(Q38075043)

English

Exploring avidity: understanding the potential gains in functional affinity and target residence time of bivalent and heterobivalent ligands

scientific article published on April 2013

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

1 reference

Europe PubMed Central

Exploring avidity: understanding the potential gains in functional affinity and target residence time of bivalent and heterobivalent ligands (English)

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

author name string

Georges Vauquelin

1

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

Steven J Charlton

2

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

language of work or name

0 references

publication date

1 April 2013

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

British Journal of Pharmacology

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

168

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

8

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

1771-1785

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

Rebinding: or why drugs may act longer in vivo than expected from their in vitro target residence time

1 reference

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Guide to Receptors and Channels (GRAC), 5th edition

1 reference

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The best of both worlds? Bitopic orthosteric/allosteric ligands of g protein-coupled receptors

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Long-lasting target binding and rebinding as mechanisms to prolong in vivo drug action

1 reference

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Ligands, their receptors and ... plasma membranes

1 reference

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The importance of drug-target residence time.

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Identifiers

10.1111/BPH.12106

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

28 August 2017

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