(Q36343185)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

title

Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

author name string

K A Jacobson

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

L Kiriasis

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

S Barone

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

B J Bradbury

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

U Kammula

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

J M Campagne

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

S Secunda

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

J W Daly

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

W Pfleiderer

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

language of work or name

English

0 references

publication date

1 August 1989

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

Journal of Medicinal Chemistry

4 October 2019

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

volume

32

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

issue

8

1 reference

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4 October 2019

page(s)

1873-1879

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

Adenosine receptor binding: structure-activity analysis generates extremely potent xanthine antagonists

4 October 2019

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Xanthine functionalized congeners as potent ligands at A2-adenosine receptors

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

A new high affinity, iodinated adenosine receptor antagonist as a radioligand/photoaffinity crosslinking probe

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Iodine-125-labeled 8-phenylxanthine derivatives: antagonist radioligands for adenosine A1 receptors

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors.

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

[3H]xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

A functionalized congener approach to adenosine receptor antagonists: amino acid conjugates of 1,3-dipropylxanthine

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Functionalized congeners of 1,3-dialkylxanthines: preparation of analogues with high affinity for adenosine receptors

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Non-xanthine heterocycles: activity as antagonists of A1- and A2-adenosine receptors

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Evidence that a novel 8-phenyl-substituted xanthine derivative is a cardioselective adenosine receptor antagonist in vivo

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Two distinct adenosine-sensitive sites on adenylate cyclase

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

The Synthesis and Pharmacologic Evaluation of a Series of 8-Alkylthio-Thiated Theophyllines1

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

PD 115,199: an antagonist ligand for adenosine A2 receptors

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

8-Aryl-and 8-cycloalkyl-1,3-dipropylxanthines: further potent and selective antagonists for A1-adenosine receptors

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

New methylxanthine thio-derivatives inducing marked tracheal relaxation without increasing cardiac inotropism or motor activity

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Characterization of the A2 adenosine receptor labeled by [3H]NECA in rat striatal membranes

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

A caffeine analogue (1,3,7-trimethyl-6-thioxo-2-oxopurine) with a negative inotropic and chronotropic effect

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Alkylxanthines as adenosine receptor antagonists and membrane phosphodiesterase inhibitors in central nervous tissue: Evaluation of structure-activity relationships

29 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3479653

Characterization of adenosine receptors in rat brain by (?)[3H]N6-phenylisopropyladenosine

22 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/2754711

12 December 2020

inferred from PubMed ID database lookup

Adenosine antagonism by purines, pteridines and benzopteridines in human fibroblasts

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/2754711

12 December 2020

inferred from PubMed ID database lookup

The adenosine receptor antagonist, 8-phenyltheophylline, causes diuresis and saliuresis in the rat

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/2754711

12 December 2020

inferred from PubMed ID database lookup

Identifiers

DOI

10.1021/JM00128A031

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

release_jaslaryugfasbpksasgft6vy4u

4 October 2019

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/jaslaryugfasbpksasgft6vy4u

24 November 2022

mapped directly with Wikidata item

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:2754711%20AND%20SRC:MED&resulttype=core&format=json

4 October 2019

PubMed publication ID

2754711

1 reference