(Q34169931)

31 July 2017

title

14-Methoxymetopon, a very potent mu-opioid receptor-selective analgesic with an unusual pharmacological profile (English)

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31 July 2017

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Helmut Schmidhammer

6

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author name string

Michael A King

1

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31 July 2017

Wendy Su

2

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31 July 2017

Claire L Nielan

3

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31 July 2017

Albert H Chang

4

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31 July 2017

Johannes Schütz

5

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31 July 2017

Gavril W Pasternak

7

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31 July 2017

language of work or name

English

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publication date

1 January 2003

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European Journal of Pharmacology

31 July 2017

published in

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31 July 2017

volume

459

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31 July 2017

issue

2-3

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31 July 2017

page(s)

203-209

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Expression of two variants of the human mu opioid receptor mRNA in SK-N-SH cells and human brain

31 July 2017

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3-Methoxynaltrexone, a selective heroin/morphine-6beta-glucuronide antagonist

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

7 January 2021

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14-methoxymetopon, a potent opioid, induces no respiratory depression, less sedation, and less bradycardia than sufentanil in the dog.

7 January 2021

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Irreversible opiate agonists and antagonists: the 14-hydroxydihydromorphinone azines

7 January 2021

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Intrathecal morphine in mice: a new technique

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Dissociation of morphine's analgesic and respiratory depressant actions

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Autoradiographic analysis of mu1, mu2, and delta opioid binding in the central nervous system of C57BL/6BY and CXBK (opioid receptor-deficient) mice

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7 January 2021

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7 January 2021

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Generation of the mu opioid receptor (MOR-1) protein by three new splice variants of the Oprm gene

7 January 2021

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7 January 2021

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Opiate Analgesia: Evidence for Mediation by a Subpopulation of Opiate Receptors

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Biochemical and pharmacological evidence for opioid receptor multiplicity in the central nervous system

7 January 2021

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Differential blockade by naloxonazine of two mu opiate actions: analgesia and inhibition of gastrointestinal transit

7 January 2021

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Different mu receptor subtypes mediate spinal and supraspinal analgesia in mice.

7 January 2021

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7 January 2021

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7 January 2021

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Cloning and pharmacological characterization of a rat mu opioid receptor

7 January 2021

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Antagonism of heroin and morphine self-administration in rats by the morphine-6beta-glucuronide antagonist 3-O-methylnaltrexone.

7 January 2021

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7 January 2021

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7 January 2021

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Signal transduction efficacy of the highly potent mu opioid agonist 14-methoxymetopon

7 January 2021

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Cloning and expression of an isoform of the rat mu opioid receptor (rMOR1B) which differs in agonist induced desensitization from rMOR1.

7 January 2021

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7 January 2021

Identifiers

DOI

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31 July 2017

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