(Q42164100)

English

Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.

scientific article published on January 2002

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scholarly article

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11815373%20AND%20SRC:MED&resulttype=core&format=json

6 December 2019

Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors (English)

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11815373%20AND%20SRC:MED&resulttype=core&format=json

6 December 2019

Séverine Morisset

4

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6 December 2019

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A Rouleau

1

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6 December 2019

X Ligneau

2

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6 December 2019

J Tardivel-Lacombe

3

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6 December 2019

F Gbahou

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6 December 2019

J-C Schwartz

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6 December 2019

J-M Arrang

7

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6 December 2019

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1 January 2002

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6 December 2019

British Journal of Pharmacology

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6 December 2019

135

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6 December 2019

2

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6 December 2019

383-392

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6 December 2019

Protein measurement with the Folin phenol reagent

1 reference

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26 October 2017

The physiology of brain histamine.

1 reference

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26 October 2017

High constitutive activity of native H3 receptors regulates histamine neurons in brain.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1573152

26 October 2017

Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

1 reference

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26 October 2017

Constitutive activity at serotonin 5-HT(1D) receptors: detection by homologous GTPgammaS versus [(35)S]-GTPgammaS binding isotherms.

1 reference

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26 October 2017

Inverse agonism and constitutive activity as functional correlates of serotonin h5-HT(1B) receptor/G-protein stoichiometry

1 reference

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26 October 2017

Cloning of rat histamine H(3) receptor reveals distinct species pharmacological profiles

1 reference

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26 October 2017

Inverse agonism at G protein-coupled receptors: (patho)physiological relevance and implications for drug discovery

1 reference

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26 October 2017

Constitutive activity of the histamine H(1) receptor reveals inverse agonism of histamine H(1) receptor antagonists

1 reference

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26 October 2017

Cloning and functional expression of the human histamine H3 receptor

1 reference

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26 October 2017

Novel brain-specific 5-HT4 receptor splice variants show marked constitutive activity: role of the C-terminal intracellular domain

1 reference

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26 October 2017

Neurochemical and behavioral effects of ciproxifan, a potent histamine H3-receptor antagonist

1 reference

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26 October 2017

Stimulated [35S]GTP gamma S binding by 5-HT1A receptor agonists in recombinant cell lines. Modulation of apparent efficacy by G-protein activation state

1 reference

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26 October 2017

International Union of Pharmacology. XIII. Classification of histamine receptors

1 reference

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26 October 2017

Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptors

1 reference

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26 October 2017

Constitutive activation of a single effector pathway: evidence for multiple activation states of a G protein-coupled receptor.

1 reference

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26 October 2017

Somatic mutations in the thyrotropin receptor gene cause hyperfunctioning thyroid adenomas

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26 October 2017

Constitutively active mutants of the alpha 2-adrenergic receptor

1 reference

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26 October 2017

Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

1 reference

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26 October 2017

A mutation-induced activated state of the beta 2-adrenergic receptor. Extending the ternary complex model

1 reference

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26 October 2017

Modulation of neurotransmitter release via histamine H3 heteroreceptors

2 references

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26 October 2017

https://api.crossref.org/works/10.1038%2FSJ.BJP.0704490

7 January 2021

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Inverse agonist activity of beta-adrenergic antagonists.

1 reference

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26 October 2017

Negative antagonists promote an inactive conformation of the beta 2-adrenergic receptor

1 reference

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26 October 2017

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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26 October 2017

Highly potent and selective ligands for histamine H3-receptors

1 reference

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26 October 2017

Antagonists with negative intrinsic activity at delta opioid receptors coupled to GTP-binding proteins

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26 October 2017

H3-receptors control histamine release in human brain

1 reference

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26 October 2017

S-[2-(4-imidazolyl)ethyl]isothiourea, a highly specific and potent histamine H3 receptor agonist

1 reference

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26 October 2017

Constitutive activation of the alpha 1B-adrenergic receptor by all amino acid substitutions at a single site. Evidence for a region which constrains receptor activation

1 reference

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Drug efficacy at guanine nucleotide-binding regulatory protein-linked receptors: thermodynamic interpretation of negative antagonism and of receptor activity in the absence of ligand

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26 October 2017

Use of constitutive G protein-coupled receptor activity for drug discovery.

1 reference

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29 May 2018

Constitutive activity and structural instability of the wild-type human H2 receptor

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29 May 2018

Inverse agonism at adrenergic and opioid receptors: studies with wild type and constitutively active mutant receptors.

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29 May 2018

Delta opioid modulation of the binding of guanosine-5'-O-(3-[35S]thio)triphosphate to NG108-15 cell membranes: characterization of agonist and inverse agonist effects

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Agonist and inverse agonist efficacy at human recombinant serotonin 5-HT1A receptors as a function of receptor:G-protein stoichiometry

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Structure/function relationships of calcitonin analogues as agonists, antagonists, or inverse agonists in a constitutively activated receptor cell system

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Mechanism of agonist and antagonist binding to alpha 2 adrenergic receptors: evidence for a precoupled receptor-guanine nucleotide protein complex.

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Expression analysis of the histamine H(3) receptor in developing rat tissues

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Identification of rat H3 receptor isoforms with different brain expression and signaling properties.

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Cloning and cerebral expression of the guinea pig histamine H3 receptor: evidence for two isoforms

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Facilitation of constitutive alpha(2A)-adrenoceptor activity by both single amino acid mutation (Thr(373)Lys) and g(alphao) protein coexpression: evidence for inverse agonism

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The profiles of human and primate [3H]Nalpha-methylhistamine binding differ from that of rodents

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Histamine modulates high-voltage-activated calcium channels in neurons dissociated from the rat tuberomammillary nucleus.

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Pharmacological estimation of drug-receptor dissociation constants. Statistical evaluation. I. Agonists

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Identifiers

10.1038/SJ.BJP.0704490

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11815373%20AND%20SRC:MED&resulttype=core&format=json

6 December 2019

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11815373%20AND%20SRC:MED&resulttype=core&format=json

6 December 2019

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11815373%20AND%20SRC:MED&resulttype=core&format=json

6 December 2019

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