(Q36216496)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

title

Structure-based virtual screening and identification of a novel androgen receptor antagonist (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

1 reference

6

1 reference

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8 February 2020

author name string

Chin-Hee Song

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

Su Hui Yang

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

Eunsook Park

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

Suk Hee Cho

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

Eun-Yeung Gong

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

Won-Jea Cho

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

Keesook Lee

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

language of work or name

English

0 references

publication date

13 July 2012

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

Journal of Biological Chemistry

8 February 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

volume

287

1 reference

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8 February 2020

issue

36

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

page(s)

30769-30780

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

MAP Kinases and Prostate Cancer

8 February 2020

cites work

1 reference

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Inhibitors of androgen receptor activation function-2 (AF2) site identified through virtual screening

1 October 2017

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Mechanism of androgen receptor antagonism by bicalutamide in the treatment of prostate cancer

1 October 2017

1 reference

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Biological properties of androgen receptor pure antagonist for treatment of castration-resistant prostate cancer: optimization from lead compound to CH5137291.

1 October 2017

1 reference

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Resveratrol regulates the PTEN/AKT pathway through androgen receptor-dependent and -independent mechanisms in prostate cancer cell lines

1 October 2017

1 reference

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Regression of castrate-recurrent prostate cancer by a small-molecule inhibitor of the amino-terminus domain of the androgen receptor

1 October 2017

1 reference

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Limitations of MTT and MTS-based assays for measurement of antiproliferative activity of green tea polyphenols

1 October 2017

1 reference

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Structure-activity relationship for thiohydantoin androgen receptor antagonists for castration-resistant prostate cancer (CRPC)

1 October 2017

1 reference

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HDAC6 regulates androgen receptor hypersensitivity and nuclear localization via modulating Hsp90 acetylation in castration-resistant prostate cancer

1 October 2017

1 reference

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Androgen receptor regulates a distinct transcription program in androgen-independent prostate cancer

1 October 2017

1 reference

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Nonsteroidal selective androgen receptor modulators (SARMs): dissociating the anabolic and androgenic activities of the androgen receptor for therapeutic benefit

1 October 2017

1 reference

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Development of a second-generation antiandrogen for treatment of advanced prostate cancer

1 October 2017

1 reference

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Regulation of androgen receptor transcriptional activity by rapamycin in prostate cancer cell proliferation and survival

1 October 2017

1 reference

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Computationally identified novel diphenyl- and phenylpyridine androgen receptor antagonist structures

1 October 2017

1 reference

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1 October 2017

Cancer statistics, 2008

1 reference

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CR6-interacting factor 1 represses the transactivation of androgen receptor by direct interaction.

1 October 2017

1 reference

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Crystal Structure of the T877A Human Androgen Receptor Ligand-binding Domain Complexed to Cyproterone Acetate Provides Insight for Ligand-induced Conformational Changes and Structure-based Drug Design

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Evaluation of an in vitro model of androgen ablation and identification of the androgen responsive proteome in LNCaP cells

1 October 2017

1 reference

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Antiandrogens in the treatment of prostate cancer

1 October 2017

1 reference

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Pharmacokinetics and pharmacodynamics of nonsteroidal androgen receptor ligands

1 October 2017

1 reference

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Targeting the androgen receptor in hormone-refractory prostate cancer--new concepts

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

The CCAAT enhancer-binding protein-alpha negatively regulates the transactivation of androgen receptor in prostate cancer cells

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

The corepressors silencing mediator of retinoid and thyroid hormone receptor and nuclear receptor corepressor are involved in agonist- and antagonist-regulated transcription by androgen receptor

1 October 2017

1 reference

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Structural basis for accommodation of nonsteroidal ligands in the androgen receptor

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Modulation of the expression and transactivation of androgen receptor by the basic helix-loop-helix transcription factor Pod-1 through recruitment of histone deacetylase 1

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Structural basis for antagonism and resistance of bicalutamide in prostate cancer

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Signal transduction pathways in androgen-dependent and -independent prostate cancer cell proliferation

1 October 2017

1 reference

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Global cancer statistics, 2002

1 October 2017

1 reference

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Targeting prostate cancer with conditionally replicative adenovirus using PSMA enhancer

1 October 2017

1 reference

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Androgen deprivation therapy for prostate cancer: current status and future prospects

1 October 2017

1 reference

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Prostate specific antigen gene regulation by androgen receptor

1 October 2017

1 reference

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Androgen receptor in prostate cancer

1 October 2017

1 reference

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Androgen receptor coregulators in prostate cancer: mechanisms and clinical implications.

1 October 2017

1 reference

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Molecular determinants of resistance to antiandrogen therapy

1 October 2017

1 reference

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Ras signaling in prostate cancer progression

1 October 2017

1 reference

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PTEN: one gene, many syndromes

1 October 2017

1 reference

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Expression of MIS in the testis is downregulated by tumor necrosis factor alpha through the negative regulation of SF-1 transactivation by NF-kappa B.

1 October 2017

1 reference

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Androgen receptor gene amplification and protein expression in hormone refractory prostate cancer.

1 October 2017

1 reference

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The role of antiandrogen monotherapy in the treatment of prostate cancer

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Evidence that chlormadinone acetate exhibits antiandrogenic activity in androgen-dependent cell line

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Novel mutations of androgen receptor: a possible mechanism of bicalutamide withdrawal syndrome.

1 October 2017

1 reference

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Mechanism of antiandrogen action: key role of hsp90 in conformational change and transcriptional activity of the androgen receptor

1 October 2017

1 reference

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The program of androgen-responsive genes in neoplastic prostate epithelium

1 October 2017

1 reference

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Phosphatidylinositol 3-kinase/Akt stimulates androgen pathway through GSK3beta inhibition and nuclear beta-catenin accumulation

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Bicalutamide functions as an androgen receptor antagonist by assembly of a transcriptionally inactive receptor

1 October 2017

1 reference

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Androgen receptor expression is regulated by the phosphoinositide 3-kinase/Akt pathway in normal and tumoral epithelial cells

1 October 2017

1 reference

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Androgen receptor (AR) coregulators: an overview

1 October 2017

1 reference

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The development of androgen-independent prostate cancer

1 October 2017

1 reference

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Akt suppresses androgen-induced apoptosis by phosphorylating and inhibiting androgen receptor

1 October 2017

1 reference

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From transforming growth factor-beta signaling to androgen action: identification of Smad3 as an androgen receptor coregulator in prostate cancer cells

1 October 2017

1 reference

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Pregnenolone stimulates LNCaP prostate cancer cell growth via the mutated androgen receptor.

1 October 2017

1 reference

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HER-2/neu promotes androgen-independent survival and growth of prostate cancer cells through the Akt pathway.

1 October 2017

1 reference

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LNCaP progression model of human prostate cancer: androgen-independence and osseous metastasis

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Structural evidence for ligand specificity in the binding domain of the human androgen receptor. Implications for pathogenic gene mutations

1 October 2017

1 reference

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Antiandrogens in prostate cancer

1 October 2017

1 reference

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A nuclear factor, ASC-2, as a cancer-amplified transcriptional coactivator essential for ligand-dependent transactivation by nuclear receptors in vivo

1 October 2017

1 reference

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Mechanistic concepts in androgen-dependence of prostate cancer

1 October 2017

1 reference

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Selection for androgen receptor mutations in prostate cancers treated with androgen antagonist

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

From HER2/Neu signal cascade to androgen receptor and its coactivators: a novel pathway by induction of androgen target genes through MAP kinase in prostate cancer cells

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Distinguishing androgen receptor agonists and antagonists: distinct mechanisms of activation by medroxyprogesterone acetate and dihydrotestosterone

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Molecular action of androgen in the normal and neoplastic prostate

1 October 2017

2 references

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1 October 2017

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Androgen receptor expression in androgen-independent prostate cancer is associated with increased expression of androgen-regulated genes

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Promotion of agonist activity of antiandrogens by the androgen receptor coactivator, ARA70, in human prostate cancer DU145 cells

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

From estrogen to androgen receptor: a new pathway for sex hormones in prostate

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Inactivation of the tumor suppressor PTEN/MMAC1 in advanced human prostate cancer through loss of expression

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

GRIP1, a transcriptional coactivator for the AF-2 transactivation domain of steroid, thyroid, retinoid, and vitamin D receptors

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

In vivo amplification of the androgen receptor gene and progression of human prostate cancer

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Synthesis and biological activity of novel nonsteroidal progesterone receptor antagonists

1 October 2017

1 reference

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Hormone-refractory (D3) prostate cancer: refining the concept.

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Androgen receptor activation in prostatic tumor cell lines by insulin-like growth factor-I, keratinocyte growth factor, and epidermal growth factor

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Sequence and characterization of a coactivator for the steroid hormone receptor superfamily

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Comparison of the antiandrogenic/androgenic activities of flutamide, cyproterone acetate and megestrol acetate

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Domains of the Human Androgen Receptor Involved in Steroid Binding, Transcriptional Activation, and Subcellular Localization

1 October 2017

1 reference

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Anti-androgens and the mutated androgen receptor of LNCaP cells: differential effects on binding affinity, heat-shock protein interaction, and transcription activation

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Mutant androgen receptor detected in an advanced-stage prostatic carcinoma is activated by adrenal androgens and progesterone

1 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

A mutation in the ligand binding domain of the androgen receptor of human LNCaP cells affects steroid binding characteristics and response to anti-androgens

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Comparative effects of bicalutamide (Casodex) versus orchidectomy on bone mineral density, bone remodelling, and bone biomechanics in healthy rats

29 June 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

N-Arylpiperazine-1-carboxamide derivatives: a novel series of orally active nonsteroidal androgen receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

(+)-(2R,5S)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3- yl]piperazine-1-carboxamide (YM580) as an orally potent and peripherally selective nonsteroidal androgen receptor antagonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Antiandrogenic effects of bisphenol A and nonylphenol on the function of androgen receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Preclinical pharmacology of a nonsteroidal ligand for androgen receptor-mediated imaging of prostate cancer.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Reduced testicular steroidogenesis in tumor necrosis factor-alpha knockout mice

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Androgen Receptor (AR) Coregulators: An Overview

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Stabilization of androgen receptor protein is induced by agonist, not by antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Androgen receptor mutations in androgen-independent prostate cancer: Cancer and Leukemia Group B Study 9663.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Antiandrogen bicalutamide promotes tumor growth in a novel androgen-dependent prostate cancer xenograft model derived from a bicalutamide-treated patient

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Structure based approach to the design of bicyclic-1H-isoindole-1,3(2H)-dione based androgen receptor antagonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Switch from antagonist to agonist of the androgen receptor bicalutamide is associated with prostate tumour progression in a new model system

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

AKT regulates androgen receptor-dependent growth and PSA expression in prostate cancer

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

A mechanism for androgen receptor-mediated prostate cancer recurrence after androgen deprivation therapy

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3436320

Current Thoughts on the Role of the Androgen Receptor and Prostate Cancer Progression

22 September 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M112.379107

Suberoylanilide hydroxamic acid, an inhibitor of histone deacetylase, suppresses the growth of prostate cancer cells in vitro and in vivo

21 January 2018

1 reference

12 December 2020

Activating signal cointegrator 1 is highly expressed in murine testicular Leydig cells and enhances the ligand-dependent transactivation of androgen receptor

1 reference

12 December 2020

Intermolecular NH2-/carboxyl-terminal interactions in androgen receptor dimerization revealed by mutations that cause androgen insensitivity

1 reference

12 December 2020

Aberrant response in vitro of hormone-responsive prostate cancer cells to antiandrogens

1 reference

12 December 2020

A novel synthetic compound that interrupts androgen receptor signaling in human prostate cancer cells

1 reference

12 December 2020

Hepatocyte nuclear factor-3 alpha (HNF-3alpha) negatively regulates androgen receptor transactivation in prostate cancer cells

1 reference

12 December 2020

Dehydroepiandrosterone activates mutant androgen receptors expressed in the androgen-dependent human prostate cancer xenograft CWR22 and LNCaP cells

1 reference

12 December 2020

Identifiers

DOI

10.1074/JBC.M112.379107

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22798067%20AND%20SRC:MED&resulttype=core&format=json

8 February 2020

1 reference