(Q34107343)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

title

4'-Ethynyl-2-fluoro-2'-deoxyadenosine (EFdA) inhibits HIV-1 reverse transcriptase with multiple mechanisms (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

10

1 reference

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21 March 2020

Eleftherios Michailidis

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Andrew D Huber

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

author name string

Emily M Ryan

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Yee T Ong

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Maxwell D Leslie

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Kayla B Matzek

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Kamalendra Singh

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Bruno Marchand

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Ariel N Hagedorn

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Lisa C Rohan

11

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Eiichi N Kodama

12

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Hiroaki Mitsuya

13

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Michael A Parniak

14

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

Stefan G Sarafianos

15

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

language of work or name

English

0 references

publication date

26 June 2014

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

Journal of Biological Chemistry

21 March 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

volume

289

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

issue

35

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

page(s)

24533-24548

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

describes a project that uses

21 March 2020

ImageQuant

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC4148878/fullTextXML

inferred from PubMed Central ID database lookup

cites work

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5 July 2018

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5 July 2018

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5 July 2018

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Evaluation of Combinations of 4'-Ethynyl-2-Fluoro-2'-Deoxyadenosine with Clinically Used Antiretroviral Drugs

5 July 2018

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Effect of translocation defective reverse transcriptase inhibitors on the activity of N348I, a connection subdomain drug resistant HIV-1 reverse transcriptase mutant

5 July 2018

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5 July 2018

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Response of simian immunodeficiency virus to the novel nucleoside reverse transcriptase inhibitor 4'-ethynyl-2-fluoro-2'-deoxyadenosine in vitro and in vivo

5 July 2018

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5 July 2018

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Structural and Inhibition Studies of the RNase H Function of Xenotropic Murine Leukemia Virus-Related Virus Reverse Transcriptase

5 July 2018

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Nucleocapsid protein annealing of a primer-template enhances (+)-strand DNA synthesis and fidelity by HIV-1 reverse transcriptase

5 July 2018

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5 July 2018

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4'-C-methyl-2'-deoxyadenosine and 4'-C-ethyl-2'-deoxyadenosine inhibit HIV-1 replication

5 July 2018

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K70Q adds high-level tenofovir resistance to "Q151M complex" HIV reverse transcriptase through the enhanced discrimination mechanism

5 July 2018

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The N348I mutation at the connection subdomain of HIV-1 reverse transcriptase decreases binding to nevirapine.

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Structural Basis for the Role of the K65R Mutation in HIV-1 Reverse Transcriptase Polymerization, Excision Antagonism, and Tenofovir Resistance

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

1 reference

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Structure of a covalently trapped catalytic complex of HIV-1 reverse transcriptase: implications for drug resistance

5 July 2018

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Unblocking of chain-terminated primer by HIV-1 reverse transcriptase through a nucleotide-dependent mechanism

5 July 2018

1 reference

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Conformational coupling in DNA polymerase fidelity

5 July 2018

1 reference

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Anti-HIV drugs: 25 compounds approved within 25 years after the discovery of HIV.

5 July 2018

1 reference

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Site-specific footprinting reveals differences in the translocation status of HIV-1 reverse transcriptase. Implications for polymerase translocation and drug resistance.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M114.562694

Structures of HIV-1 RT-DNA complexes before and after incorporation of the anti-AIDS drug tenofovir

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M114.562694

Effects of primer-template sequence on ATP-dependent removal of chain-terminating nucleotide analogues by HIV-1 reverse transcriptase

21 January 2018

1 reference

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21 January 2018

1 reference

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2'-deoxy-4'-C-ethynyl-2-fluoroadenosine, a nucleoside reverse transcriptase inhibitor, is highly potent against all human immunodeficiency viruses type 1 and has low toxicity

28 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24970894

12 December 2020

inferred from PubMed ID database lookup

Enantioselective total synthesis of the potent anti-HIV nucleoside EFdA

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24970894

12 December 2020

inferred from PubMed ID database lookup

The generation of hydroxyl radicals in the reaction of molecular oxygen with polyphosphate complexes of ferrous ion

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24970894

12 December 2020

inferred from PubMed ID database lookup

Identifiers

DOI

10.1074/JBC.M114.562694

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24970894%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

1 reference