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Mechanisms of inverse agonism at G-protein-coupled receptors
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scholarly article
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
review article
1 reference
stated in
Europe PubMed Central
title
Mechanisms of inverse agonism at G-protein-coupled receptors
(English)
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
main subject
G protein-coupled receptor
0 references
author name string
Philip G Strange
series ordinal
1
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
publication date
1 February 2002
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
published in
Trends in Pharmacological Sciences
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
volume
23
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
page(s)
89-95
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
issue
2
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
cites work
An allosteric model for benzodiazepine receptor function
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7 January 2021
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Inverse, protean, and ligand-selective agonism: matters of receptor conformation
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7 January 2021
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Inverse agonism and the regulation of receptor number
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7 January 2021
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Inverse agonism at heptahelical receptors: concept, experimental approach and therapeutic potential
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7 January 2021
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Inverse agonism at G protein-coupled receptors: (patho)physiological relevance and implications for drug discovery
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS0165-6147%2802%2901993-4
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7 January 2021
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Agonist-independent regulation of constitutively active G-protein-coupled receptors
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7 January 2021
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Inverse agonism and neutral antagonism at alpha(1a)- and alpha(1b)-adrenergic receptor subtypes
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Agonist-independent activation of Gz by the 5-hydroxytryptamine1A receptor co-expressed in Spodoptera frugiperda cells. Distinguishing inverse agonists from neutral antagonists
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Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptors
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Evidence that antipsychotic drugs are inverse agonists at D2 dopamine receptors
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High constitutive activity of native H3 receptors regulates histamine neurons in brain.
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Constitutive activity and structural instability of the wild-type human H2 receptor
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Nicotinic receptors at the amino acid level
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Selective and nonselective inverse agonists for constitutively active type-1 parathyroid hormone receptors: evidence for altered receptor conformations
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Inverse agonist activity at the alpha(2A)-adrenergic receptor.
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Fluorescent labeling of purified beta 2 adrenergic receptor. Evidence for ligand-specific conformational changes
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Mechanisms of agonism and inverse agonism at serotonin 5-HT1A receptors
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Two populations of binding sites for muscarinic antagonists in the rat heart
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A Selective Inverse Agonist for Central Cannabinoid Receptor Inhibits Mitogen-activated Protein Kinase Activation Stimulated by Insulin or Insulin-like Growth Factor 1
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Characterization of recombinant human serotonin 5HT1A receptors expressed in Chinese hamster ovary cells. [3H]spiperone discriminates between the G-protein-coupled and -uncoupled forms
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Site-directed mutations in the third intracellular loop of the serotonin 5-HT(1A) receptor alter G protein coupling from G(i) to G(s) in a ligand-dependent manner
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Effects of GTP on 3H-domperidone binding and its displacement by dopamine in rat striatal homogenates
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Heterogeneity of D2 dopamine receptors in different brain regions
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G protein-coupled receptors. II. Mechanism of agonist activation.
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Porcine m2 muscarinic acetylcholine receptor-effector coupling in Chinese hamster ovary cells
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Dopamine D2 receptors selectively labeled by a benzamide neuroleptic: [3H]-YM-09151-2.
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7 January 2021
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Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation
1 reference
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Crossref
reference URL
https://api.crossref.org/works/10.1016%2FS0165-6147%2802%2901993-4
retrieved
7 January 2021
based on heuristic
inferred from DOI database lookup
Identifiers
DOI
10.1016/S0165-6147(02)01993-4
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
PubMed ID
11830266
1 reference
stated in
Europe PubMed Central
PubMed ID
11830266
retrieved
2 August 2017
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