(Q34112759)

31 July 2017

title

Selective delivery of 2-hydroxy APA to Trypanosoma brucei using the melamine motif (English)

1 reference

31 July 2017

0 references

6

Michael P Barrett

0 references

Beatriz Baragaña

object named as

Beatriz Baragaña

3

0 references

Ian H. Gilbert

object named as

Ian H Gilbert

7

0 references

Margaret A. Phillips

5

object named as

Margaret A Phillips

1 reference

31 July 2017

Nina Klee

1

1 reference

31 July 2017

Pui Ee Wong

2

1 reference

31 July 2017

Farah El Mazouni

4

1 reference

31 July 2017

Michael P Barrett

6

1 reference

31 July 2017

language of work or name

English

0 references

publication date

17 June 2010

1 reference

Bioorganic & Medicinal Chemistry Letters

31 July 2017

published in

1 reference

31 July 2017

volume

20

1 reference

31 July 2017

issue

15

1 reference

31 July 2017

page(s)

4364-4366

1 reference

Novel functionalized melamine-based nitroheterocycles: synthesis and activity against trypanosomatid parasites

31 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Targeted delivery of compounds to Trypanosoma brucei using the melamine motif

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Targeting of toxic compounds to the trypanosome's interior

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Antileishmanial effect of 3-aminooxy-1-aminopropane is due to polyamine depletion

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Roles for the Trypanosoma brucei P2 transporter in DB75 uptake and resistance

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Opportunities and Challenges in Antiparasitic Drug Discovery

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Design and synthesis of a series of melamine-based nitroheterocycles with activity against Trypanosomatid parasites

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

3-Aminooxy-1-aminopropane and derivatives have an antiproliferative effect on cultured Plasmodium falciparum by decreasing intracellular polyamine concentrations

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Trypanocidal activity of melamine-based nitroheterocycles

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Chemotherapy of human African trypanosomiasis: current and future prospects

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Mechanisms of arsenical and diamidine uptake and resistance in Trypanosoma brucei

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

A perspective of polyamine metabolism

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Synthesis and biological evaluation of s-triazine substituted polyamines as potential new anti-trypanosomal drugs.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Uptake of pentamidine in Trypanosoma brucei brucei is mediated by three distinct transporters: implications for cross-resistance with arsenicals

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

X-ray structure of ornithine decarboxylase from Trypanosoma brucei: the native structure and the structure in complex with alpha-difluoromethylornithine

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Arsenical-resistant trypanosomes lack an unusual adenosine transporter

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Formation of functional cross-species heterodimers of ornithine decarboxylase

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Uptake of diamidine drugs by the P2 nucleoside transporter in melarsen-sensitive and -resistant Trypanosoma brucei brucei

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Recent advances in the biochemistry of polyamines in eukaryotes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

2-substituted 3-(aminooxy)propanamines as inhibitors of ornithine decarboxylase: synthesis and biological activity

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Loss of the high-affinity pentamidine transporter is responsible for high levels of cross-resistance between arsenical and diamidine drugs in African trypanosomes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2935964

Hypoxanthine uptake through a purine-selective nucleobase transporter in Trypanosoma brucei brucei procyclic cells is driven by protonmotive force

28 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20615694

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Characterization of a Nucleoside/Proton Symporter in ProcyclicTrypanosoma brucei brucei

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20615694

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

An approach to use an unusual adenosine transporter to selectively deliver polyamine analogues to trypanosomes

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20615694

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BMCL.2010.06.070

1 reference

31 July 2017

1 reference

31 July 2017

1 reference