(Q38876007)

English

Discovery of 1-(3,3-dimethylbutyl)-3-(2-fluoro-4-methyl-5-(7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl)phenyl)urea (LY3009120) as a pan-RAF inhibitor with minimal paradoxical activation and activity against BRAF or RAS mutant tumor cells

scientific article published on 12 May 2015

Statements

Discovery of 1-(3,3-dimethylbutyl)-3-(2-fluoro-4-methyl-5-(7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl)phenyl)urea (LY3009120) as a pan-RAF inhibitor with minimal paradoxical activation and activity against BRAF or RAS mutant tumor cells (English)
James R Henry
Michael D Kaufman
Sheng-Bin Peng
Yu Mi Ahn
Timothy M Caldwell
Lakshminarayana Vogeti
Hanumaiah Telikepalli
Wei-Ping Lu
Molly M Hood
Thomas J Rutkoski
Bryan D Smith
Subha Vogeti
Scott C Wise
Lawrence Chun
Xiaoyi Zhang
Youyan Zhang
Lisa Kays
Philip A Hipskind
Aaron D Wrobleski
Karen L Lobb
Julia M Clay
Jeffrey D Cohen
Jennie L Walgren
Denis McCann
Phenil Patel
David K Clawson
Sherry Guo
Danalyn Manglicmot
Chris Groshong
Cheyenne Logan
James J Starling
Daniel L Flynn
12 May 2015
4165-4179

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