(Q37636314)

English

Selective allosteric enhancement of agonist binding and function at human A3 adenosine receptors by a series of imidazoquinoline derivatives

scientific article published on July 2002

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Selective allosteric enhancement of agonist binding and function at human A3 adenosine receptors by a series of imidazoquinoline derivatives (English)

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Kenneth A. Jacobson

6

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Adriaan P IJzerman

object named as

Adriaan P IJzerman

5

0 references

1

object named as

Zhan-Guo Gao

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

Kelly A Soltysiak

3

object named as

Kelly A Soltysiak

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

4

object named as

Neli Melman

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

author name string

Seong Gon Kim

2

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

publication date

1 July 2002

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

number of pages

9

1 reference

based on heuristic

inferred from page(s)

Molecular Pharmacology

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

62

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

1

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

81-89

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

[(3)H]8-Ethyl-4-methyl-2-phenyl-(8R)-4,5,7,8-tetrahydro-1H-imidazo[2,1-i]-purin-5-one ([(3)H]PSB-11), a novel high-affinity antagonist radioligand for human A(3) adenosine receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

23 August 2017

Allosteric modulation of A(3) adenosine receptors by a series of 3-(2-pyridinyl)isoquinoline derivatives

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

23 August 2017

Positive allosteric modulation of native and recombinant gamma-aminobutyric acid(B) receptors by 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its aldehyde analog CGP13501

1 reference

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23 August 2017

Positive allosteric modulators of metabotropic glutamate 1 receptor: characterization, mechanism of action, and binding site

1 reference

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23 August 2017

Novel allosteric antagonists shed light on mglu(5) receptors and CNS disorders

1 reference

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23 August 2017

Ring-Constrained (N)-methanocarba nucleosides as adenosine receptor agonists: independent 5'-uronamide and 2'-deoxy modifications

1 reference

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23 August 2017

Allosteric activation of the CaR by L-amino acids

1 reference

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23 August 2017

Biochemical methods for detection and measurement of cyclic AMP and adenylyl cyclase activity.

1 reference

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23 August 2017

Subtype-selective positive cooperative interactions between brucine analogs and acetylcholine at muscarinic receptors: functional studies

1 reference

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23 August 2017

CPCCOEt, a noncompetitive metabotropic glutamate receptor 1 antagonist, inhibits receptor signaling without affecting glutamate binding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

23 August 2017

Pharmacological characterization of novel A3 adenosine receptor-selective antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

23 August 2017

Effects of long-term treatment with the allosteric enhancer, PD81,723, on Chinese hamster ovary cells expressing recombinant human A1 adenosine receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

23 August 2017

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

23 August 2017

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

23 August 2017

Muscarinic receptor subtypes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

6 September 2017

Allosteric regulation of G-protein-linked receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

14 September 2017

GABAA receptor channels

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

14 September 2017

Allosteric enhancement of adenosine A1 receptor binding and function by 2-amino-3-benzoylthiophenes

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

25 June 2018

1H-imidazo[4,5-c]quinolin-4-amines: novel non-xanthine adenosine antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

25 June 2018

Positive allosteric modulators for gamma-aminobutyric acid(B) receptors open new routes for the development of drugs targeting family 3 G-protein-coupled receptors

1 reference

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1 September 2018

Modeling the functional effects of allosteric modulators at pharmacological receptors: an extension of the two-state model of receptor activation.

1 reference

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1 September 2018

Galantamine for Alzheimer's disease.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3953617

2 October 2018

A modification of a protein-binding method for rapid quantification of cAMP in cell-culture supernatants and body fluid

1 reference

https://pubmed.ncbi.nlm.nih.gov/12065758

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Allosteric modulation of A2A adenosine receptors by amiloride analogues and sodium ions

1 reference

https://pubmed.ncbi.nlm.nih.gov/12065758

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1124/MOL.62.1.81

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

21 August 2017

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