(Q40388658)

English

Expression of a G protein-coupled receptor (GPCR) leads to attenuation of signaling by other GPCRs: experimental evidence for a spontaneous GPCR constitutive inactive form.

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scholarly article

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

Expression of a G protein-coupled receptor (GPCR) leads to attenuation of signaling by other GPCRs: experimental evidence for a spontaneous GPCR constitutive inactive form (English)

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

G protein-coupled receptor

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Carlos Fitzsimons

3

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

author name string

Maria Rosario Tubio

1

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21 January 2020

Natalia Fernandez

2

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

Sabrina Copsel

4

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21 January 2020

Sergio Santiago

5

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21 January 2020

Carina Shayo

6

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21 January 2020

Carlos Davio

7

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

Federico Monczor

8

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21 January 2020

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publication date

18 March 2010

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21 January 2020

Journal of Biological Chemistry

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

285

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21 January 2020

20

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21 January 2020

14990-14998

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

Calcitonin targets extracellular signal-regulated kinase signaling pathway in human cancers

1 reference

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Histamine-mediated signaling processes in human malignant mammary cells

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22 September 2017

Overexpression of G protein-coupled receptors in cancer cells: involvement in tumor progression

1 reference

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22 September 2017

Activation of adenylyl cyclase by endogenous G(s)-coupled receptors in human embryonic kidney 293 cells is attenuated by 5-HT(7) receptor expression.

1 reference

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22 September 2017

Multiple signaling states of G-protein-coupled receptors

1 reference

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22 September 2017

Principles: receptor theory in pharmacology

1 reference

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Histamine H1 and H2 receptor gene and protein levels are differentially expressed in the hearts of rodents and humans.

1 reference

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22 September 2017

Cardiac-specific overexpression of human beta2 adrenoceptors in mice exposes coupling to both Gs and Gi proteins

1 reference

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22 September 2017

Histamine H2 receptor desensitization: involvement of a select array of G protein-coupled receptor kinases

1 reference

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22 September 2017

G-protein-coupled receptor heterodimerization modulates receptor function

1 reference

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22 September 2017

Mechanisms governing the activation and trafficking of yeast G protein-coupled receptors.

1 reference

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22 September 2017

Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptors

1 reference

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Dopamine D4 receptors elevated in schizophrenia

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22 September 2017

A mutation-induced activated state of the beta 2-adrenergic receptor. Extending the ternary complex model

1 reference

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22 September 2017

The guinea pig histamine H2 receptor: gene cloning, tissue expression and chromosomal localization of its human counterpart

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2865266

22 September 2017

Antagonists with negative intrinsic activity at delta opioid receptors coupled to GTP-binding proteins

1 reference

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22 September 2017

Cloning and tissue expression of a rat histamine H2-receptor gene

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2865266

22 September 2017

Molecular cloning of the human histamine H2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2865266

22 September 2017

Molecular cloning of a gene encoding the histamine H2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2865266

22 September 2017

Mepyramine, a histamine H1 receptor inverse agonist, binds preferentially to a G protein-coupled form of the receptor and sequesters G protein.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2865266

17 June 2018

Role of prostaglandin E2 receptors in migration of murine and human breast cancer cells.

1 reference

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17 June 2018

Tiotidine, a histamine H2 receptor inverse agonist that binds with high affinity to an inactive G-protein-coupled form of the receptor. Experimental support for the cubic ternary complex model

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2865266

17 June 2018

Retrovirally mediated transfer of a G protein-coupled receptor kinase (GRK) dominant-negative mutant enhances endogenous calcitonin receptor signaling in Chinese hamster ovary cells. GRK inhibition enhances expression of receptors and receptor mRNA.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2865266

17 June 2018

Synergistic receptor-activated calcium increases in single nonpigmented epithelial cells

1 reference

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The cubic ternary complex receptor-occupancy model. III. resurrecting efficacy

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1 reference

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1 reference

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Histamine H2 receptor overexpression induces U937 cell differentiation despite triggered mechanisms to attenuate cAMP signalling

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1 reference

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1 reference

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1 reference

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1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Different calcium-mobilizing receptors share the same guanine nucleotide-binding protein pool in hepatocytes

1 reference

https://pubmed.ncbi.nlm.nih.gov/20299453

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

H1 and H2 histamine receptors in n-nitroso-N-methylurea (NMU)-induced carcinomas with atypical coupling to signal transducers

1 reference

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based on heuristic

inferred from PubMed ID database lookup

Collisions and encounters in simulations of receptor/GTP-binding protein interactions via simple diffusion

1 reference

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inferred from PubMed ID database lookup

A Selective Inverse Agonist for Central Cannabinoid Receptor Inhibits Mitogen-activated Protein Kinase Activation Stimulated by Insulin or Insulin-like Growth Factor 1

1 reference

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inferred from PubMed ID database lookup

Functional coupling of endogenous serotonin (5-HT1B) and calcitonin (C1a) receptors in CHO cells to a cyclic AMP-responsive luciferase reporter gene

1 reference

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inferred from PubMed ID database lookup

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1 reference

https://pubmed.ncbi.nlm.nih.gov/20299453

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1074/JBC.M109.099689

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

PMC publication ID

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

PubMed publication ID

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20299453%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

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