(Q38016197)

27 August 2017

title

TRP channels as therapeutic targets in airway disorders: a patent review (English)

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27 August 2017

Delia Preti

1

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author name string

Arpad Szallasi

series ordinal

2

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27 August 2017

Riccardo Patacchini

series ordinal

3

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27 August 2017

language of work or name

English

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publication date

6 June 2012

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Expert Opinion on Therapeutic Patents

27 August 2017

published in

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27 August 2017

volume

22

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27 August 2017

issue

6

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27 August 2017

page(s)

663-695

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The global burden of asthma: executive summary of the GINA Dissemination Committee report

27 August 2017

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Analogues of morphanthridine and the tear gas dibenz[b,f][1,4]oxazepine (CR) as extremely potent activators of the human transient receptor potential ankyrin 1 (TRPA1) channel.

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Capsaicin responsiveness and cough in asthma and chronic obstructive pulmonary disease

21 January 2018

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Local and systemic capsaicin pretreatment inhibits sneezing and the increase in nasal vascular permeability induced by certain chemical irritants

21 January 2018

1 reference

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Secretion, pain and sneezing induced by the application of capsaicin to the nasal mucosa in man

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Identification and biological evaluation of 4-(3-trifluoromethylpyridin-2-yl)piperazine-1-carboxylic acid (5-trifluoromethylpyridin-2-yl)amide, a high affinity TRPV1 (VR1) vanilloid receptor antagonist

21 January 2018

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Pharmacology and antitussive efficacy of 4-(3-trifluoromethyl-pyridin-2-yl)-piperazine-1-carboxylic acid (5-trifluoromethyl-pyridin-2-yl)-amide (JNJ17203212), a transient receptor potential vanilloid 1 antagonist in guinea pigs.

21 January 2018

1 reference

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Characterization of 2-(2,6-dichloro-benzyl)-thiazolo[5,4-d]pyrimidin-7-yl]-(4-trifluoromethyl-phenyl)-amine (JNJ-39729209) as a novel TRPV1 antagonist

21 January 2018

1 reference

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Discovery of SB-705498: a potent, selective and orally bioavailable TRPV1 antagonist suitable for clinical development

21 January 2018

1 reference

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TRPV4-mediated calcium influx into human bronchial epithelia upon exposure to diesel exhaust particles.

21 January 2018

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TRPC1, a human homolog of a Drosophila store-operated channel

21 January 2018

1 reference

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Expression profile of the transient receptor potential (TRP) family in neutrophil granulocytes: evidence for currents through long TRP channel 2 induced by ADP-ribose and NAD.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2012.696099

E-selectin permits communication between PAF receptors and TRPC channels in human neutrophils.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2012.696099

The calcium-conducting ion channel transient receptor potential canonical 6 is involved in macrophage inflammatory protein-2-induced migration of mouse neutrophils

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2012.696099

Selective blockade of TRPA1 channel attenuates pathological pain without altering noxious cold sensation or body temperature regulation

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2012.696099

10.1517/13543776.2012.696099

21 January 2018

Identifiers

DOI

1 reference

27 August 2017

1 reference