(Q34409107)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

title

Discovery of ML314, a Brain Penetrant Non-Peptidic β-Arrestin Biased Agonist of the Neurotensin NTR1 Receptor (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

22

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Anthony B Pinkerton

28

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

26

Marc G Caron

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

author name string

Satyamaheshwar Peddibhotla

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Michael P Hedrick

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Paul Hershberger

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Patrick R Maloney

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Yujie Li

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Monika Milewski

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Palak Gosalia

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Wilson Gray

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Alka Mehta

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Eliot Sugarman

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Becky Hood

11

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Eigo Suyama

12

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Kevin Nguyen

13

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Susanne Heynen-Genel

14

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Stefan Vasile

15

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Sumeet Salaniwal

16

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Derek Stonich

17

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Ying Su

18

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Arianna Mangravita-Novo

19

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Michael Vicchiarelli

20

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Gregory P Roth

21

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Thomas D Y Chung

23

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Glen R Hanson

24

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

James B Thomas

25

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

Lawrence S Barak

27

1 reference

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10 March 2020

publication date

1 July 2013

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

ACS Medicinal Chemistry Letters

10 March 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

volume

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

issue

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

page(s)

846-851

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

Structure of the agonist-bound neurotensin receptor

10 March 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

The potential for selective pharmacological therapies through biased receptor signaling

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Neuropeptide receptor ligands as drugs for psychiatric diseases: the end of the beginning?

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Response of limbic neurotensin systems to methamphetamine self-administration

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Modeling of bias for the analysis of receptor signaling in biochemical systems

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Discovery of β-arrestin-biased dopamine D2 ligands for probing signal transduction pathways essential for antipsychotic efficacy

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Therapeutic potential of β-arrestin- and G protein-biased agonists.

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Teaching old receptors new tricks: biasing seven-transmembrane receptors

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Discovery of N-(4-methoxyphenyl)-N,2-dimethylquinazolin-4-amine, a potent apoptosis inducer and efficacious anticancer agent with high blood brain barrier penetration

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

The identification of nonpeptide neurotensin receptor partial agonists from the potent antagonist SR48692 using a calcium mobilization assay

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Beta-arrestins and cell signaling

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Transduction of receptor signals by beta-arrestins

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

A beta-arrestin/green fluorescent protein biosensor for detecting G protein-coupled receptor activation

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Biochemical and pharmacological activities of SR 142948A, a new potent neurotensin receptor antagonist

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Tyrosine kinase inhibitors. 8. An unusually steep structure-activity relationship for analogues of 4-(3-bromoanilino)-6,7-dimethoxyquinazoline (PD 153035), a potent inhibitor of the epidermal growth factor receptor

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Biochemical and pharmacological profile of a potent and selective nonpeptide antagonist of the neurotensin receptor

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

The Isolation of a New Hypotensive Peptide, Neurotensin, from Bovine Hypothalami

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

Characterization of radioimmunoassayable neurotensin in the rat. Its differential distribution in the central nervous system, small intestine, and stomach

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

The identification of neurotensin NTS1 receptor partial agonists through a ligand-based virtual screening approach

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

PAMPA--a drug absorption in vitro model 11. Matching the in vivo unstirred water layer thickness by individual-well stirring in microtitre plates

27 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3940307

SR142948A is a potent antagonist of the cardiovascular effects of neurotensin

27 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24611085

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML400176N

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

release_p6fnt3vs3beybdr5obtuhdbfvy

10 March 2020

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/p6fnt3vs3beybdr5obtuhdbfvy

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json

10 March 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24611085%20AND%20SRC:MED&resulttype=core&format=json