(Q34979043)

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Differential effects of acute and repeat dosing with the H3 antagonist GSK189254 on the sleep-wake cycle and narcoleptic episodes in Ox-/- mice

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

5 August 2017

Differential effects of acute and repeat dosing with the H3 antagonist GSK189254 on the sleep-wake cycle and narcoleptic episodes in Ox-/- mice (English)

1 reference

Europe PubMed Central

PubMed publication ID

5 August 2017

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author name string

R X Guo

1

1 reference

Europe PubMed Central

PubMed publication ID

5 August 2017

C Anaclet

2

1 reference

Europe PubMed Central

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5 August 2017

J C Roberts

3

1 reference

Europe PubMed Central

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5 August 2017

R Parmentier

4

1 reference

Europe PubMed Central

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5 August 2017

M Zhang

5

1 reference

Europe PubMed Central

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5 August 2017

G Guidon

6

1 reference

Europe PubMed Central

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5 August 2017

C Buda

7

1 reference

Europe PubMed Central

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5 August 2017

J P Sastre

8

1 reference

Europe PubMed Central

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5 August 2017

J Q Feng

9

1 reference

Europe PubMed Central

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5 August 2017

P Franco

10

1 reference

Europe PubMed Central

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5 August 2017

S H Brown

11

1 reference

Europe PubMed Central

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5 August 2017

N Upton

12

1 reference

Europe PubMed Central

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5 August 2017

A D Medhurst

13

1 reference

Europe PubMed Central

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5 August 2017

J S Lin

14

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5 August 2017

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publication date

1 May 2009

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5 August 2017

British Journal of Pharmacology

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5 August 2017

157

1 reference

Europe PubMed Central

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5 August 2017

1

1 reference

Europe PubMed Central

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5 August 2017

104-117

1 reference

Europe PubMed Central

PubMed publication ID

5 August 2017

The histamine H3 receptor: an attractive target for the treatment of cognitive disorders

1 reference

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8 July 2018

Correlation between ex vivo receptor occupancy and wake-promoting activity of selective H3 receptor antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

An inverse agonist of the histamine H(3) receptor improves wakefulness in narcolepsy: studies in orexin-/- mice and patients

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Novel histamine H3 receptor antagonists GSK189254 and GSK334429 are efficacious in surgically-induced and virally-induced rat models of neuropathic pain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

GSK189254, a novel H3 receptor antagonist that binds to histamine H3 receptors in Alzheimer's disease brain and improves cognitive performance in preclinical models

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Narcolepsy with cataplexy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

The brain H3-receptor as a novel therapeutic target for vigilance and sleep-wake disorders

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Brain structures and mechanisms involved in the control of cortical activation and wakefulness, with emphasis on the posterior hypothalamus and histaminergic neurons

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Histamine H3 receptor antagonists: from target identification to drug leads

1 reference

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8 July 2018

Neuronal activity of histaminergic tuberomammillary neurons during wake-sleep states in the mouse.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

BF2.649 [1-{3-[3-(4-Chlorophenyl)propoxy]propyl}piperidine, hydrochloride], a nonimidazole inverse agonist/antagonist at the human histamine H3 receptor: Preclinical pharmacology

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Narcolepsy and the hypocretin system--where motion meets emotion

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

EFNS guidelines on management of narcolepsy.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Keynote review: histamine H3 receptor antagonists reach out for the clinic

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

The histamine H3 receptor as a novel therapeutic target for cognitive and sleep disorders

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Acute wake-promoting actions of JNJ-5207852, a novel, diamine-based H3 antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Genetic and pharmacological aspects of histamine H3 receptor heterogeneity

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

The role of histamine and the tuberomamillary nucleus in the nervous system

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Narcolepsy: genetic predisposition and neuropharmacological mechanisms. REVIEW ARTICLE.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Tolerance to daytime sedative effects of H1 antihistamines

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Anatomical, physiological, and pharmacological characteristics of histidine decarboxylase knock-out mice: evidence for the role of brain histamine in behavioral and sleep-wake control

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Behavioral characterization of mice lacking histamine H(3) receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

The physiology of brain histamine.

1 reference

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8 July 2018

Narcolepsy in orexin knockout mice: molecular genetics of sleep regulation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Neurochemical and behavioral effects of ciproxifan, a potent histamine H3-receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Inhibition of cortical acetylcholine release and cognitive performance by histamine H3 receptor activation in rats

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Histaminergic descending inputs to the mesopontine tegmentum and their role in the control of cortical activation and wakefulness in the cat.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Modulation of neurotransmitter release via histamine H3 heteroreceptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Sedative effects of antihistamines.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Potential interest in powerful and specific ligands for the histamine H3 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Involvement of histaminergic neurons in arousal mechanisms demonstrated with H3-receptor ligands in the cat.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Effects of selective activation or blockade of the histamine H3 receptor on sleep and wakefulness

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

8 July 2018

Histamine H1 receptors identified in mammalian brain membranes with [3H]mepyramine

1 reference

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8 July 2018

Slow wave sleep-inducing effects of first generation H1-antagonists.

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2009.00205.X

21 January 2018

Specificity of direct transition from wake to REM sleep in orexin/ataxin-3 transgenic narcoleptic mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

26 October 2018

Evidence for tolerance following repeated dosing in rats with ciproxifan, but not with A-304121.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

26 October 2018

[3H]Resiniferatoxin autoradiography in the CNS of wild-type and TRPV1 null mice defines TRPV1 (VR-1) protein distribution

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

26 October 2018

Waking selective neurons in the posterior hypothalamus and their response to histamine H3-receptor ligands: an electrophysiological study in freely moving cats.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

26 October 2018

Decreased brain histamine content in hypocretin/orexin receptor-2 mutated narcoleptic dogs

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2697793

26 October 2018

Sleep and waking during acute histamine H3 agonist BP 2.94 or H3 antagonist carboperamide (MR 16155) administration in rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/19413575

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

[Long-term recording of cerebral, muscular and ocular electric activities in mice]

1 reference

https://pubmed.ncbi.nlm.nih.gov/19413575

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The distribution of histamine H1-receptors in the rat brain: An autoradiographic study

1 reference

https://pubmed.ncbi.nlm.nih.gov/19413575

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Changes in histamine H3 receptor responsiveness in mouse brain

1 reference

https://pubmed.ncbi.nlm.nih.gov/19413575

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

[Genetic factors as determinants of the waking-sleep cycle in the mouse (author's transl)]

1 reference

https://pubmed.ncbi.nlm.nih.gov/19413575

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1111/J.1476-5381.2009.00205.X

1 reference

Europe PubMed Central

PubMed publication ID

5 August 2017

release_qjkanbglfrbyjnviizauev7tgu

1 reference

https://api.fatcat.wiki/v0/release/qjkanbglfrbyjnviizauev7tgu

24 November 2022

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PMC publication ID

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Europe PubMed Central

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5 August 2017

PubMed publication ID

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Europe PubMed Central

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5 August 2017

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