(Q34190604)

31 July 2017

Glucocorticoid Receptor Antagonism by Cyproterone Acetate and RU486 (English)

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

24 December 2023

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

24 December 2023

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

24 December 2023

author name string

Christian Honer

1

1 reference

31 July 2017

Kiyean Nam

2

1 reference

31 July 2017

Cynthia Fink

3

1 reference

31 July 2017

Paul Marshall

4

1 reference

31 July 2017

Gary Ksander

5

1 reference

31 July 2017

Wendy Cornell

7

1 reference

31 July 2017

Ronald Steele

8

1 reference

31 July 2017

Robert Schweitzer

9

1 reference

31 July 2017

Christoph Schumacher

10

1 reference

31 July 2017

Ricardo E. Chatelain

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12695529

24 December 2023

language of work or name

English

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=12695529

24 December 2023

publication date

1 May 2003

1 reference

full work available at URL

31 July 2017

https://syndication.highwire.org/content/doi/10.1124/mol.63.5.1012

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

24 December 2023

published in

Molecular Pharmacology

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31 July 2017

63

1 reference

31 July 2017

5

1 reference

31 July 2017

1012-1020

1 reference

Cyproterone. A review of its pharmacology and therapeutic efficacy in prostate cancer

31 July 2017

1

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Crystal structure of the glucocorticoid receptor ligand binding domain reveals a novel mode of receptor dimerization and coactivator recognition

24 December 2023

2

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Effect of hormone replacement therapy on insulin secretion and insulin sensitivity in postmenopausal diabetic women

24 December 2023

3

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Nuclear receptor ligand-binding domains: three-dimensional structures, molecular interactions and pharmacological implications

24 December 2023

4

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Crystal structure of the ligand-binding domain of the human nuclear receptor RXR-alpha

24 December 2023

5

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Molecular basis of agonism and antagonism in the oestrogen receptor

24 December 2023

6

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

RU486 (mifepristone): mechanisms of action and clinical uses

24 December 2023

7

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

A transcriptional co-repressor that interacts with nuclear hormone receptors

24 December 2023

8

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

24 December 2023

9

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Mechanisms of antihormone action

24 December 2023

13

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

New twists in gene regulation by glucocorticoid receptor: is DNA binding dispensable?

24 December 2023

15

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Nuclear receptor coregulators: cellular and molecular biology

24 December 2023

18

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Endocrine and metabolic effects of metformin versus ethinyl estradiol-cyproterone acetate in obese women with polycystic ovary syndrome: a randomized study

24 December 2023

19

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

The antiandrogen cyproterone acetate: discovery, chemistry, basic pharmacology, clinical use and tool in basic research

24 December 2023

20

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

24 December 2023

RU 486 development

21

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

DNA binding of the glucocorticoid receptor is not essential for survival

24 December 2023

22

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Crystal structure of the RAR-gamma ligand-binding domain bound to all-trans retinoic acid

24 December 2023

23

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Crystallographic structures of the ligand-binding domains of the androgen receptor and its T877A mutant complexed with the natural agonist dihydrotestosterone

24 December 2023

24

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

How do glucocorticoids influence stress responses? Integrating permissive, suppressive, stimulatory, and preparative actions

24 December 2023

25

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

24 December 2023

26

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism

24 December 2023

27

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Androgen receptor antagonists (antiandrogens): structure-activity relationships

24 December 2023

28

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

The mineralocorticoid activity of progesterone derivatives depends on the nature of the C18 substituent

24 December 2023

29

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Overexpression of full-length human glucocorticoid receptor in Spodoptera frugiperda cells using the baculovirus expression vector system

24 December 2023

30

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Design of ligands for the glucocorticoid and progestin receptors

24 December 2023

31

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Genetic dissection of glucocorticoid receptor function in mice

24 December 2023

32

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Experience in the long-term treatment of patients with hirsutism and/or acne with cyproterone acetate-containing preparations: Efficacy, metabolic and endocrine effects

24 December 2023

33

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

A structural role for hormone in the thyroid hormone receptor.

24 December 2023

34

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

Atomic structure of progesterone complexed with its receptor

24 December 2023

35

1 reference

https://api.crossref.org/works/10.1124/MOL.63.5.1012

24 December 2023

Identifiers

1 reference

31 July 2017

1 reference