(Q40716260)

English

Characterization of the efflux transporter(s) responsible for restricting intestinal mucosa permeation of the coumarinic acid-based cyclic prodrug of the opioid peptide DADLE.

scientific article published on June 2002

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scholarly article

1 reference

Europe PubMed Central

23 September 2017

Characterization of the efflux transporter(s) responsible for restricting intestinal mucosa permeation of the coumarinic acid-based cyclic prodrug of the opioid peptide DADLE. (English)

1 reference

Europe PubMed Central

23 September 2017

author name string

Fuxing Tang

1

1 reference

Europe PubMed Central

23 September 2017

Ronald T Borchardt

2

1 reference

Europe PubMed Central

23 September 2017

language of work or name

1 reference

based on heuristic

inferred from title

publication date

1 June 2002

1 reference

Europe PubMed Central

23 September 2017

Pharmaceutical Research

1 reference

Europe PubMed Central

23 September 2017

19

1 reference

Europe PubMed Central

23 September 2017

6

1 reference

Europe PubMed Central

23 September 2017

787-793

1 reference

Europe PubMed Central

23 September 2017

Increased bioavailability of the food-derived carcinogen 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine in MRP2-deficient rats.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Age-dependent expression of P-glycoprotein gp170 in Caco-2 cell monolayers

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Conjugate export pumps of the multidrug resistance protein (MRP) family: localization, substrate specificity, and MRP2-mediated drug resistance

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Acyloxyalkoxy-based cyclic prodrugs of opioid peptides: evaluation of the chemical and enzymatic stability as well as their transport properties across Caco-2 cell monolayers

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

P-Glycoprotein (P-gp) mediated efflux in Caco-2 cell monolayers: the influence of culturing conditions and drug exposure on P-gp expression levels.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Intestinal drug absorption and metabolism in cell cultures: Caco-2 and beyond

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Expression of the apical conjugate export pump, Mrp2, in the polarized hepatoma cell line, WIF-B.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Functional expression of P-glycoprotein in apical membranes of human intestinal Caco-2 cells. Kinetics of vinblastine secretion and interaction with modulators

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Characterization of the efflux transporter(s) responsible for restricting intestinal mucosa permeation of an acyloxyalkoxy-based cyclic prodrug of the opioid peptide DADLE.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Association of intestinal peptide transport with a protein related to the cadherin superfamily

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Analysis of expression of cMOAT (MRP2), MRP3, MRP4, and MRP5, homologues of the multidrug resistance-associated protein gene (MRP1), in human cancer cell lines

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Transport of the flavonoid chrysin and its conjugated metabolites by the human intestinal cell line Caco-2.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Availability of PSC833, a substrate and inhibitor of P-glycoproteins, in various concentrations of serum.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evaluation of the bile acid transporter in enhancing intestinal permeability to renin-inhibitory peptides

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Are MDCK cells transfected with the human MRP2 gene a good model of the human intestinal mucosa?

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Active secretion and enterocytic drug metabolism barriers to drug absorption

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The multidrug resistance protein family.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effects of a potent and specific P-glycoprotein inhibitor on the blood-brain barrier distribution and antinociceptive effect of morphine in the rat.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A functional assay for quantitation of the apparent affinities of ligands of P-glycoprotein in Caco-2 cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Coumarinic acid-based cyclic prodrugs of opioid peptides that exhibit metabolic stability to peptidases and excellent cellular permeability

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Are MDCK cells transfected with the human MDR1 gene a good model of the human intestinal mucosa?

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Caco-2 monolayers in experimental and theoretical predictions of drug transport

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

cDNA cloning of the hepatocyte canalicular isoform of the multidrug resistance protein, cMrp, reveals a novel conjugate export pump deficient in hyperbilirubinemic mutant rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Evidence for a polarized efflux system for peptides in the apical membrane of Caco-2 cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Disruption of the mouse mdr1a P-glycoprotein gene leads to a deficiency in the blood-brain barrier and to increased sensitivity to drugs

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Drug export activity of the human canalicular multispecific organic anion transporter in polarized kidney MDCK cells expressing cMOAT (MRP2) cDNA

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Transport of glutathione prostaglandin A conjugates by the multidrug resistance protein 1.

1 reference

https://pubmed.ncbi.nlm.nih.gov/12134948

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1023/A:1016196514217

1 reference

Europe PubMed Central

23 September 2017

1 reference

Europe PubMed Central

23 September 2017

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