(Q35181936)

7 August 2017

title

Bodilisant-a novel fluorescent, highly affine histamine h3 receptor ligand (English)

1 reference

7 August 2017

Miriam Tomasch

1

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7 August 2017

J Stephan Schwed

series ordinal

2

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7 August 2017

Alexander Paulke

series ordinal

3

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7 August 2017

Holger Stark

series ordinal

4

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7 August 2017

publication date

12 December 2012

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ACS Medicinal Chemistry Letters

7 August 2017

published in

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7 August 2017

volume

4

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7 August 2017

issue

2

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7 August 2017

page(s)

269-273

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Novel chalcone-based fluorescent human histamine h(3) receptor ligands as pharmacological tools

7 August 2017

cites work

1 reference

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A novel fluorescent histamine H(1) receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands

13 July 2018

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Search for novel, high affinity histamine H3 receptor ligands with fluorescent properties

13 July 2018

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Histamine H3 receptor antagonists go to clinics

13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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The CD11a binding site of efalizumab in psoriatic skin tissue as analyzed by Multi-Epitope Ligand Cartography robot technology. Introduction of a novel biological drug-binding biochip assay

13 July 2018

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BODIPY-conjugated neuropeptide Y ligands: new fluorescent tools to tag Y1, Y2, Y4 and Y5 receptor subtypes

13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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Pharmacology and direct visualisation of BODIPY-TMR-CGP: a long-acting fluorescent beta2-adrenoceptor agonist

13 July 2018

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Immunological identification of the mammalian H3 histamine receptor in the mouse brain

13 July 2018

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Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

13 July 2018

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Characterization of novel fluorescent ligands with high affinity for D1 and D2 dopaminergic receptors

13 July 2018

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Three histamine receptors (H1, H2 and H3) visualized in the brain of human and non-human primates.

13 July 2018

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

13 July 2018

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Novel fluorescent probe for analysis of hydroperoxides based on boron dipyrromethane fluorophore.

13 July 2018

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Generation and characterisation of the first anti-human H3R445/453 isoform specific antibody probe

27 September 2018

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Immunolocalization of histamine H3 receptors on endocrine cells in the rat gastrointestinal tract

27 September 2018

1 reference

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Fluorescent non-imidazole histamine H3 receptor ligands with nanomolar affinities

27 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4027500

Search for histamine H3 receptor antagonists with combined inhibitory potency at Ntau-methyltransferase: ether derivatives.

27 September 2018

1 reference

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Application of fluorescence correlation spectroscopy to the measurement of agonist binding to a G-protein coupled receptor at the single cell level

27 September 2018

1 reference

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Fluorescence quantum yields and their relation to lifetimes of rhodamine 6G and fluorescein in nine solvents: improved absolute standards for quantum yields

27 September 2018

1 reference

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Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine

27 September 2018

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12 December 2020

Highly potent fluorescence-tagged nonimidazole histamine H3 receptor ligands

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12 December 2020

GPCR targeted library design: novel dopamine D3 receptor ligands

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12 December 2020

Histamine H1, H3 and H4 receptors are involved in pruritus

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12 December 2020

Receptor-specific functional efficacies of alkyl imidazoles as dual histamine H3/H4 receptor ligands

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12 December 2020

Identifiers

DOI

10.1021/ML300383N

1 reference

7 August 2017

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7 August 2017

1 reference