(Q37388364)

20 August 2017

A naphthyridine carboxamide provides evidence for discordant resistance between mechanistically identical inhibitors of HIV-1 integrase (English)

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20 August 2017

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Daria J Hazuda

1

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20 August 2017

Neville J Anthony

2

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20 August 2017

Robert P Gomez

3

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20 August 2017

Samson M Jolly

4

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20 August 2017

John S Wai

5

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20 August 2017

Linghang Zhuang

6

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20 August 2017

Thorsten E Fisher

7

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20 August 2017

Mark Embrey

8

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20 August 2017

James P Guare

9

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20 August 2017

Melissa S Egbertson

10

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20 August 2017

Joseph P Vacca

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20 August 2017

Joel R Huff

12

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20 August 2017

Peter J Felock

13

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20 August 2017

Marc V Witmer

14

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20 August 2017

Kara A Stillmock

15

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20 August 2017

Robert Danovich

16

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20 August 2017

Jay Grobler

17

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20 August 2017

Michael D Miller

18

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20 August 2017

Amy S Espeseth

19

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20 August 2017

Lixia Jin

20

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20 August 2017

I-Wu Chen

21

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20 August 2017

Jiunn H Lin

22

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20 August 2017

Kelem Kassahun

23

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20 August 2017

Joan D Ellis

24

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20 August 2017

Bradley K Wong

25

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20 August 2017

Wei Xu

26

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20 August 2017

Paul G Pearson

27

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20 August 2017

William A Schleif

28

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20 August 2017

Riccardo Cortese

29

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20 August 2017

Emilio Emini

30

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20 August 2017

Vincenzo Summa

31

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20 August 2017

M Katharine Holloway

32

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20 August 2017

Steven D Young

33

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20 August 2017

language of work or name

English

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publication date

26 July 2004

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Proceedings of the National Academy of Sciences of the United States of America

20 August 2017

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20 August 2017

101

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20 August 2017

31

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20 August 2017

11233-11238

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Discovery of a novel binding trench in HIV integrase.

20 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Development of resistance against diketo derivatives of human immunodeficiency virus type 1 by progressive accumulation of integrase mutations

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Inhibition of human immunodeficiency virus type 1 integration by diketo derivatives

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Diketo acid inhibitor mechanism and HIV-1 integrase: implications for metal binding in the active site of phosphotransferase enzymes

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Inhibition of HIV-1 integrase by small molecules: the potential for a new class of AIDS chemotherapeutics.

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

4-Aryl-2,4-dioxobutanoic acid inhibitors of HIV-1 integrase and viral replication in cells

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

HIV-1 integrase inhibitors that compete with the target DNA substrate define a unique strand transfer conformation for integrase

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Crystal structure of the HIV-1 integrase catalytic core and C-terminal domains: A model for viral DNA binding

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Inhibitors of strand transfer that prevent integration and inhibit HIV-1 replication in cells

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Structure of the HIV-1 integrase catalytic domain complexed with an inhibitor: a platform for antiviral drug design

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

HIV-1 integrase: structural organization, conformational changes, and catalysis

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

HIV integrase structure and function.

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Crystal structures of the catalytic domain of HIV-1 integrase free and complexed with its metal cofactor: high level of similarity of the active site with other viral integrases

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

L-735,524: an orally bioavailable human immunodeficiency virus type 1 protease inhibitor

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Design and synthesis of 8-hydroxy-[1,6]naphthyridines as novel inhibitors of HIV-1 integrase in vitro and in infected cells

6 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Differential divalent cation requirements uncouple the assembly and catalytic reactions of human immunodeficiency virus type 1 integrase.

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

A quantitative assay for HIV DNA integration in vivo

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Inhibition of HIV-1 ribonuclease H by a novel diketo acid, 4-[5-(benzoylamino)thien-2-yl]-2,4-dioxobutanoic acid

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

A short-term clinical evaluation of L-697,661, a non-nucleoside inhibitor of HIV-1 reverse transcriptase. L-697,661 Working Group

26 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Sampling and efficiency of metric matrix distance geometry: a novel partial metrization algorithm.

26 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Discovery of alpha,gamma-diketo acids as potent selective and reversible inhibitors of hepatitis C virus NS5b RNA-dependent RNA polymerase

26 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Antiretroviral-drug resistance among patients recently infected with HIV.

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=509174

Merck molecular force field. I. Basis, form, scope, parameterization, and performance of MMFF94

2 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.0402357101

21 January 2018

Identifiers

DOI

10.1073/PNAS.0402357101

1 reference

20 August 2017

0 references

1 reference

20 August 2017

PubMed publication ID

15277684

1 reference