(Q37098728)

English

First small molecular inhibitors of T. brucei dolicholphosphate mannose synthase (DPMS), a validated drug target in African sleeping sickness

scientific article published on 30 January 2009

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

First small molecular inhibitors of T. brucei dolicholphosphate mannose synthase (DPMS), a validated drug target in African sleeping sickness (English)

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Trypanosoma brucei

0 references

African trypanosomiasis

1 reference

based on heuristic

inferred from title

author name string

Terry K Smith

1

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Benjamin L Young

2

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Helen Denton

3

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

David L Hughes

4

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Gerd K Wagner

5

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

language of work or name

0 references

publication date

30 January 2009

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Bioorganic & Medicinal Chemistry Letters

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

19

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

6

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

1749-1752

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

Drugs and drug resistance in African trypanosomiasis

1 reference

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Chemical probes of UDP-galactopyranose mutase

1 reference

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Identification of active-site inhibitors of MurG using a generalizable, high-throughput glycosyltransferase screen

1 reference

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Opportunities and Challenges in Antiparasitic Drug Discovery

1 reference

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14 September 2017

VSG switching in Trypanosoma brucei: antigenic variation analysed using RNAi in the absence of immune selection.

1 reference

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14 September 2017

Chemical validation of GPI biosynthesis as a drug target against African sleeping sickness

1 reference

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Roles of N-linked glycans in the endoplasmic reticulum

1 reference

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Eflornithine for the treatment of human African trypanosomiasis

1 reference

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Waking up to sleeping sickness

1 reference

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14 September 2017

Essential roles for GPI-anchored proteins in African trypanosomes revealed using mutants deficient in GPI8

1 reference

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Pharmacokinetic investigations in patients from northern Angola refractory to melarsoprol treatment

1 reference

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Glycosylphosphatidylinositol biosynthesis validated as a drug target for African sleeping sickness

1 reference

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14 September 2017

Critical roles of glycosylphosphatidylinositol for Trypanosoma brucei

1 reference

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14 September 2017

The GPI biosynthetic pathway as a therapeutic target for African sleeping sickness.

1 reference

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Antigenic variation in trypanosomes: secrets surface slowly

1 reference

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A structural motif in the variant surface glycoproteins of Trypanosoma brucei

1 reference

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14 September 2017

Glycosyl-sn-1,2-dimyristylphosphatidylinositol is covalently linked to Trypanosoma brucei variant surface glycoprotein

1 reference

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14 September 2017

Biosynthesis of glycosyl-phosphatidylinositol lipids in Trypanosoma brucei: involvement of mannosyl-phosphoryldolichol as the mannose donor

1 reference

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14 September 2017

Enzymes that recognize dolichols participate in three glycosylation pathways and are required for protein secretion

1 reference

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14 September 2017

Cloning of Trypanosoma brucei and Leishmania major genes encoding the GlcNAc-phosphatidylinositol de-N-acetylase of glycosylphosphatidylinositol biosynthesis that is essential to the African sleeping sickness parasite.

1 reference

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29 September 2017

The role of the lipid matrix in the biosynthesis of dolichyl-linked oligosaccharides

1 reference

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29 September 2017

Selective inhibitors of the glycosylphosphatidylinositol biosynthetic pathway of Trypanosoma brucei.

1 reference

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27 June 2018

Rhodanine derivatives as novel inhibitors of PDE4.

1 reference

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3 September 2018

Identification of inhibitors for UDP-galactopyranose mutase

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3744937

3 September 2018

Rhodanine-3-acetic acid derivatives as inhibitors of fungal protein mannosyl transferase 1 (PMT1).

1 reference

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3 September 2018

Identification of selective inhibitors for the glycosyltransferase MurG via high-throughput screening

1 reference

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A simple colorimetric method to screen drug cytotoxicity against Leishmania using the dye Alamar Blue.

1 reference

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3 September 2018

Trial of prednisolone for prevention of melarsoprol-induced encephalopathy in gambiense sleeping sickness

1 reference

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4 December 2018

4-Thiazolidinones: novel inhibitors of the bacterial enzyme MurB

1 reference

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12 December 2020

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Myristylation of the membrane form of a Trypanosoma brucei variant surface glycoprotein

1 reference

https://pubmed.ncbi.nlm.nih.gov/19217283

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based on heuristic

inferred from PubMed ID database lookup

Preparations of 5-alkylmethylidene-3-carboxymethylrhodanine derivatives and their aldose reductase inhibitory activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/19217283

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.BMCL.2009.01.083

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

18 August 2017

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