(Q36603195)

English

Selectivity profiling of the novel EP2 receptor antagonist, PF-04418948, in functional bioassay systems: atypical affinity at the guinea pig EP2 receptor.

scientific article published on January 2013

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Selectivity profiling of the novel EP2 receptor antagonist, PF-04418948, in functional bioassay systems: atypical affinity at the guinea pig EP2 receptor (English)

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

3

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

5

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Kristof Raemdonck

6

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Maria G Belvisi

9

object named as

Maria G Belvisi

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

author name string

Mark A Birrell

1

1 reference

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6 February 2020

Sarah A Maher

2

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Nicole Dale

4

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Nick Pullen

7

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

Mark A Giembycz

8

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

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publication date

1 January 2013

1 reference

Europe PubMed Central

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6 February 2020

British Journal of Pharmacology

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

168

1 reference

Europe PubMed Central

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6 February 2020

1

1 reference

Europe PubMed Central

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6 February 2020

129-138

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

PGE(2) receptor (EP(4)) agonists: potent dilators of human bronchi and future asthma therapy?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

International Union of Basic and Clinical Pharmacology. LXXXIII: classification of prostanoid receptors, updating 15 years of progress

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

EP4 receptor as a new target for bronchodilator therapy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

In vitro and in vivo characterization of PF-04418948, a novel, potent and selective prostaglandin EP₂ receptor antagonist

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

Animal research: reporting in vivo experiments: the ARRIVE guidelines

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

Guidelines for reporting experiments involving animals: the ARRIVE guidelines

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

Prostaglandin E2 mediates cough via the EP3 receptor: implications for future disease therapy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

TRPA1 agonists evoke coughing in guinea pig and human volunteers

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

Prostanoid receptor antagonists: development strategies and therapeutic applications

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. XXXVIII. Update on terms and symbols in quantitative pharmacology

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

The prostaglandin receptor EP4 suppresses colitis, mucosal damage and CD4 cell activation in the gut

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

The role of prostaglandin E receptor subtypes (EP1, EP2, EP3, and EP4) in bone resorption: an analysis using specific agonists for the respective EPs

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

The utilization of recombinant prostanoid receptors to determine the affinities and selectivities of prostaglandins and related analogs

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

Prostanoid receptors: structures, properties, and functions

2 references

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

20 September 2018

Beta 1-adrenoceptors mediate smooth muscle relaxation in mouse isolated trachea

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

30 September 2017

pAx and competitive drug antagonism

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

28 June 2018

Host prostaglandin E(2)-EP3 signaling regulates tumor-associated angiogenesis and tumor growth

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

28 June 2018

EP2 receptors mediate airway relaxation to substance P, ATP, and PGE2.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

28 June 2018

Characterization of the prostaglandin E2 sensitive (EP)-receptor in the rat isolated trachea

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

28 June 2018

Characterisation of receptors mediating the contractile effects of prostanoids in guinea-pig and human airways

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

28 June 2018

Kinetic and empirical analysis of dose-response curves illustrated with a cardiac example

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

28 June 2018

Guide to Receptors and Channels (GRAC), 5th edition

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.02088.X

21 January 2018

Liver X receptor agonists increase airway reactivity in a model of asthma via increasing airway smooth muscle growth

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.02088.X

21 January 2018

The discovery of 6-[2-(5-chloro-2-{[(2,4-difluorophenyl)methyl]oxy}phenyl)-1-cyclopenten-1-yl]-2-pyridinecarboxylic acid, GW848687X, a potent and selective prostaglandin EP1 receptor antagonist for the treatment of inflammatory pain.

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.02088.X

21 January 2018

Distribution of prostaglandins in human tissues

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.02088.X

21 January 2018

Receptors and pathways mediating the effects of prostaglandin E2 on airway tone

1 reference

https://api.crossref.org/works/10.1111%2FJ.1476-5381.2012.02088.X

21 January 2018

Guide to Receptors and Channels (GRAC), 3rd edition

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

20 September 2018

EP(2) receptor mediates bronchodilation by PGE(2) in mice.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3570009

20 September 2018

Characterisation of the prostanoid receptors mediating contraction of guinea-pig isolated trachea

1 reference

https://pubmed.ncbi.nlm.nih.gov/22747912

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

EP1 receptor blockade attenuates both spontaneous tone and PGE2-elicited contraction in guinea pig trachealis

1 reference

https://pubmed.ncbi.nlm.nih.gov/22747912

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Theories of drug antagonism

1 reference

https://pubmed.ncbi.nlm.nih.gov/22747912

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1111/J.1476-5381.2012.02088.X

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22747912%20AND%20SRC:MED&resulttype=core&format=json

6 February 2020

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