(Q36208408)

12 August 2017

Molecular probes for muscarinic receptors: derivatives of the M1-antagonist telenzepine (English)

1 reference

12 August 2017

Y Karton

1

1 reference

12 August 2017

J Baumgold

series ordinal

2

1 reference

12 August 2017

J S Handen

series ordinal

3

1 reference

12 August 2017

K A Jacobson

series ordinal

4

1 reference

12 August 2017

1 May 1992

1 reference

12 August 2017

Bioconjugate Chemistry

1 reference

12 August 2017

3

1 reference

12 August 2017

3

1 reference

12 August 2017

234-240

1 reference

Oligomeric structure of muscarinic receptors is shown by photoaffinity labeling: subunit assembly may explain high- and low-affinity agonist states

12 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Cloning and expression of the human and rat m5 muscarinic acetylcholine receptor genes

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Identification of a family of muscarinic acetylcholine receptor genes

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Molecular probes for extracellular adenosine receptors

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Demonstration of distinct agonist and antagonist conformations of the A1 adenosine receptor

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Structure-function relationships in nicotinic acetylcholine receptors

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Functionalized congener approach to muscarinic antagonists: analogues of pirenzepine

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Trifunctional agents as a design strategy for tailoring ligand properties: irreversible inhibitors of A1 adenosine receptors

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Model systems for the study of seven-transmembrane-segment receptors

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Affinity chromatography of the muscarinic acetylcholine receptor.

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

The labelling of proteins to high specific radioactivities by conjugation to a 125I-containing acylating agent. Application to the radioimmunoassay

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Photoaffinity labeling of the human erythrocyte monosaccharide transporter with an aryl azide derivative of D-glucose.

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Pharmacological evidence for selective inhibition of gastric acid secretion by telenzepine, a new antimuscarinic drug

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Site-directed mutagenesis of m1 muscarinic acetylcholine receptors: conserved aspartic acids play important roles in receptor function

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

The affinity, selectivity and biological activity of telenzepine enantiomers

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Photosensitized labeling of a functional multidrug transporter in living drug-resistant tumor cells.

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3433723

Characterization of benzodiazepine receptors with fluorescent ligands

29 June 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/1520727

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Propylbenzilylcholine mustard labels an acidic residue in transmembrane helix 3 of the muscarinic receptor

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/1520727

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Differential regulation of PI hydrolysis and adenylyl cyclase by muscarinic receptor subtypes

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/1520727

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/BC00015A006

1 reference

12 August 2017

1 reference

12 August 2017

PubMed publication ID

1520727

1 reference