(Q34143238)

31 July 2017

A fluopol-ABPP HTS assay to identify PAD inhibitors (English)

1 reference

31 July 2017

8

Benjamin F Cravatt

1 reference

31 July 2017

Bryan Knuckley

1

1 reference

31 July 2017

Justin E Jones

2

1 reference

31 July 2017

Daniel A Bachovchin

3

1 reference

31 July 2017

Jessica Slack

4

1 reference

31 July 2017

Corey P Causey

5

1 reference

31 July 2017

Steven J Brown

6

1 reference

31 July 2017

Hugh Rosen

7

1 reference

31 July 2017

Paul R Thompson

9

1 reference

31 July 2017

language of work or name

English

0 references

publication date

25 August 2010

1 reference

31 July 2017

Chemical Communications

1 reference

31 July 2017

46

1 reference

31 July 2017

38

1 reference

31 July 2017

7175-7177

1 reference

Substrate specificity and kinetic studies of PADs 1, 3, and 4 identify potent and selective inhibitors of protein arginine deiminase 3.

31 July 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Haloacetamidine-based inactivators of protein arginine deiminase 4 (PAD4): evidence that general acid catalysis promotes efficient inactivation

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Protein arginine deiminase 4 (PAD4): Current understanding and future therapeutic potential

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Identification of selective inhibitors of uncharacterized enzymes by high-throughput screening with fluorescent activity-based probes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Increased PADI4 expression in blood and tissues of patients with malignant tumors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Histone hypercitrullination mediates chromatin decondensation and neutrophil extracellular trap formation.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Regulation of p53 target gene expression by peptidylarginine deiminase 4

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Histone Arg modifications and p53 regulate the expression of OKL38, a mediator of apoptosis

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Activity-based protein profiling: from enzyme chemistry to proteomic chemistry

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Histone deimination as a response to inflammatory stimuli in neutrophils.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Protein arginine deiminase 4: evidence for a reverse protonation mechanism

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Activity-based protein profiling reagents for protein arginine deiminase 4 (PAD4): synthesis and in vitro evaluation of a fluorescently labeled probe

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Inhibitors and inactivators of protein arginine deiminase 4: functional and structural characterization.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

A fluoroacetamidine-based inactivator of protein arginine deiminase 4: design, synthesis, and in vitro and in vivo evaluation

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Kinetic characterization of protein arginine deiminase 4: a transcriptional corepressor implicated in the onset and progression of rheumatoid arthritis

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

PAD, a growing family of citrullinating enzymes: genes, features and involvement in disease

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Genotoxicity of streptonigrin: a review

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Metabolism of bioreductive antitumor compounds by purified rat and human DT-diaphorases.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Nicotinamide adenine dinucleotide (phosphate): quinone oxidoreductase (DT-diaphorase) as a target for bioreductive antitumor quinones: quinone cytotoxicity and selectivity in human lung and breast cancer cell lines

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

Profiling Protein Arginine Deiminase 4 (PAD4): a novel screen to identify PAD4 inhibitors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2943038

The effects of streptonigrin on experimental tumors

28 October 2018

1 reference

12 December 2020

Transplantable human tumors in experimental chemotherapy: effects of streptonigrin on HS No. 1 and HEp No. 3 in the rat

1 reference

12 December 2020

Preliminary observations on the use of streptonigrin as an antitumor agent in human beings

1 reference

12 December 2020

A colorimetric 96-well microtiter plate assay for the determination of enzymatically formed citrulline

1 reference

12 December 2020

An antitumor spectrum of streptonigrin

1 reference

12 December 2020

Identifiers

DOI

10.1039/C0CC02634D

1 reference

31 July 2017

1 reference

31 July 2017

1 reference