(Q40169268)

18 September 2017

Characterization of the potency, selectivity, and pharmacokinetic profile for six adenosine A2A receptor antagonists (English)

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18 September 2017

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Ming Yang

1

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18 September 2017

Daniel Soohoo

2

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18 September 2017

Sandriyana Soelaiman

3

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18 September 2017

Rao Kalla

4

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18 September 2017

Jeff Zablocki

5

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18 September 2017

Nancy Chu

6

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18 September 2017

Kwan Leung

7

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18 September 2017

Lina Yao

8

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18 September 2017

Ivan Diamond

9

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18 September 2017

Luiz Belardinelli

10

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18 September 2017

John C Shryock

11

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18 September 2017

20 February 2007

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Naunyn-Schmiedeberg's Archives of Pharmacology

18 September 2017

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18 September 2017

375

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18 September 2017

2

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18 September 2017

133-144

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https://scigraph.springernature.com/pub.10.1007/s00210-007-0135-0

18 September 2017

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cites work

Discovery of nonxanthine adenosine A2A receptor antagonists for the treatment of Parkinson's disease

1 reference

Crossref

https://api.crossref.org/works/10.1007%2FS00210-007-0135-0

Water-soluble phosphate prodrugs of 1-propargyl-8-styrylxanthine derivatives, A(2A)-selective adenosine receptor antagonists

21 January 2018

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12 December 2020

The non-xanthine heterocyclic compound SCH 58261 is a new potent and selective A2a adenosine receptor antagonist.

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12 December 2020

8-(Sulfostyryl)xanthines: water-soluble A2A-selective adenosine receptor antagonists.

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12 December 2020

Piperazine derivatives of [1,2,4]triazolo[1,5-a][1,3,5]triazine as potent and selective adenosine A2a receptor antagonists

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12 December 2020

KW-6002 (Kyowa Hakko Kogyo).

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12 December 2020

Receptors for purines and pyrimidines

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12 December 2020

Selective adenosine A2A receptor antagonists

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12 December 2020

125I-4-aminobenzyl-5'-N-methylcarboxamidoadenosine, a high affinity radioligand for the rat A3 adenosine receptor

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12 December 2020

Adenosine receptors and their ligands.

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12 December 2020

Multigram-scale syntheses, stability, and photoreactions of A2A adenosine receptor antagonists with 8-styrylxanthine structure: potential drugs for Parkinson's disease

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12 December 2020

Distribution of adenosine A(2A) receptor antagonist KW-6002 and its effect on gene expression in the rat brain

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12 December 2020

Analogues of 1,3-dipropyl-8-phenylxanthine: enhancement of selectivity at A1-adenosine receptors by aryl substituents

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12 December 2020

Studies on adenosine A2a receptor antagonists: comparison of three core heterocycles

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12 December 2020

Differences in the order of potency for agonists but not antagonists at human and rat adenosine A2A receptors

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12 December 2020

Hydrophilic side chains in the third and seventh transmembrane helical domains of human A2A adenosine receptors are required for ligand recognition

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12 December 2020

Medicinal chemistry of A2A adenosine receptor antagonists

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12 December 2020

Characterization of human A2A adenosine receptors with the antagonist radioligand [3H]-SCH 58261

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12 December 2020

Pharmacological and biochemical characterization of adenosine receptors in the human malignant melanoma A375 cell line

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12 December 2020

Motor effects induced by a blockade of adenosine A2A receptors in the caudate-putamen.

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12 December 2020

International Union of Pharmacology. XXV. Nomenclature and classification of adenosine receptors

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12 December 2020

Binding of adenosine receptor ligands to brain of adenosine receptor knock-out mice: evidence that CGS 21680 binds to A1 receptors in hippocampus.

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12 December 2020

Binding of [3H]MSX-2 (3-(3-hydroxypropyl)-7-methyl-8-(m-methoxystyryl)-1-propargylxanthine) to rat striatal membranes--a new, selective antagonist radioligand for A(2A) adenosine receptors

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12 December 2020

G protein coupling of CGS 21680 binding sites in the rat hippocampus and cortex is different from that of adenosine A1 and striatal A2A receptors.

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12 December 2020

Chronic effects of xanthines on levels of central receptors in mice

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12 December 2020

Pharmacodynamics of ZM 241385, a potent A2a adenosine receptor antagonist, after enteric administration in rat, cat and dog

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12 December 2020

Effects of an adenosine A2A receptor blockade in the nucleus accumbens on locomotion, feeding, and prepulse inhibition in rats

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12 December 2020

3,7-Dimethyl-1-propargylxanthine: a potent and selective in vivo antagonist of adenosine analogs

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12 December 2020

Evidence for high-affinity binding sites for the adenosine A2A receptor agonist [3H] CGS 21680 in the rat hippocampus and cerebral cortex that are different from striatal A2A receptors.

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12 December 2020

10.1007/S00210-007-0135-0

Identifiers

DOI

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18 September 2017

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