(Q36617205)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18083520%20AND%20SRC:MED&resulttype=core&format=json

29 December 2019

title

Docking and hydropathic scoring of polysubstituted pyrrole compounds with antitubulin activity (English)

1 reference

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29 December 2019

3

1 reference

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29 December 2019

author name string

Ashutosh Tripathi

1

1 reference

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29 December 2019

Micaela Fornabaio

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18083520%20AND%20SRC:MED&resulttype=core&format=json

29 December 2019

John T Gupton

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18083520%20AND%20SRC:MED&resulttype=core&format=json

29 December 2019

David A Gewirtz

5

1 reference

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29 December 2019

W Andrew Yeudall

6

1 reference

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29 December 2019

Nina E Vega

7

1 reference

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29 December 2019

Susan L Mooberry

8

1 reference

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29 December 2019

language of work or name

English

0 references

publication date

4 December 2007

1 reference

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Bioorganic & Medicinal Chemistry

29 December 2019

published in

1 reference

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29 December 2019

volume

16

1 reference

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29 December 2019

issue

5

1 reference

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29 December 2019

page(s)

2235-2242

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18083520%20AND%20SRC:MED&resulttype=core&format=json

Autophagic cell death, polyploidy and senescence induced in breast tumor cells by the substituted pyrrole JG-03-14, a novel microtubule poison

29 December 2019

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Anticancer drugs from nature--natural products as a unique source of new microtubule-stabilizing agents

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

2-amino and 2'-aminocombretastatin derivatives as potent antimitotic agents

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Laulimalide and synthetic laulimalide analogues are synergistic with paclitaxel and 2-methoxyestradiol

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Novel combretastatin analogues endowed with antitumor activity

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Intrinsic chemotherapy resistance to the tubulin-binding antimitotic agents in renal cell carcinoma.

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Synthesis and antimitotic activity of novel 2-methoxyestradiol analogs

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Hydrophobicity: is LogP(o/w) more than the sum of its parts?

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Comparative molecular field analysis of colchicine inhibition and tubulin polymerization for combretastatins binding to the colchicine binding site on beta-tubulin

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Development and validation of a genetic algorithm for flexible docking

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Podophyllotoxin, steganacin and combretastatin: natural products that bind at the colchicine site of tubulin

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Tubulin as a target for anticancer drugs: agents which interact with the mitotic spindle

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Probing the environment of tubulin-bound paclitaxel using fluorescent paclitaxel analogues.

28 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

The binding of vincristine, vinblastine and colchicine to tubulin.

28 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

The consequences of scoring docked ligand conformations using free energy correlations.

28 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

A common pharmacophore for a diverse set of colchicine site inhibitors using a structure-based approach

20 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Insight into tubulin regulation from a complex with colchicine and a stathmin-like domain.

20 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Simple, intuitive calculations of free energy of binding for protein-ligand complexes. 1. Models without explicit constrained water

20 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Protein-based virtual screening of chemical databases. 1. Evaluation of different docking/scoring combinations.

20 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Mapping the binding site of colchicinoids on beta -tubulin. 2-Chloroacetyl-2-demethylthiocolchicine covalently reacts predominantly with cysteine 239 and secondarily with cysteine 354.

20 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Structure-activity analysis of the interaction of curacin A, the potent colchicine site antimitotic agent, with tubulin and effects of analogs on the growth of MCF-7 breast cancer cells.

20 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Site of action of two novel pyrimidine biosynthesis inhibitors accurately predicted by the compare program.

20 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2362145

Identification and characterization of a new tubulin-binding tetrasubstituted brominated pyrrole

20 September 2018

1 reference

12 December 2020

Synthesis and cytotoxicity of 2,4-disubstituted and 2,3,4-trisubstituted brominated pyrroles in murine and human cultured tumor cells

1 reference

12 December 2020

Taxol-induced polymerization of purified tubulin. Mechanism of action

1 reference

12 December 2020

Synthesis, tubulin binding, antineoplastic evaluation, and structure-activity relationship of oncodazole analogues

1 reference

12 December 2020

Studies on the nocodazole-induced GTPase activity of tubulin

1 reference

12 December 2020

Isolation and structure of combretastatin

1 reference

12 April 2024

https://opencitations.net/index/api/v1/citations/10.1139/V82-202

Identifiers

DOI

10.1016/J.BMC.2007.11.076

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18083520%20AND%20SRC:MED&resulttype=core&format=json

29 December 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18083520%20AND%20SRC:MED&resulttype=core&format=json

29 December 2019

PubMed publication ID

18083520

1 reference