(Q35041394)

6 August 2017

Stereoselective interaction of thiopentone enantiomers with the GABA(A) receptor (English)

1 reference

6 August 2017

1 reference

1 reference

D J Cordato

1

1 reference

6 August 2017

M Chebib

2

1 reference

6 August 2017

L E Mather

3

1 reference

6 August 2017

G K Herkes

4

1 reference

6 August 2017

G A Johnston

5

1 reference

6 August 2017

language of work or name

English

0 references

publication date

1 September 1999

1 reference

British Journal of Pharmacology

6 August 2017

1 reference

6 August 2017

128

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6 August 2017

1

1 reference

6 August 2017

77-82

1 reference

Electroencephalographic effects of thiopentone and its enantiomers in the rat: correlation with drug tissue distribution.

6 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Binding, gating, affinity and efficacy: the interpretation of structure-activity relationships for agonists and of the effects of mutating receptors

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Nitric oxide-induced cytotoxicity attenuation by thiopentone sodium but not pentobarbitone sodium in primary brain cultures

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

The effect of thiopental and propofol on NMDA- and AMPA-mediated glutamate excitotoxicity.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pharmacokinetics of thiopentone enantiomers following intravenous injection or prolonged infusion of rac-thiopentone

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

The systemic and cerebral kinetics of thiopental in sheep: enantiomeric analysis.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Barbiturate interactions at the human GABAA receptor: dependence on receptor subunit combination

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

GABAA receptor pharmacology

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

The role of the GABAA receptor/chloride channel complex in anesthesia.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pharmacokinetics of high-dose thiopental used in cerebral resuscitation.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pharmacokinetics and plasma binding of thiopental. I: Studies in surgical patients

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Anesthetic potency and acute toxicity of optically active disubstituted barbituric acids

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pentobarbitone formation during thiopentone infusion.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Thiopental pharmacokinetics under conditions of long-term infusion

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Actions of pentobarbital on rat brain receptors expressed in Xenopus oocytes.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Modulation of the GABAA receptor by depressant barbiturates and pregnane steroids

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Affinities of barbiturates for the GABA-receptor complex and A1 adenosine receptors: a possible explanation of their excitatory effects.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pharmacokinetic effects of vigabatrin on cerebrospinal fluid amino acids in humans

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

gamma-Aminobutyric-acid- and pentobarbitone-gated chloride currents in internally perfused frog sensory neurones

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Barbiturate and benzodiazepine modulation of GABA receptor binding and function

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Thiopental pharmacodynamics. II. Quantitation of clinical and electroencephalographic depth of anesthesia

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pharmacological comparison of R(+), S(−) and racemic thiopentone in mice

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

The fate of thiopental in man and a method for its estimation in biological material.

8 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pharmacokinetics of thiopental enantiomers during and following prolonged high-dose therapy.

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Enantioselectivity of thiopental distribution into the central neural tissue of rats: an interaction with halothane.

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Barbiturates impair astrocyte glutamate uptake.

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Pharmacokinetics of thiopental and pentobarbital enantiomers after intravenous administration of racemic thiopental.

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

High-performance liquid chromatographic determination of thiopentone enantiomers in sheep plasma.

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Non linear disposition of thiopentone following long-term infusion.

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Calcium current block by (-)-pentobarbital, phenobarbital, and CHEB but not (+)-pentobarbital in acutely isolated hippocampal CA1 neurons: comparison with effects on GABA-activated Cl- current

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Interactions of barbiturates of various pharmacological categories with benzodiazepine receptors

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Barbiturates: Their in vivo effects and potential biochemical mechanisms

25 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1571590

Electroencephalographic effects of thiopentone and its enantiomers in the rat.

25 October 2018

1 reference

12 December 2020

Biophysical and pharmacological properties of cloned GABAA receptor subunits expressed in Xenopus oocytes

1 reference

12 December 2020

Kinetic properties of the pentobarbitone-gated chloride current in frog sensory neurones

1 reference

12 December 2020

Chloride current induced by injection of calcium into Xenopus oocytes

1 reference

12 December 2020

(-)Pentobarbital opens ion channels of long duration in cultured mouse spinal neurons

1 reference

12 December 2020

Cholinergic and catecholaminergic receptors in the Xenopus oocyte membrane

1 reference

12 December 2020

Pentobarbital: stereospecific actions of (+) and (-) isomers revealed on cultured mammalian neurons

1 reference

12 December 2020

Identifiers

DOI

10.1038/SJ.BJP.0702744

1 reference

6 August 2017

1 reference

6 August 2017

1 reference