(Q38166973)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

1 March 2020

title

Radiosynthesis of carbon-11 and fluorine-18 labelled radiotracers to image the ionotropic and metabotropic glutamate receptors (English)

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

1 March 2020

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1

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

1 March 2020

author name string

Franck Sobrio

series ordinal

1

1 reference

30 August 2017

publication date

1 March 2013

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

Journal of Labelled Compounds and Radiopharmaceuticals

1 March 2020

published in

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

1 March 2020

volume

56

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

1 March 2020

issue

3-4

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

1 March 2020

page(s)

180-186

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

Ionotropic and metabotropic glutamate receptor structure and pharmacology

1 March 2020

cites work

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NMDA-receptor activity visualized with (S)-[N-methyl-11C]ketamine and positron emission tomography in patients with medial temporal lobe epilepsy

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Fluorine-18 radiolabelling, biodistribution studies and preliminary PET evaluation of a new memantine derivative for imaging the NMDA receptor

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In vivo evaluation of [11C]N-(2-chloro-5-thiomethylphenyl)-N'-(3-methoxy-phenyl)-N'-methylguanidine ([11C]GMOM) as a potential PET radiotracer for the PCP/NMDA receptor.

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Closing in on the AMPA receptor: synthesis and evaluation of 2-acetyl-1-(4'-chlorophenyl)-6-methoxy-7-[11C]methoxy-1,2,3,4-tetrahydroisoquinoline as a potential PET tracer

21 January 2018

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A remote-controlled high pressure reactor for radiotracer synthesis with [11C]carbon monoxide

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21 January 2018

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Synthesis, structure-activity relationship, and receptor pharmacology of a new series of quinoline derivatives acting as selective, noncompetitive mGlu1 antagonists

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Radiosynthesis and evaluation of [11C]YM-202074 as a PET ligand for imaging the metabotropic glutamate receptor type 1.

21 January 2018

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Synthesis, in vitro and in vivo evaluation of [11C]MMTP: a potential PET ligand for mGluR1 receptors

21 January 2018

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Synthesis, characterization, and monkey PET studies of [¹⁸F]MK-1312, a PET tracer for quantification of mGluR1 receptor occupancy by MK-5435.

21 January 2018

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Characterization of 1-(2-[18F] fluoro-3-pyridyl)-4-(2-isopropyl-1-oxo- isoindoline-5-yl)-5-methyl-1H-1,2,3-triazole, a PET ligand for imaging the metabotropic glutamate receptor type 1 in rat and monkey brains

21 January 2018

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Synthesis and evaluation of 6-[1-(2-[(18)F]fluoro-3-pyridyl)-5-methyl-1H-1,2,3-triazol-4-yl]quinoline for positron emission tomography imaging of the metabotropic glutamate receptor type 1 in brain

21 January 2018

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Radiosynthesis and preliminary evaluation of 4-[18F]fluoro-N-[4-[6-(isopropylamino)pyrimidin-4-yl]-1,3-thiazol-2-yl]-N-methylbenzamide as a new positron emission tomography ligand for metabotropic glutamate receptor subtype 1.

21 January 2018

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21 January 2018

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21 January 2018

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Modulation of dopaminergic and glutamatergic brain function: PET studies on parkinsonian rats

21 January 2018

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Enhanced binding of metabotropic glutamate receptor type 5 (mGluR5) PET tracers in the brain of parkinsonian primates

21 January 2018

1 reference

Biodistribution and radiation dosimetry of [18F]F-PEB in nonhuman primates

21 January 2018

1 reference

Synthesis and simple 18F-labeling of 3-fluoro-5-(2-(2-(fluoromethyl)thiazol-4-yl)ethynyl)benzonitrile as a high affinity radioligand for imaging monkey brain metabotropic glutamate subtype-5 receptors with positron emission tomography

21 January 2018

1 reference

Metabotropic glutamate subtype 5 receptors are quantified in the human brain with a novel radioligand for PET

21 January 2018

1 reference

Quantification of metabotropic glutamate subtype 5 receptors in the brain by an equilibrium method using 18F-SP203

21 January 2018

1 reference

Biodistribution and radiation dosimetry of a positron emission tomographic ligand, 18F-SP203, to image metabotropic glutamate subtype 5 receptors in humans

21 January 2018

1 reference

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21 January 2018

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Synthesis, characterization, and first successful monkey imaging studies of metabotropic glutamate receptor subtype 5 (mGluR5) PET radiotracers

21 January 2018

1 reference

In vivo positron emission tomography imaging with [¹¹C]ABP688: binding variability and specificity for the metabotropic glutamate receptor subtype 5 in baboons.

21 January 2018

1 reference

Evaluation of the metabotropic glutamate receptor subtype 5 using PET and 11C-ABP688: assessment of methods

21 January 2018

1 reference

ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: identification, in vitro pharmacology, pharmacokinetic and biodistribution studies

21 January 2018

1 reference

In vivo and in vitro validation of reference tissue models for the mGluR(5) ligand [(11)C]ABP688.

21 January 2018

1 reference

Quantitative evaluation of 11C-ABP688 as PET ligand for the measurement of the metabotropic glutamate receptor subtype 5 using autoradiographic studies and a beta-scintillator

21 January 2018

1 reference

Metabotropic glutamate receptor modulation, translational methods, and biomarkers: relationships with anxiety.

21 January 2018

1 reference

Radiation dosimetry and biodistribution of 11C-ABP688 measured in healthy volunteers

21 January 2018

1 reference

Evaluation of a bolus/infusion protocol for 11C-ABP688, a PET tracer for mGluR5.

21 January 2018

1 reference

Reduced metabotropic glutamate receptor 5 density in major depression determined by [(11)C]ABP688 PET and postmortem study

21 January 2018

1 reference

In vivo variation in metabotropic glutamate receptor subtype 5 binding using positron emission tomography and [11C]ABP688.

21 January 2018

1 reference

Synthesis, radiolabeling, in vitro and in vivo evaluation of [18F]-FPECMO as a positron emission tomography radioligand for imaging the metabotropic glutamate receptor subtype 5.

21 January 2018

1 reference

Radiolabeling and in vitro and in vivo evaluation of [18F]-FE-DABP688 as a PET radioligand for the metabotropic glutamate receptor subtype 5.

21 January 2018

1 reference

In vitro and in vivo evaluation of [18F]-FDEGPECO as a PET tracer for imaging the metabotropic glutamate receptor subtype 5 (mGluR5).

21 January 2018

1 reference

Syntheses and pharmacological characterization of novel thiazole derivatives as potential mGluR5 PET ligands

21 January 2018

1 reference

21 January 2018

Identifiers

DOI

10.1002/JLCR.2995

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24285324%20AND%20SRC:MED&resulttype=core&format=json

1 March 2020

1 reference