(Q34983501)

5 August 2017

title

Identification of a series of CCK-2 receptor nonpeptide agonists: sensitivity to stereochemistry and a receptor point mutation (English)

1 reference

5 August 2017

Identification of a series of CCK-2 receptor nonpeptide agonists: Sensitivity to stereochemistry and a receptor point mutation (English)

1 reference

https://api.crossref.org/works/10.1073/PNAS.0831223100

24 December 2023

author name string

Ci Chen

3

1 reference

5 August 2017

Duan Chen

5

1 reference

5 August 2017

Chun-Mei Zhao

6

1 reference

5 August 2017

Martin Beinborn

7

1 reference

5 August 2017

Alan S. Kopin

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12697901

24 December 2023

Edward W. McBride

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12697901

24 December 2023

Roger M. Freidinger

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12697901

24 December 2023

language of work or name

English

0 references

publication date

15 April 2003

1 reference

full work available at URL

5 August 2017

http://www.pnas.org/content/100/9/5525.full.pdf

file format

Portable Document Format

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12697901

https://europepmc.org/articles/PMC154378

24 December 2023

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12697901

https://europepmc.org/articles/PMC154378?pdf=render

24 December 2023

file format

Portable Document Format

online access status

open access

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12697901

https://doi.org/10.1073/pnas.0831223100

24 December 2023

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A12697901

https://pnas.org/doi/pdf/10.1073/pnas.0831223100

24 December 2023

1 reference

https://api.crossref.org/works/10.1073/PNAS.0831223100

Proceedings of the National Academy of Sciences of the United States of America

24 December 2023

published in

1 reference

5 August 2017

volume

100

1 reference

5 August 2017

issue

9

1 reference

5 August 2017

page(s)

5525-5530

1 reference

Nonpeptide cholecystokinin-2 receptor agonists

5 August 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

CCK receptor polymorphisms: an illustration of emerging themes in pharmacogenomics

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

CCK-B antagonists in the control of anxiety and gastric acid secretion.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

International Union of Pharmacology. XXI. Structure, distribution, and functions of cholecystokinin receptors

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Chimeric G proteins allow a high-throughput signaling assay of Gi-coupled receptors

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

The design and pharmacology of novel selective muscarinic agonists and antagonists

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Novel aspects of gastrin-induced activation of histidine decarboxylase in rat stomach ECL cells

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Mutations within the cholecystokinin-B/gastrin receptor ligand 'pocket' interconvert the functions of nonpeptide agonists and antagonists.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Inter- and intraspecies polymorphisms in the cholecystokinin-B/gastrin receptor alter drug efficacy

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

A beta-arrestin/green fluorescent protein biosensor for detecting G protein-coupled receptor activation

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Abnormal gastric histology and decreased acid production in cholecystokinin-B/gastrin receptor-deficient mice.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Discovery of 1,5-benzodiazepines with peripheral cholecystokinin (CCK-A) receptor agonist activity. 1. Optimization of the agonist "trigger".

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

High-affinity and potent, water-soluble 5-amino-1,4-benzodiazepine CCKB/gastrin receptor antagonists containing a cationic solubilizing group

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Biological actions of cholecystokinin

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

The human brain cholecystokinin-B/gastrin receptor. Cloning and characterization

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Tools for investigating functional interactions between ligands and G-protein-coupled receptors

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Benzodiazepine gastrin and brain cholecystokinin receptor ligands: L-365,260.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=154378

Minor modifications of a cholecystokinin-B/gastrin receptor non-peptide antagonist confer a broad spectrum of functional properties

8 July 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0831223100

A quantitative method for measuring spontaneous gastric secretion in the rat

21 January 2018

1 reference

12 December 2020

Discovery of L-162,313: a nonpeptide that mimics the biological actions of angiotensin II

1 reference

12 December 2020

Characterization of novel peptoid agonists for the CCK-A receptor

1 reference

12 December 2020

Dual agonistic and antagonistic property of nonpeptide angiotensin AT1 ligands: susceptibility to receptor mutations

1 reference

12 December 2020

Protean agonism at alpha2A-adrenoceptors

1 reference

12 December 2020

Plasma gastrin and gastric enterochromaffinlike cell activation and proliferation. Studies with omeprazole and ranitidine in intact and antrectomized rats

1 reference

12 December 2020

A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260

1 reference

12 December 2020

The role of the cholecystokinin-B/gastrin receptor transmembrane domains in determining affinity for subtype-selective ligands

1 reference

12 December 2020

Pharmacological Reviews

4

51

745

Noble F

1999

1 reference

https://api.crossref.org/works/10.1073/PNAS.0831223100

24 December 2023

Molecular Pharmacology

22

53

963

Jansson C C

1998

1 reference

https://api.crossref.org/works/10.1073/PNAS.0831223100

American Journal of Physiology

24 December 2023

28

268

R820

Kivlighn S D

1995

1 reference

https://api.crossref.org/works/10.1073/PNAS.0831223100

Progress in drug research. Fortschritte der Arzneimittelforschung. Progres des recherches pharmaceutiques

24 December 2023

29

8

262

Archer S

1965

1 reference

https://api.crossref.org/works/10.1073/PNAS.0831223100

24 December 2023

Identifiers

1 reference

release_6uxzletfpbc4novi4trqtl7sry

5 August 2017

0 references

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/6uxzletfpbc4novi4trqtl7sry

24 November 2022

mapped directly with Wikidata item

PMC publication ID

154378

1 reference

5 August 2017

1 reference