(Q36876855)

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Structure-activity relationship studies of gonadotropin-releasing hormone antagonists containing S-aryl/alkyl norcysteines and their oxidized derivatives

scientific article published on 3 April 2007

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Structure-activity relationship studies of gonadotropin-releasing hormone antagonists containing S-aryl/alkyl norcysteines and their oxidized derivatives (English)

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

P. Michael Conn

5

object named as

P Michael Conn

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

author name string

Manoj P Samant

1

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Richard White

2

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Doley J Hong

3

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Glenn Croston

4

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Jo Ann Janovick

6

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Jean Rivier

7

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

language of work or name

0 references

publication date

3 April 2007

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Journal of Medicinal Chemistry

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

50

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

9

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

2067-2077

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Novel analogues of degarelix incorporating hydroxy-, methoxy-, and pegylated-urea moieties at positions 3, 5, 6 and the N-terminus. Part III

1 reference

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29 September 2017

Portage of various compounds into bacteria by attachment to glycine residues in peptides

1 reference

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29 September 2017

Iterative approach to the discovery of novel degarelix analogues: substitutions at positions 3, 7, and 8. Part II.

1 reference

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29 September 2017

Novel sst(4)-selective somatostatin (SRIF) agonists. 1. Lead identification using a betide scan

1 reference

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29 September 2017

Biological characterization of a novel, orally active small molecule gonadotropin-releasing hormone (GnRH) antagonist using castrated and intact rats

1 reference

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29 September 2017

GnRH antagonists: a new generation of long acting analogues incorporating p-ureido-phenylalanines at positions 5 and 6.

1 reference

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29 September 2017

SST3-selective potent peptidic somatostatin receptor antagonists

1 reference

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29 September 2017

Solution structure of methionine-oxidized amyloid beta-peptide (1-40). Does oxidation affect conformational switching?

1 reference

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Two new forms of gonadotropin-releasing hormone in a protochordate and the evolutionary implications

1 reference

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Betidamino acids: versatile and constrained scaffolds for drug discovery

1 reference

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Characterization of a teleost gonadotropin-releasing hormone

1 reference

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29 September 2017

Gonadotropin-releasing hormone analog design. Structure-function studies toward the development of agonists and antagonists: rationale and perspective

1 reference

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29 September 2017

Distinct sequence of gonadotropin-releasing hormone (GnRH) in dogfish brain provides insight into GnRH evolution

1 reference

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29 September 2017

The dynamics of gonadotropin inhibition in women induced by an antagonistic analog of gonadotropin-releasing hormone

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536683

29 September 2017

Betidamino acid scan of the GnRH antagonist acyline

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536683

27 June 2018

Primary structure and biological activity of a third gonadotropin-releasing hormone from lamprey brain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536683

27 June 2018

Gonadotropin-Releasing Hormone Antagonists: Novel Members of the Azaline B Family

1 reference

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27 June 2018

Gonadotropin-releasing hormone causes transcriptional stimulation followed by desensitization of the glycoprotein hormone alpha promoter in transfected alpha T3 gonadotrope cells

1 reference

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27 June 2018

Synthetic luteinizing hormone releasing factor analogs. Series of short-chain amide LRF homologs converging to the amino terminus

1 reference

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27 June 2018

Structure-activity relationships in the C-terminal part of luteinizing hormone releasing hormone (LH-RH)

1 reference

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27 June 2018

Primary structure of gonadotropin-releasing hormone from lamprey brain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2536683

27 June 2018

Use of lithium ion in measurement of stimulated pituitary inositol phospholipid turnover

1 reference

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27 June 2018

Novel gonadotropin-releasing hormone antagonists: peptides incorporating modified N omega-cyanoguanidino moieties

1 reference

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27 June 2018

Gonadotropin-releasing hormone antagonists with N.omega.-triazolylornithine, -lysine, or -p-aminophenylalanine residues at positions 5 and 6

1 reference

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27 June 2018

Parallel regulation of membrane trafficking and dominant-negative effects by misrouted gonadotropin-releasing hormone receptor mutants

1 reference

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4 September 2018

A single dose of the potent gonadotropin-releasing hormone antagonist acyline suppresses gonadotropins and testosterone for 2 weeks in healthy young men.

1 reference

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4 September 2018

Six novel gonadotropin-releasing hormones are encoded as triplets on each of two genes in the protochordate, Ciona intestinalis.

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Oxidative induction of beta-turn conformations in cyclic peptidomimetics: conformational analyses as indicators of configuration.

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1 reference

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1 reference

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New effective gonadotropin releasing hormone antagonists with minimal potency for histamine release in vitro

1 reference

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Antagonists of luteinizing hormone releasing hormone bind to rat mast cells and induce histamine release

1 reference

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1 reference

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1 reference

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1 reference

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Identifiers

10.1021/JM0613931

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

ResearchGate publication ID

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