(Q35556324)

8 August 2017

1 reference

title

Genetic and pharmacological aspects of histamine H3 receptor heterogeneity (English)

1 reference

8 August 2017

Betty Bei Yao

4

1 reference

8 August 2017

Arthur A. Hancock

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14550847

20 March 2024

Timothy A. Esbenshade

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14550847

20 March 2024

Kathleen M. Krueger

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A14550847

20 March 2024

language of work or name

English

0 references

publication date

1 October 2003

1 reference

8 August 2017

31 October 2003

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=14550847

full work available at URL

20 March 2024

number of pages

30

1 reference

based on heuristic

inferred from page(s)

https://api.elsevier.com/content/article/PII:S0024320503007410?httpAccept=text/xml

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

https://api.elsevier.com/content/article/PII:S0024320503007410?httpAccept=text/plain

20 March 2024

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

20 March 2024

1 reference

8 August 2017

volume

73

1 reference

8 August 2017

issue

24

1 reference

8 August 2017

page(s)

3043-3072

1 reference

Pharmacological analysis of immepip and imetit homologues. Further evidence for histamine H(3) receptor heterogeneity?

8 August 2017

cites work

1

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

H3-receptors control histamine release in human brain

20 March 2024

3

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

20 March 2024

4

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine H3 receptor binding sites in rat brain membranes: modulations by guanine nucleotides and divalent cations

20 March 2024

5

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Dynamics of histamine H(3) receptor antagonists on brain histamine metabolism: do all histamine H(3) receptor antagonists act at a single site?

20 March 2024

9

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

An update on histamine H3 receptors and gastrointestinal functions

20 March 2024

10

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Definition and antagonism of histamine H 2 -receptors

20 March 2024

12

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Molecular tinkering of G protein-coupled receptors: an evolutionary success

20 March 2024

14

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Characterisation of the specific binding of the histamine H3 receptor antagonist radioligand [3H]GR168320.

20 March 2024

15

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

The physiology of brain histamine.

20 March 2024

16

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Possible participation of histamine H3 receptors in the modulation of noradrenaline release from rat spinal cord slices

20 March 2024

18

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine H3 receptor-mediated inhibition of excitatory synaptic transmission in the rat dentate gyrus in vivo.

20 March 2024

19

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Molecular and pharmacological characterization of the mouse histamine H3 receptor

20 March 2024

21

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine H3 receptors modulate the release of [3H]-acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes

20 March 2024

22

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Differential effect of sodium ions and guanine nucleotides on the binding of thioperamide and clobenpropit to histamine H3-receptors in rat cerebral cortical membranes

20 March 2024

23

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Sensitivity of histamine H3 receptor agonist-stimulated [35S]GTP gamma[S] binding to pertussis toxin.

20 March 2024

24

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

High affinity histamine H3 receptors regulate ACTH release by AtT-20 cells

20 March 2024

25

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Genomic organization and characterization of splice variants of the human histamine H3 receptor

20 March 2024

26

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine H3 receptors and the gastrointestinal tract

20 March 2024

28

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Genomic cloning, heterologous expression and pharmacological characterization of a human histamine H1 receptor

20 March 2024

30

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Effect of R-(-)-alpha-methylhistamine and thioperamide on in vivo release of norepinephrine in the rat hippocampus.

20 March 2024

31

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Identification of rat H3 receptor isoforms with different brain expression and signaling properties.

20 March 2024

32

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Two novel and selective nonimidazole histamine H3 receptor antagonists A-304121 and A-317920: I. In vitro pharmacological effects

20 March 2024

34

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Involvement of presynaptic H3 receptors in the inhibitory effect of histamine on serotonin release in the rat brain cortex.

20 March 2024

35

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Molecular cloning of the human histamine H2 receptor

20 March 2024

36

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

G-protein-coupled receptor oligomerization and its potential for drug discovery

20 March 2024

37

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Local GABAergic modulation of acetylcholine release from the cortex of freely moving rats

20 March 2024

38

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Presynaptic H3 autoreceptors modulate histamine synthesis through cAMP pathway.

20 March 2024

39

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Genomic organization and characterization of splice variants of the human histamine H3 receptor

20 March 2024

43

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Evidence that histamine homologues discriminate between H3-receptors in guinea-pig cerebral cortex and ileum longitudinal muscle myenteric plexus

20 March 2024

45

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Inhibition of sympathetic hypertensive responses in the guinea-pig by prejunctional histamine H3-receptors

20 March 2024

46

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Genomics meets histamine receptors: new subtypes, new receptors.

20 March 2024

47

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Functional identification of histamine H3-receptors in the human heart

20 March 2024

48

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

20 March 2024

49

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Characterization of the binding of the first selective radiolabelled histamine H3-receptor antagonist, [125I]-iodophenpropit, to rat brain

20 March 2024

52

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Regional expression of the histamine H(2) receptor in adult and developing rat brain

20 March 2024

53

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Autoregulation of enterochromaffin-like cell histamine secretion via the histamine 3 receptor subtype

20 March 2024

54

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Norepinephrine release from the ischemic heart is greatly enhanced in mice lacking histamine H3 receptors.

20 March 2024

55

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Guanosine 5'-(gamma-[35S]thio)triphosphate autoradiography allows selective detection of histamine H3 receptor-dependent G protein activation in rat brain tissue sections.

20 March 2024

57

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

H3 receptor gene is cloned at last

20 March 2024

59

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

20 March 2024

62

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Design, synthesis, and structure-activity relationships of novel non-imidazole histamine H(3) receptor antagonists

20 March 2024

63

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Alternative splicing of the histamine H(3) receptor mRNA at the third cytoplasmic loop is not detectable in humans

20 March 2024

65

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Cloning and functional expression of the human histamine H3 receptor

20 March 2024

69

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

G protein-linked receptors: pharmacological evidence for the formation of heterodimers

20 March 2024

70

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Inhibition of noradrenaline release from the sympathetic nerves of the human saphenous vein by presynaptic histamine H3 receptors

20 March 2024

71

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

High constitutive activity of native H3 receptors regulates histamine neurons in brain.

20 March 2024

72

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

The rat H3 receptor: gene organization and multiple isoforms.

20 March 2024

73

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Molecular cloning and characterization of a new human histamine receptor, HH4R

20 March 2024

74

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

cDNA cloning and characterization of porcine histamine H4 receptor

20 March 2024

75

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

20 March 2024

76

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

A detailed mapping of the histamine H(3) receptor and its gene transcripts in rat brain

20 March 2024

77

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histaminergic neurons modulate acetylcholine release in the ventral striatum: role of H3 histamine receptors

20 March 2024

79

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine secretion from rat enterochromaffinlike cells.

20 March 2024

80

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.

20 March 2024

81

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine H3A receptor-mediated inhibition of noradrenaline release in the mouse brain cortex

20 March 2024

82

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Potencies of antagonists chemically related to iodoproxyfan at histamine H3 receptors in mouse brain cortex and guinea-pig ileum: evidence for H3 receptor heterogeneity?

20 March 2024

83

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Modulation of neurotransmitter release via histamine H3 heteroreceptors

20 March 2024

84

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histaminergic transmission in the mammalian brain

20 March 2024

85

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Application of genomics to drug design: the example of the histamine H3 receptor.

20 March 2024

86

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Characterization of histamine H3 receptors inhibiting 5-HT release from porcine enterochromaffin cells: further evidence for H3 receptor heterogeneity

20 March 2024

87

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Long-term increase of hippocampal excitability by histamine and cyclic AMP.

20 March 2024

88

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Coupling of histamine H3 receptors to neuronal Na+/H+ exchange: a novel protective mechanism in myocardial ischemia

20 March 2024

89

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Decreased intracellular calcium mediates the histamine H3-receptor-induced attenuation of norepinephrine exocytosis from cardiac sympathetic nerve endings

20 March 2024

90

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

[125I]iodoproxyfan and related compounds: a reversible radioligand and novel classes of antagonists with high affinity and selectivity for the histamine H3 receptor.

20 March 2024

91

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Histamine modulates high-voltage-activated calcium channels in neurons dissociated from the rat tuberomammillary nucleus.

20 March 2024

92

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Cloning and cerebral expression of the guinea pig histamine H3 receptor: evidence for two isoforms

20 March 2024

93

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Chromosomal mapping and organization of the human histamine H3 receptor gene.

20 March 2024

94

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Pharmacological characterization of GT-2016, a non-thiourea-containing histamine H3 receptor antagonist: in vitro and in vivo studies

20 March 2024

95

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

The role of transmembrane helix 5 in agonist binding to the human H3 receptor

20 March 2024

99

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Pharmacological characterization of histamine H3 receptors in human saphenous vein and guinea pig ileum

20 March 2024

100

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

A new potent and selective histamine H3 receptor agonist, 4-(1H-imidazol-4-ylmethyl)piperidine.

20 March 2024

101

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Molecular cloning and pharmacology of functionally distinct isoforms of the human histamine H(3) receptor

20 March 2024

102

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

The profiles of human and primate [3H]Nalpha-methylhistamine binding differ from that of rodents.

20 March 2024

104

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Biexponential kinetics of (R)-alpha-[3H]methylhistamine binding to the rat brain H3 histamine receptor.

20 March 2024

105

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Identification of two H3-histamine receptor subtypes

20 March 2024

106

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Structure of the human histamine H3 receptor gene (HRH3) and identification of naturally occurring variations

20 March 2024

107

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Effect of blockade of postsynaptic H1 or H2 receptors or activation of presynaptic H3 receptors on catecholamine-induced stimulation of ACTH and prolactin secretion

20 March 2024

109

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Characteristics of recombinantly expressed rat and human histamine H3 receptors

20 March 2024

111

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Molecular modeling and pharmacological analysis of species-related histamine H(3) receptor heterogeneity

20 March 2024

114

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

Cloning and pharmacological characterization of the monkey histamine H3 receptor

20 March 2024

115

1 reference

https://api.crossref.org/works/10.1016/J.LFS.2003.06.003

20 March 2024

Identifiers

1 reference

8 August 2017

1 reference