(Q36276693)

English

Structure-activity relationships and pharmacophore model of a noncompetitive pyrazoline containing class of GluN2C/GluN2D selective antagonists

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Structure-activity relationships and pharmacophore model of a noncompetitive pyrazoline containing class of GluN2C/GluN2D selective antagonists (English)

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Cathryn Slabber

object named as

Cathryn Slabber

4

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Dennis C. Liotta

8

object named as

Dennis C Liotta

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

2

object named as

Alpa Khatri

1 reference

Europe PubMed Central

13 August 2017

PMC publication ID

5

object named as

John Bacsa

1 reference

Europe PubMed Central

13 August 2017

PMC publication ID

Timothy M Acker

1

object named as

Timothy M Acker

1 reference

Europe PubMed Central

13 August 2017

PMC publication ID

author name string

Katie M Vance

3

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

James P Snyder

6

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Stephen F Traynelis

7

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Europe PubMed Central

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13 August 2017

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publication date

2 August 2013

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Europe PubMed Central

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13 August 2017

Journal of Medicinal Chemistry

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Europe PubMed Central

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13 August 2017

56

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Europe PubMed Central

PMC publication ID

13 August 2017

16

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

6434-6456

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

Synthesis and structure activity relationship of tetrahydroisoquinoline-based potentiators of GluN2C and GluN2D containing N-methyl-D-aspartate receptors

1 reference

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30 September 2017

Mechanism for noncompetitive inhibition by novel GluN2C/D N-methyl-D-aspartate receptor subunit-selective modulators

1 reference

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30 September 2017

Intrinsic dynamics and synaptic inputs control the activity patterns of subthalamic nucleus neurons in health and in Parkinson's disease

1 reference

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30 September 2017

Functional NMDA receptors at axonal growth cones of young hippocampal neurons

1 reference

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30 September 2017

Ligand-specific deactivation time course of GluN1/GluN2D NMDA receptors

1 reference

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30 September 2017

Halogen bonding in halocarbon-protein complexes: a structural survey.

1 reference

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Behavioral analysis of NR2C knockout mouse reveals deficit in acquisition of conditioned fear and working memory

1 reference

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30 September 2017

Systematic investigation of halogen bonding in protein-ligand interactions

1 reference

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30 September 2017

Glutamate receptor ion channels: structure, regulation, and function

1 reference

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30 September 2017

Quinazolin-4-one derivatives: A novel class of noncompetitive NR2C/D subunit-selective N-methyl-D-aspartate receptor antagonists

1 reference

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30 September 2017

Structural determinants of D-cycloserine efficacy at the NR1/NR2C NMDA receptors

1 reference

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30 September 2017

Control of NMDA receptor function by the NR2 subunit amino-terminal domain

1 reference

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30 September 2017

Allosteric modulators of NR2B-containing NMDA receptors: molecular mechanisms and therapeutic potential

1 reference

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30 September 2017

Mechanism of differential control of NMDA receptor activity by NR2 subunits

1 reference

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30 September 2017

Once-weekly D-cycloserine effects on negative symptoms and cognition in schizophrenia: an exploratory study

1 reference

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30 September 2017

Pathophysiology of parkinsonism

1 reference

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Circuit-based framework for understanding neurotransmitter and risk gene interactions in schizophrenia

1 reference

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A short history of SHELX

1 reference

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30 September 2017

Structure-brain exposure relationships

1 reference

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30 September 2017

NMDA receptor subunits: function and pharmacology.

1 reference

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30 September 2017

The chemical biology of clinically tolerated NMDA receptor antagonists

1 reference

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30 September 2017

NMDA receptor NR2 subunit dependence of the slow component of magnesium unblock.

1 reference

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30 September 2017

Pharmacological insights obtained from structure-function studies of ionotropic glutamate receptors

1 reference

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30 September 2017

Subunit arrangement and function in NMDA receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4643674

30 September 2017

Glutamate receptor ion channels

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4643674

30 September 2017

Autonomous pacemakers in the basal ganglia: who needs excitatory synapses anyway?

1 reference

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30 September 2017

Homeostatic plasticity and NMDA receptor trafficking

1 reference

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30 September 2017

Evaluation of the MDR-MDCK cell line as a permeability screen for the blood-brain barrier.

1 reference

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30 September 2017

Role of distinct NMDA receptor subtypes at central synapses

1 reference

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30 September 2017

Rationale for and use of NMDA receptor antagonists in Parkinson's disease.

1 reference

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Mechanisms of activation, inhibition and specificity: crystal structures of the NMDA receptor NR1 ligand-binding core

1 reference

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Synaptic organisation of the basal ganglia

1 reference

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Ligands for glutamate receptors: design and therapeutic prospects

1 reference

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Cloned glutamate receptors

1 reference

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Organization of N-methyl-D-aspartate glutamate receptor gene expression in the basal ganglia of the rat.

1 reference

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Developmental and regional expression in the rat brain and functional properties of four NMDA receptors

1 reference

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Voltage-dependent block by Mg2+ of NMDA responses in spinal cord neurones

1 reference

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Magnesium gates glutamate-activated channels in mouse central neurones

1 reference

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Cloning of an apparent splice variant of the rat N-methyl-D-aspartate receptor NMDAR1 with altered sensitivity to polyamines and activators of protein kinase C

1 reference

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1 reference

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30 September 2017

A subunit-selective potentiator of NR2C- and NR2D-containing NMDA receptors.

1 reference

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29 June 2018

Models of basal ganglia function and pathophysiology of movement disorders.

1 reference

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29 June 2018

Alternatively spliced isoforms of the NMDAR1 glutamate receptor subunit: differential expression in the basal ganglia of the rat.

1 reference

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29 June 2018

Channel kinetics determine the time course of NMDA receptor-mediated synaptic currents.

1 reference

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29 June 2018

Structural and mechanistic determinants of a novel site for noncompetitive inhibition of GluN2D-containing NMDA receptors

1 reference

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22 September 2018

Facile nucleophilic fluorination reactions using tert-alcohols as a reaction medium: significantly enhanced reactivity of alkali metal fluorides and improved selectivity

1 reference

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22 September 2018

Regional and developmental heterogeneity in splicing of the rat brain NMDAR1 mRNA.

1 reference

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22 September 2018

Differential expression of five N-methyl-D-aspartate receptor subunit mRNAs in the cerebellum of developing and adult rats.

1 reference

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22 September 2018

Identifiers

10.1021/JM400652R

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

ResearchGate publication ID

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