(Q36339669)

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Thiadiazolidinones: a new class of alanine racemase inhibitors with antimicrobial activity against methicillin-resistant Staphylococcus aureus

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Europe PubMed Central

PMC publication ID

13 August 2017

Thiadiazolidinones: a new class of alanine racemase inhibitors with antimicrobial activity against methicillin-resistant Staphylococcus aureus (English)

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

methicillin-resistant Staphylococcus aureus

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1 reference

based on heuristic

inferred from title

Staphylococcus aureus

1 reference

based on heuristic

inferred from title

Adriana E. Rosato

3

object named as

Adriana E Rosato

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

7

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Michel Ledizet

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author name string

Mihai Ciustea

1

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Europe PubMed Central

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13 August 2017

Sara Mootien

2

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Europe PubMed Central

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13 August 2017

Oriana Perez

4

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Europe PubMed Central

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13 August 2017

Pier Cirillo

5

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Europe PubMed Central

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13 August 2017

Kacheong R Yeung

6

1 reference

Europe PubMed Central

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13 August 2017

Michael H Cynamon

8

1 reference

Europe PubMed Central

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13 August 2017

Paul A Aristoff

9

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Europe PubMed Central

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13 August 2017

Raymond A Koski

10

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Europe PubMed Central

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13 August 2017

Paul A Kaplan

11

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Europe PubMed Central

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13 August 2017

Karen G Anthony

12

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13 August 2017

language of work or name

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publication date

29 November 2011

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13 August 2017

Biochemical Pharmacology

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13 August 2017

83

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Europe PubMed Central

PMC publication ID

13 August 2017

3

1 reference

Europe PubMed Central

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13 August 2017

368-377

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Europe PubMed Central

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13 August 2017

New classes of alanine racemase inhibitors identified by high-throughput screening show antimicrobial activity against Mycobacterium tuberculosis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Vancomycin-resistant Staphylococcus aureus, Michigan, USA, 2007.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Structural and Kinetic Analyses of Macrophage Migration Inhibitory Factor Active Site Interactions † ‡

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Teichoic acids and related cell-wall glycopolymers in Gram-positive physiology and host interactions.

1 reference

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30 September 2017

Inhibitors of Helicobacter pylori ATPase Cagalpha block CagA transport and cag virulence

1 reference

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30 September 2017

Reaction specificity in pyridoxal phosphate enzymes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Functional characterization of alanine racemase from Schizosaccharomyces pombe: a eucaryotic counterpart to bacterial alanine racemase

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Structure of a Michaelis complex analogue: propionate binds in the substrate carboxylate site of alanine racemase

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Staphylococcus aureus infections

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Inhibition of cell wall biosynthesis by analogues and alanine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Enzymes in the D-alanine branch of bacterial cell wall peptidoglycan assembly

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

30 September 2017

Inactivation of the dadB Salmonella typhimurium alanine racemase by D and L isomers of beta-substituted alanines: kinetics, stoichiometry, active site peptide sequencing, and reaction mechanism

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

29 June 2018

1-Aminocyclopropanephosphonate: time-dependent inactivation of 1-aminocyclopropanecarboxylate deaminase and Bacillus stearothermophilus alanine racemase by slow dissociation behavior.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

29 June 2018

Biosynthetic alanine racemase of Salmonella typhimurium: purification and characterization of the enzyme encoded by the alr gene

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

29 June 2018

Inhibition of alanine racemase by alanine phosphonate: detection of an imine linkage to pyridoxal 5'-phosphate in the enzyme-inhibitor complex by solid-state 15N nuclear magnetic resonance

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

29 June 2018

Mechanism of inhibition of fatty acid amide hydrolase by sulfonamide-containing benzothiazoles: long residence time derived from increased kinetic barrier and not exclusively from thermodynamic potency

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

Fate of mutation rate depends on agr locus expression during oxacillin-mediated heterogeneous-homogeneous selection in methicillin-resistant Staphylococcus aureus clinical strains

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

Use of NMR metabolomics to analyze the targets of D-cycloserine in mycobacteria: role of D-alanine racemase

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

Fifteen-year study of the changing epidemiology of methicillin-resistant Staphylococcus aureus.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

SAR and 3D-QSAR studies on thiadiazolidinone derivatives: exploration of structural requirements for glycogen synthase kinase 3 inhibitors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

N(2)-substituted D,L-cycloserine derivatives: synthesis and evaluation as alanine racemase inhibitors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

A eukaryotic alanine racemase gene involved in cyclic peptide biosynthesis

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

Teichoic acid content in different lineages of Staphylococcus aureus NCTC8325.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

Purification and characterization of eucaryotic alanine racemase acting as key enzyme in cyclosporin biosynthesis.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3478562

22 September 2018

Improved method for electroporation of Staphylococcus aureus

1 reference

https://pubmed.ncbi.nlm.nih.gov/22146584

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Selective inhibition of bacterial dihydroorotate dehydrogenases by thiadiazolidinediones

1 reference

https://pubmed.ncbi.nlm.nih.gov/22146584

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Properties of a cryptic high-frequency transducing phage in Staphylococcus aureus

1 reference

https://pubmed.ncbi.nlm.nih.gov/22146584

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.BCP.2011.11.021

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

ResearchGate publication ID

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