(Q35714170)

English

5-aminomethyloxazolidine-2,4-dione hybrid α/β-dipeptide scaffolds as inductors of constrained conformations: Applications to the synthesis of integrin antagonists

scientific article published on 25 July 2015

In more languages

Statements

scholarly article

1 reference

Europe PubMed Central

9 August 2017

5-aminomethyloxazolidine-2,4-dione hybrid α/β-dipeptide scaffolds as inductors of constrained conformations: Applications to the synthesis of integrin antagonists (English)

1 reference

Europe PubMed Central

9 August 2017

object named as

Monica Baiula

4

0 references

Santi Spampinato

object named as

Santi Spampinato

5

0 references

author name string

Rossella De Marco

1

1 reference

Europe PubMed Central

9 August 2017

Giacomo Mazzotti

2

1 reference

Europe PubMed Central

9 August 2017

Samantha D Dattoli

3

1 reference

Europe PubMed Central

9 August 2017

Arianna Greco

6

1 reference

Europe PubMed Central

9 August 2017

Luca Gentilucci

7

1 reference

Europe PubMed Central

9 August 2017

publication date

25 July 2015

1 reference

Europe PubMed Central

9 August 2017

1 reference

Europe PubMed Central

9 August 2017

104

1 reference

Europe PubMed Central

9 August 2017

636-649

1 reference

Europe PubMed Central

9 August 2017

5

1 reference

Europe PubMed Central

9 August 2017

Peptides and proteins as a continuing exciting source of inspiration for peptidomimetics

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Natural and artificial peptide motifs: their origins and the application of motif-programming

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Tripeptide motifs in biology: targets for peptidomimetic design.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Synthesis of tripeptides containing D-Trp substituted at the indole ring, assessment of opioid receptor binding and in vivo central antinociception

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Opioid activity profiles of oversimplified peptides lacking in the protonable N-terminus

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Peptides and peptidomimetics in medicine, surgery and biotechnology

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Chemical modifications designed to improve peptide stability: incorporation of non-natural amino acids, pseudo-peptide bonds, and cyclization

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Azapeptides and their therapeutic potential.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Efficient method for the preparation of peptoids [oligo(N-substituted glycines)] by submonomer solid-phase synthesis

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

The partial retro-inverso modification: a road traveled together

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Conformational and topographical considerations in designing agonist peptidomimetics from peptide leads

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Protein design with L- and D-alpha-amino acid structures as the alphabet

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Structures of peptides from alpha-amino acids methylated at the alpha-carbon.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Control of peptide conformation by the Thorpe-Ingold effect (C alpha-tetrasubstitution).

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

β-Peptides: Synthesis by Arndt-Eistert homologation with concomitant peptide coupling. Structure determination by NMR and CD spectroscopy and by X-ray crystallography. Helical secondary structure of a β-hexapeptide in solution and its stability tow

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

The world of beta- and gamma-peptides comprised of homologated proteinogenic amino acids and other components

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

β-Peptide Foldamers: Robust Helix Formation in a New Family of β-Amino Acid Oligomers

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

beta-Peptides: from structure to function

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Foldamers as versatile frameworks for the design and evolution of function

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Synthesis and conformational analysis of a cyclic peptide obtained via i to i+4 intramolecular side-chain to side-chain azide-alkyne 1,3-dipolar cycloaddition

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Activation of apoptosis in vivo by a hydrocarbon-stapled BH3 helix

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Synthesis and conformational studies of peptidomimetics containing a new bifunctional diketopiperazine scaffold acting as a beta-hairpin inducer.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Beta2-amino acids-syntheses, occurrence in natural products, and components of beta-peptides1,2.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Integrin modulation and signaling in leukocyte adhesion and migration

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Therapeutic anti-integrin (alpha4 and alphaL) monoclonal antibodies: two-edged swords?

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Monoclonal antibodies in the treatment of neuroimmunological diseases

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Alpha 4 integrin antagonists

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

VLA-4 antagonists: potent inhibitors of lymphocyte migration

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Rational design of potent and selective VLA-4 inhibitors and their utility in the treatment of asthma

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Selective, tight-binding inhibitors of integrin alpha4beta1 that inhibit allergic airway responses

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Identification of potent and novel alpha4beta1 antagonists using in silico screening

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Effect of enalapril on the in vitro and in vivo peptidyl cleavage of a potent VLA-4 antagonist.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

LC/MS/MS plasma assay for the peptidomimetic VLA4 antagonist I and its major active metabolite II: for treatment of asthma by inhalation

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Synthesis and binding activity of endomorphin-1 analogues containing beta-amino acids.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Endomorphin-1 analogues containing beta-proline are mu-opioid receptor agonists and display enhanced enzymatic hydrolysis resistance

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

A straightforward route to enantiopure 2-substituted-3,4-dehydro-β-proline via ring closing metathesis

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Antinociception by a peripherally administered novel endomorphin-1 analogue containing beta-proline

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Stability against enzymatic hydrolysis of endomorphin-1 analogues containing beta-proline

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Development of isoxazoline-containing peptidomimetics as dual αvβ3 and α5β1 integrin ligands

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Modulation of αvβ₃- and α₅β₁-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Targeting integrins αvβ3 and α5β1 with new β-lactam derivatives

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Synthesis and assay of retro-α4β1 integrin-targeting motifs.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Synthesis and conformational analysis of cyclotetrapeptide mimetic beta-turn templates and validation as 3D scaffolds

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Antiangiogenic effect of dual/selective alpha(5)beta(1)/alpha(v)beta(3) integrin antagonists designed on partially modified retro-inverso cyclotetrapeptide mimetics

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Discovery of potent and selective thienopyrimidine inhibitors of Aurora kinases.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

3D QSAR (COMFA) of a series of potent and highly selective VLA-4 antagonists

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Novel C2-C3' N-peptide linked macrocyclic taxoids. Part 2: synthesis and biological activities of docetaxel analogues with a peptide side chain at C2 and their macrocyclic derivatives

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Peripheral antinociceptive effects of the cyclic endomorphin-1 analog c[YpwFG] in a mouse visceral pain model

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

A 3D structure model of integrin alpha 4 beta 1 complex: I. Construction of a homology model of beta 1 and ligand binding analysis

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Insights into phenylalanine derivatives recognition of VLA-4 integrin: from a pharmacophoric study to 3D-QSAR and molecular docking analyses

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Conformational analysis of an opioid peptide in solvent media that mimic cytoplasm viscosity

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Natural peptide analgesics: the role of solution conformation

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Structural comparison of mu-opioid receptor selective peptides confirmed four parameters of bioactivity

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Comparison of simple potential functions for simulating liquid water

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

A Second Generation Force Field for the Simulation of Proteins, Nucleic Acids, and Organic Molecules

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Contribution of alpha4beta1 integrin to the antiallergic effect of levocabastine.

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Solution conformation of proteinase inhibitor IIA from bull seminal plasma by 1H nuclear magnetic resonance and distance geometry

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Application of Ring-Closing Metathesis to the Synthesis of Rigidified Amino Acids and Peptides

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Expedient synthesis of pseudo-Pro-containing peptides: towards constrained peptidomimetics and foldamers

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Synthesis and analysis of the conformational preferences of 5-aminomethyloxazolidine-2,4-dione scaffolds: first examples of β(2)- and β(2, 2)-homo-Freidinger lactam analogues

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

EC3, a Novel Heterodimeric Disintegrin fromEchis carinatusVenom, Inhibits α4 and α5 Integrins in an RGD-independent Manner

1 reference

https://api.crossref.org/works/10.1002%2FBIP.22704

21 January 2018

Identifiers

10.1002/BIP.22704

1 reference

Europe PubMed Central

9 August 2017

1 reference

Europe PubMed Central

9 August 2017

Sitelinks

Wikipedia(0 entries)

Wikibooks(0 entries)

Wikinews(0 entries)

Wikiquote(0 entries)

Wikisource(0 entries)

Wikiversity(0 entries)

Wikivoyage(0 entries)

Wiktionary(0 entries)

Multilingual sites(0 entries)

Retrieved from "https://www.wikidata.org/w/index.php?title=Q35714170&oldid=1584283496"