(Q34105493)

31 July 2017

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title

Estrogen receptor beta selective nonsteroidal estrogens: seeking clinical indications (English)

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31 July 2017

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James T Dalton

10

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author name string

Michael L Mohler

1

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31 July 2017

Ramesh Narayanan

2

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31 July 2017

Christopher C Coss

3

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31 July 2017

Kejiang Hu

4

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31 July 2017

Yali He

5

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31 July 2017

Zhongzhi Wu

6

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31 July 2017

Seoung-Soo Hong

7

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31 July 2017

Dong Jin Hwang

8

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31 July 2017

Duane D Miller

9

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31 July 2017

language of work or name

English

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publication date

1 April 2010

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Expert Opinion on Therapeutic Patents

31 July 2017

published in

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31 July 2017

volume

20

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31 July 2017

issue

4

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31 July 2017

page(s)

507-534

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Molecular mechanisms of action of steroid/thyroid receptor superfamily members

31 July 2017

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21 January 2018

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Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors alpha and beta

21 January 2018

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Comparative distribution of estrogen receptor-alpha (ER-alpha) and beta (ER-beta) mRNA in the rat pituitary, gonad, and reproductive tract.

21 January 2018

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Non-steroidal subtype selective estrogens

21 January 2018

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Oestrogen receptors, receptor variants and oestrogen actions in the hypothalamic-pituitary axis

21 January 2018

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Generation and reproductive phenotypes of mice lacking estrogen receptor beta

21 January 2018

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Estrogen receptor-beta: recent lessons from in vivo studies

21 January 2018

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Elucidation of estrogen receptor function in bone with the use of mouse models

21 January 2018

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Biological role of pituitary estrogen receptors ERalpha and ERbeta on progesterone receptor expression and action and on gonadotropin and prolactin secretion in the rat.

21 January 2018

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A role for estrogen receptor beta in the regulation of growth of the ventral prostate

21 January 2018

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Estrogenic effects on prostatic differentiation and carcinogenesis

21 January 2018

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Prostatic hormonal carcinogenesis is mediated by in situ estrogen production and estrogen receptor alpha signaling.

21 January 2018

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Essential role for estrogen receptor beta in stromal-epithelial regulation of prostatic hyperplasia.

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

Benzopyrans are selective estrogen receptor beta agonists with novel activity in models of benign prostatic hyperplasia

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

Estrogen receptor beta: expression profile and possible anti-inflammatory role in disease

21 January 2018

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Selective estrogen receptor-beta agonists repress transcription of proinflammatory genes

21 January 2018

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ERbeta ligands. 3. Exploiting two binding orientations of the 2-phenylnaphthalene scaffold to achieve ERbeta selectivity

21 January 2018

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Evaluation of an Estrogen Receptor-β Agonist in Animal Models of Human Disease

21 January 2018

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Estrogen receptor beta inhibits angiogenesis and growth of T47D breast cancer xenografts

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

ERbeta isoform expression in colorectal carcinoma: an in vivo and in vitro study of clinicopathological and molecular correlates.

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

Involvement of estrogen receptor beta in terminal differentiation of mammary gland epithelium

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

Phytoestrogens regulate transcription and translation of vitamin D receptor in colon cancer cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Estrogen receptor beta functions through nongenomic mechanisms in lung cancer cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

The selective estrogen receptor-beta agonist biochanin A shows vasculoprotective effects without uterotrophic activity.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Mechanism of cardioprotection following trauma-hemorrhagic shock by a selective estrogen receptor-beta agonist: up-regulation of cardiac heat shock factor-1 and heat shock proteins

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Role of estrogen receptor subtypes in estrogen-induced organ-specific vasorelaxation after trauma-hemorrhage

21 January 2018

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Increased mortality and aggravation of heart failure in estrogen receptor-beta knockout mice after myocardial infarction

21 January 2018

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Nuclear receptor coregulators: judges, juries, and executioners of cellular regulation

21 January 2018

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Coregulator function: a key to understanding tissue specificity of selective receptor modulators

21 January 2018

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Nuclear and extranuclear pathway inputs in the regulation of global gene expression by estrogen receptors

21 January 2018

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Nuclear receptors: genomic and non-genomic effects converge.

21 January 2018

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Rapid signaling by steroid receptors

21 January 2018

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Reversal of bone loss in mice by nongenotropic signaling of sex steroids

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Frailty, osteoporosis and hip fracture: causes, consequences and therapeutic perspectives.

21 January 2018

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Estrogen receptor interaction with estrogen response elements

21 January 2018

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21 January 2018

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Structural evolutions of salicylaldoximes as selective agonists for estrogen receptor beta

21 January 2018

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ERbeta ligands. Part 2: Synthesis and structure-activity relationships of a series of 4-hydroxy-biphenyl-carbaldehyde oxime derivatives

21 January 2018

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Regulation of progesterone receptor messenger ribonucleic acid in the rat medial preoptic nucleus by estrogenic and antiestrogenic compounds: an in situ hybridization study.

21 January 2018

1 reference

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The effect of estrogens and antiestrogens in a rat model for hot flush.

21 January 2018

1 reference

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Glutamate receptor requirement for neuronal death from anoxia-reoxygenation: an in Vitro model for assessment of the neuroprotective effects of estrogens

21 January 2018

1 reference

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Synthesis and biological evaluation of 17beta-alkoxyestra-1,3, 5(10)-trienes as potential neuroprotectants against oxidative stress.

21 January 2018

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Rat uterine complement C3 expression as a model for progesterone receptor modulators: characterization of the new progestin trimegestone

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Estrogen receptor-beta potency-selective ligands: structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Regulation of metallothionein II messenger ribonucleic acid measures exogenous estrogen receptor-beta activity in SAOS-2 and LNCaPLN3 cells

21 January 2018

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Pyrazole ligands: structure-affinity/activity relationships and estrogen receptor-alpha-selective agonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Characterization of the biological roles of the estrogen receptors, ERalpha and ERbeta, in estrogen target tissues in vivo through the use of an ERalpha-selective ligand

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Broad modulation of neuropathic pain states by a selective estrogen receptor beta agonist

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

2-Phenylspiroindenes: a novel class of selective estrogen receptor modulators (SERMs).

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Bridged bicyclic cores containing a 1,1-diarylethylene motif are high-affinity subtype-selective ligands for the estrogen receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Exploration of the bicyclo[3.3.1]nonane system as a template for the development of new ligands for the estrogen receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Synthesis and evaluation of estrogen receptor ligands with bridged oxabicyclic cores containing a diarylethylene motif: estrogen antagonists of unusual structure

21 January 2018

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7-Substituted 2-phenyl-benzofurans as ER beta selective ligands

21 January 2018

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Design and synthesis of aryl diphenolic azoles as potent and selective estrogen receptor-beta ligands

21 January 2018

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Indazole estrogens: highly selective ligands for the estrogen receptor beta.

21 January 2018

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Selective activation of estrogen receptor-beta transcriptional pathways by an herbal extract.

21 January 2018

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Intermolecular interactions identify ligand-selective activity of estrogen receptor alpha/beta dimers

21 January 2018

1 reference

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Liquiritigenin is a plant-derived highly selective estrogen receptor beta agonist

21 January 2018

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Synthesis and structure-activity relationship of 3-arylbenzoxazines as selective estrogen receptor beta agonists

21 January 2018

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Benzopyrans as selective estrogen receptor beta agonists (SERBAs). Part 5: Combined A- and C-ring structure-activity relationship studies

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Benzopyrans as selective estrogen receptor beta agonists (SERBAs). Part 3: synthesis of cyclopentanone and cyclohexanone intermediates for C-ring modification

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Benzopyrans as selective estrogen receptor beta agonists (SERBAs). Part 4: functionalization of the benzopyran A-ring

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

The discovery of tetrahydrofluorenones as a new class of estrogen receptor beta-subtype selective ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Drug and cell type-specific regulation of genes with different classes of estrogen receptor beta-selective agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

ERbeta: a novel estrogen receptor offers the potential for new drug development

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

ERbeta ligands. Part 1: the discovery of ERbeta selective ligands which embrace the 4-hydroxy-biphenyl template

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

ERbeta ligands. Part 4: Synthesis and structure-activity relationships of a series of 2-phenylquinoline derivatives

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Estrogen receptor ligands: design and synthesis of new 2-arylindene-1-ones

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Structure-based design of estrogen receptor-beta selective ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Benzopyrans as selective estrogen receptor beta agonists (SERBAs). Part 2: structure-activity relationship studies on the benzopyran scaffold

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Estrogen receptor beta selective ligands: discovery and SAR of novel heterocyclic ligands

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

Toward selective ERbeta agonists for central nervous system disorders: synthesis and characterization of aryl benzthiophenes

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Isocoumarins as estrogen receptor beta selective ligands: Isomers of isoflavone phytoestrogens and their metabolites

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Bridged androstenediol analogs as ER-beta selective SERMs

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Androstene-3,5-dienes as ER-beta selective SERMs

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Androstenediol analogs as ER-beta-selective SERMs

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

6H-Benzo[c]chromen-6-one derivatives as selective ERbeta agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Estradiol or diarylpropionitrile decrease anxiety-like behavior of wildtype, but not estrogen receptor beta knockout, mice

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Adult female wildtype, but not oestrogen receptor beta knockout, mice have decreased depression-like behaviour during pro-oestrus and following administration of oestradiol or diarylpropionitrile

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

The inhibitory effect of diarylpropionitrile, a selective agonist of estrogen receptor beta, on the growth of MC38 colon cancer line

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

Genistein and phycocyanobilin may prevent hepatic fibrosis by suppressing proliferation and activation of hepatic stellate cells

21 January 2018

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https://api.crossref.org/works/10.1517%2F13543771003657164

Activation of estrogen receptor-beta regulates hippocampal synaptic plasticity and improves memory

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Estrogen receptor beta protects against acoustic trauma in mice

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

Differential involvement of estrogen receptor alpha and estrogen receptor beta in the healing promoting effect of estrogen in human keratinocytes

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543771003657164

10.1517/13543771003657164

21 January 2018

Identifiers

DOI

1 reference

31 July 2017

1 reference