis for the observation that CXCL10 and CXCL11 are allosteric ligands of CXCR3 (English)

1 reference

30 July 2017

James E Pease

12

1 reference

ORCID Public Data File 2021

author name string

Belinda Nedjai

1

1 reference

30 July 2017

Hubert Li

2

1 reference

30 July 2017

Ilana L Stroke

3

1 reference

30 July 2017

Emma L Wise

4

1 reference

30 July 2017

Maria L Webb

5

1 reference

30 July 2017

J Robert Merritt

6

1 reference

30 July 2017

Ian Henderson

7

1 reference

30 July 2017

Anthony E Klon

8

1 reference

30 July 2017

Andrew G Cole

9

1 reference

30 July 2017

Richard Horuk

10

1 reference

30 July 2017

Nagarajan Vaidehi

11

1 reference

30 July 2017

language of work or name

English

0 references

publication date

1 June 2012

1 reference

British Journal of Pharmacology

30 July 2017

published in

1 reference

30 July 2017

volume

166

1 reference

30 July 2017

issue

3

1 reference

30 July 2017

page(s)

912-923

1 reference

Guide to Receptors and Channels (GRAC), 5th edition

30 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Structures of the CXCR4 chemokine GPCR with small-molecule and cyclic peptide antagonists

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Modeling small molecule-compound binding to G-protein-coupled receptors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Chemokine receptor antagonists: part 2.

5 July 2018

1 reference

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The chemokine receptor CXCR3 is degraded following internalization and is replenished at the cell surface by de novo synthesis of receptor

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Identification of CXCR3 receptor agonists in combinatorial small-molecule libraries

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

CXCR3 requires tyrosine sulfation for ligand binding and a second extracellular loop arginine residue for ligand-induced chemotaxis

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

The many roles of chemokines and chemokine receptors in inflammation

5 July 2018

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Role of CXCR3 carboxyl terminus and third intracellular loop in receptor-mediated migration, adhesion and internalization in response to CXCL11.

5 July 2018

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Accumulation of plasma cells expressing CXCR3 in the synovial sublining regions of early rheumatoid arthritis in association with production of Mig/CXCL9 by synovial fibroblasts

5 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Intracellular domains of CXCR3 that mediate CXCL9, CXCL10, and CXCL11 function

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

The G-protein-coupled receptors in the human genome form five main families. Phylogenetic analysis, paralogon groups, and fingerprints

5 July 2018

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Prediction of structure and function of G protein-coupled receptors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

The CXCR3 binding chemokine IP-10/CXCL10: structure and receptor interactions

5 July 2018

1 reference

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International Union of Pharmacology. XXX. Update on chemokine receptor nomenclature

5 July 2018

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Identification of nonpeptidic urotensin II receptor antagonists by virtual screening based on a pharmacophore model derived from structure-activity relationships and nuclear magnetic resonance studies on urotensin II.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Modeling of loops in protein structures

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Chemokines: a new classification system and their role in immunity

5 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

International union of pharmacology. XXII. Nomenclature for chemokine receptors

5 July 2018

1 reference

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A highly selective CC chemokine receptor (CCR)8 antagonist encoded by the poxvirus molluscum contagiosum

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Identification of surface residues of the monocyte chemotactic protein 1 that affect signaling through the receptor CCR2.

5 July 2018

1 reference

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The chemokine system: redundancy for robust outputs

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Binding and functional properties of recombinant and endogenous CXCR3 chemokine receptors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Interferon-inducible T cell alpha chemoattractant (I-TAC): a novel non-ELR CXC chemokine with potent activity on activated T cells through selective high affinity binding to CXCR3

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Broad spectrum chemokine antagonistic activity of a human poxvirus chemokine homolog

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Solution structure and basis for functional activity of stromal cell-derived factor-1; dissociation of CXCR4 activation from binding and inhibition of HIV-1.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Chemokine receptor specific for IP10 and mig: structure, function, and expression in activated T-lymphocytes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

The amino-terminal extracellular domain of the MCP-1 receptor, but not the RANTES/MIP-1alpha receptor, confers chemokine selectivity. Evidence for a two-step mechanism for MCP-1 receptor activation

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Antagonists of monocyte chemoattractant protein 1 identified by modification of functionally critical NH2-terminal residues

5 July 2018

1 reference

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Biochemical characterization of a gamma interferon-inducible cytokine (IP-10).

5 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

A macrophage mRNA selectively induced by gamma-interferon encodes a member of the platelet factor 4 family of cytokines

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Technique for generating three-dimensional alignments of multiple ligands from one-dimensional alignments.

5 July 2018

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Functional Selectivity and Biased Receptor Signaling

21 January 2018

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https://api.crossref.org/works/10.1111%2FJ.1476-5381.2011.01660.X

The N-terminal extracellular segments of the chemokine receptors CCR1 and CCR3 are determinants for MIP-1alpha and eotaxin binding, respectively, but a second domain is essential for efficient receptor activation

21 January 2018

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Ligand entry and exit pathways in the beta2-adrenergic receptor

21 January 2018

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Molecular characterization of the chemokine receptor CXCR3: evidence for the involvement of distinct extracellular domains in a multi‐step model of ligand binding and receptor activation

21 January 2018

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https://api.crossref.org/works/10.1111%2FJ.1476-5381.2011.01660.X

Human interferon-inducible 10-kDa protein and human interferon-inducible T cell alpha chemoattractant are allotopic ligands for human CXCR3: differential binding to receptor states.

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3417418

Lymphocyte-specific chemokine receptor CXCR3: regulation, chemokine binding and gene localization

29 October 2018

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12 December 2020

Reciprocal cross-talk between RANKL and interferon-gamma-inducible protein 10 is responsible for bone-erosive experimental arthritis

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12 December 2020

Structural requirements for interleukin-8 function identified by design of analogs and CXC chemokine hybrids

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12 December 2020

Positive versus negative modulation of different endogenous chemokines for CC-chemokine receptor 1 by small molecule agonists through allosteric versus orthosteric binding

1 reference

12 December 2020

10.1111/J.1476-5381.2011.01660.X

Identifiers

DOI

1 reference

30 July 2017

1 reference

30 July 2017

1 reference