(Q36929434)

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In vivo pharmacological interactions between a type II positive allosteric modulator of α7 nicotinic ACh receptors and nicotinic agonists in a murine tonic pain model

scientific article published on June 2013

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scholarly article

1 reference

Europe PubMed Central

17 August 2017

In vivo pharmacological interactions between a type II positive allosteric modulator of α7 nicotinic ACh receptors and nicotinic agonists in a murine tonic pain model (English)

1 reference

Europe PubMed Central

17 August 2017

author name string

K Freitas

1

1 reference

Europe PubMed Central

17 August 2017

S S Negus

2

1 reference

Europe PubMed Central

17 August 2017

F I Carroll

3

1 reference

Europe PubMed Central

17 August 2017

M I Damaj

4

1 reference

Europe PubMed Central

17 August 2017

language of work or name

0 references

publication date

1 June 2013

1 reference

Europe PubMed Central

17 August 2017

British Journal of Pharmacology

1 reference

Europe PubMed Central

17 August 2017

169

1 reference

Europe PubMed Central

17 August 2017

3

1 reference

Europe PubMed Central

17 August 2017

567-579

1 reference

Europe PubMed Central

17 August 2017

Varenicline blocks β2*-nAChR-mediated response and activates β4*-nAChR-mediated responses in mice in vivo

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Alpha7 nicotinic acetylcholine receptors modulate motivation to self-administer nicotine: implications for smoking and schizophrenia

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Guide to Receptors and Channels (GRAC), 5th edition

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Competitive binding at a nicotinic receptor transmembrane site of two α7-selective positive allosteric modulators with differing effects on agonist-evoked desensitization

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Positive allosteric modulators as an approach to nicotinic acetylcholine receptor-targeted therapeutics: advantages and limitations

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Activation of functional α7-containing nAChRs in hippocampal CA1 pyramidal neurons by physiological levels of choline in the presence of PNU-120596

1 reference

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29 September 2017

Role of alpha5 nicotinic acetylcholine receptors in pharmacological and behavioral effects of nicotine in mice

1 reference

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29 September 2017

Neuronal nicotinic acetylcholine receptors - targets for the development of drugs to treat cognitive impairment associated with schizophrenia and Alzheimer's disease

1 reference

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29 September 2017

Cognitive improvement by activation of alpha7 nicotinic acetylcholine receptors: from animal models to human pathophysiology

1 reference

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29 September 2017

Physiological concentrations of choline activate native alpha7-containing nicotinic acetylcholine receptors in the presence of PNU-120596 [1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-methylisoxazol-3-yl)-urea].

1 reference

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29 September 2017

Deletion of the alpha 7 nicotinic acetylcholine receptor gene improves cognitive deficits and synaptic pathology in a mouse model of Alzheimer's disease

1 reference

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29 September 2017

Activation and desensitization of nicotinic alpha7-type acetylcholine receptors by benzylidene anabaseines and nicotine

1 reference

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29 September 2017

Micro/kappa opioid interactions in rhesus monkeys: implications for analgesia and abuse liability

1 reference

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29 September 2017

Allosteric modulators of the alpha7 nicotinic acetylcholine receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Allosteric modulation of nicotinic acetylcholine receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

An allosteric modulator of the alpha7 nicotinic acetylcholine receptor possessing cognition-enhancing properties in vivo

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Distinct profiles of alpha7 nAChR positive allosteric modulation revealed by structurally diverse chemotypes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

The alpha7 nicotinic acetylcholine receptor as a pharmacological target for inflammation.

1 reference

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29 September 2017

Allosteric modifiers of neuronal nicotinic acetylcholine receptors: new methods, new opportunities.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

An overview of drug combination analysis with isobolograms

1 reference

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29 September 2017

Neuronal nicotinic receptors as targets for novel analgesics

1 reference

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29 September 2017

Nicotinic modulation of neuronal networks: from receptors to cognition

1 reference

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29 September 2017

Long-lasting cognitive improvement with nicotinic receptor agonists: mechanisms of pharmacokinetic-pharmacodynamic discordance

1 reference

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29 September 2017

A novel positive allosteric modulator of the alpha7 neuronal nicotinic acetylcholine receptor: in vitro and in vivo characterization.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Antinociceptive effects of choline against acute and inflammatory pain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Null mutant analysis of responses to nicotine: deletion of beta2 nicotinic acetylcholine receptor subunit but not alpha7 subunit reduces sensitivity to nicotine-induced locomotor depression and hypothermia

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

The blood-brain barrier choline transporter as a brain drug delivery vector

1 reference

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29 September 2017

Comparative pharmacology of rat and human alpha7 nAChR conducted with net charge analysis

1 reference

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29 September 2017

Allosteric binding sites on cell-surface receptors: novel targets for drug discovery

1 reference

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29 September 2017

The therapeutic potential of nicotinic acetylcholine receptor agonists for pain control

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3682705

29 September 2017

Antagonist of nicotinic acetylcholine receptors (nAChR) enhances formalin-induced nociception in rats: tonic role of nAChRs in the control of pain following injury

1 reference

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29 September 2017

Potential role of the alpha4 and alpha6 nicotinic receptor subunits in regulating nicotine-induced seizures

1 reference

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29 September 2017

Pharmacological characterization of nicotine-induced seizures in mice

1 reference

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29 September 2017

Sensitivity to the seizure-inducing effects of nicotine is associated with strain-specific variants of the alpha 5 and alpha 7 nicotinic receptor subunit genes

1 reference

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29 September 2017

24-hour control of body temperature in the rat: II. Diisopropyl fluorophosphate-induced hypothermia and hyperthermia

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29 September 2017

The formalin test: an evaluation of the method

1 reference

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29 September 2017

α4β2 neuronal nicotinic receptor positive allosteric modulation: an approach for improving the therapeutic index of α4β2 nAChR agonists in pain

1 reference

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27 June 2018

A new microdialysis-electrochemical device for in vivo simultaneous determination of acetylcholine and choline in rat brain treated with N-methyl-(R)-salsolinol.

1 reference

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27 June 2018

Choline is a selective agonist of alpha7 nicotinic acetylcholine receptors in the rat brain neurons.

1 reference

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The effect of various neurohumoral modulators on the activity of morphine and the narcotic antagonists in the tail-flick and phenylquinone tests.

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Approaches to the study of drug interactions in behavioral pharmacology.

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An isobolographic analysis of the antinociceptive effect of systemically and intrathecally administered combinations of clonidine and opiates

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Involvement of dopamine receptor subtypes in mouse thermoregulation

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27 June 2018

The formalin test: A quantitative study of the analgesic effects of morphine, meperidine, and brain stem stimulation in rats and cats

1 reference

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27 June 2018

The α7 nicotinic ACh receptor agonist compound B and positive allosteric modulator PNU-120596 both alleviate inflammatory hyperalgesia and cytokine release in the rat.

1 reference

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4 September 2018

Hypothermia and rewarming injury in hippocampal neurons involve intracellular Ca2+ and glutamate excitotoxicity

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4 September 2018

Dissociating beta-amyloid from alpha 7 nicotinic acetylcholine receptor by a novel therapeutic agent, S 24795, normalizes alpha 7 nicotinic acetylcholine and NMDA receptor function in Alzheimer's disease brain.

1 reference

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4 September 2018

Comparative pharmacology and computational modelling yield insights into allosteric modulation of human alpha7 nicotinic acetylcholine receptors.

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4 September 2018

Enhanced nicotine sensitivity in nociceptin/orphanin FQ receptor knockout mice

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4 September 2018

Convergence of alpha 7 nicotinic acetylcholine receptor-activated pathways for anti-apoptosis and anti-inflammation: central role for JAK2 activation of STAT3 and NF-kappaB.

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Activation of the alpha7-nicotinic acetylcholine receptor reverses complete freund adjuvant-induced mechanical hyperalgesia in the rat via a central site of action

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4 September 2018

Subtype-specific inhibition of nicotinic acetylcholine receptors by choline: a regulatory pathway.

1 reference

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4 September 2018

Activation and blockade by choline of bovine alpha7 and alpha3beta4 nicotinic receptors expressed in oocytes.

1 reference

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Lower core body temperature and attenuated nicotine-induced hypothermic response in mice lacking the beta4 neuronal nicotinic acetylcholine receptor subunit

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Regulation of neuronal function by choline and 4OH-GTS-21 through alpha 7 nicotinic receptors

1 reference

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4 September 2018

The antinociceptive effects of alpha7 nicotinic agonists in an acute pain model

1 reference

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4 September 2018

Potentiation of analgesic efficacy but not side effects: co-administration of an α4β2 neuronal nicotinic acetylcholine receptor agonist and its positive allosteric modulator in experimental models of pain in rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/23004024

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Intrathecal morphine in mice: a new technique

1 reference

https://pubmed.ncbi.nlm.nih.gov/23004024

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The formalin test in mice: dissociation between inflammatory and non-inflammatory pain

1 reference

https://pubmed.ncbi.nlm.nih.gov/23004024

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effects of bupropion on core body temperature of mice

1 reference

https://pubmed.ncbi.nlm.nih.gov/23004024

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Cholinergic/serotonergic interactions in hypothermia: implications for rat models of depression

1 reference

https://pubmed.ncbi.nlm.nih.gov/23004024

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1111/J.1476-5381.2012.02226.X

1 reference

Europe PubMed Central

17 August 2017

release_qv7csieevvdcrn4cujt4pyu6ay

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https://api.fatcat.wiki/v0/release/qv7csieevvdcrn4cujt4pyu6ay

24 November 2022

based on heuristic

mapped directly with Wikidata item

1 reference

Europe PubMed Central

17 August 2017

1 reference

Europe PubMed Central

17 August 2017

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