(Q34282526)

1 August 2017

title

Identification of potent and selective non-covalent inhibitors of the Plasmodium falciparum proteasome (English)

1 reference

1 August 2017

main subject

Plasmodium falciparum

0 references

7

Matthew Bogyo

1 reference

1 August 2017

Hao Li

1

1 reference

1 August 2017

Christopher Tsu

2

1 reference

1 August 2017

Christopher Blackburn

3

1 reference

1 August 2017

Gang Li

4

1 reference

1 August 2017

Paul Hales

5

1 reference

1 August 2017

Lawrence Dick

6

1 reference

1 August 2017

language of work or name

English

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publication date

19 September 2014

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Journal of the American Chemical Society

1 August 2017

published in

1 reference

1 August 2017

volume

136

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1 August 2017

issue

39

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1 August 2017

page(s)

13562-13565

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The proteasome of malaria parasites: A multi-stage drug target for chemotherapeutic intervention?

1 August 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

N,C-Capped dipeptides with selectivity for mycobacterial proteasome over human proteasomes: role of S3 and S1 binding pockets

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Validation of the proteasome as a therapeutic target in Plasmodium using an epoxyketone inhibitor with parasite-specific toxicity

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Proteasome inhibitors: an expanding army attacking a unique target

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Threonine peptidases as drug targets against malaria

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S β5-subunit

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Assembly, structure, and function of the 26S proteasome.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

The proteasome inhibitor epoxomicin has potent Plasmodium falciparum gametocytocidal activity

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

20S proteasome and its inhibitors: crystallographic knowledge for drug development

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Proteasome inhibitors block development of Plasmodium spp.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Structure of 20S proteasome from yeast at 2.4 A resolution

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

Evolutionary origin of Plasmodium and other Apicomplexa based on rRNA genes

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

TMC-95A analogues with endocyclic biphenyl ether group as proteasome inhibitors

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4183598

TMC-95-based inhibitor design provides evidence for the catalytic versatility of the proteasome

28 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/25226494

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JA507692Y

1 reference

1 August 2017

1 reference

1 August 2017

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