Home
Random
Nearby
Log in
Settings
Donate
About Wikidata
Disclaimers
Search
(Q41470342)
Watch
English
Small Molecule Inhibitors of Regulator of G Protein Signalling (RGS) Proteins
scientific article published on February 2012
In more languages
default for all languages
No label defined
No description defined
edit
Statements
instance of
scholarly article
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
title
Small Molecule Inhibitors of Regulator of G Protein Signalling (RGS) Proteins
(English)
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
author
Richard Neubig
series ordinal
3
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
Stephen M. Husbands
series ordinal
4
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
author name string
Emma M Turner
series ordinal
1
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
Levi L Blazer
series ordinal
2
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
publication date
1 February 2012
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
published in
ACS Medicinal Chemistry Letters
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
volume
3
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
issue
2
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
page(s)
146-150
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
cites work
A nanomolar-potency small molecule inhibitor of regulator of G-protein signaling proteins
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Opioid-induced down-regulation of RGS4: role of ubiquitination and implications for receptor cross-talk
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Inhibition of glioblastoma growth by the thiadiazolidinone compound TDZD-8
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Thinking outside of the "RGS box": new approaches to therapeutic targeting of regulators of G protein signaling.
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
RGS inhibition at G(alpha)i2 selectively potentiates 5-HT1A-mediated antidepressant effects.
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Allosteric inhibition of the regulator of G protein signaling-Galpha protein-protein interaction by CCG-4986
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Use of flow cytometric methods to quantify protein-protein interactions.
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Polyplexed flow cytometry protein interaction assay: a novel high-throughput screening paradigm for RGS protein inhibitors
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Differential modulation of mu- and delta-opioid receptor agonists by endogenous RGS4 protein in SH-SY5Y cells
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Small molecule protein-protein interaction inhibitors as CNS therapeutic agents: current progress and future hurdles.
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
R4 RGS proteins: regulation of G-protein signaling and beyond
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Efficacy of small-molecule glycogen synthase kinase-3 inhibitors in the postnatal rat model of tau hyperphosphorylation
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Rapid and selective death of leukemia stem and progenitor cells induced by the compound 4-benzyl, 2-methyl, 1,2,4-thiadiazolidine, 3,5 dione (TDZD-8)
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Active Galpha(q) subunits and M3 acetylcholine receptors promote distinct modes of association of RGS2 with the plasma membrane
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Identification of small-molecule inhibitors of RGS4 using a high-throughput flow cytometry protein interaction assay
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Mammalian RGS proteins: multifunctional regulators of cellular signalling.
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Molecular taxonomy of major neuronal classes in the adult mouse forebrain
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
The druggable genome
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Regulators of G-protein signaling (RGS) proteins: region-specific expression of nine subtypes in rat brain
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Structure of RGS4 bound to AlF4--activated G(i alpha1): stabilization of the transition state for GTP hydrolysis
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
11 June 2018
Antidepressant-like effect of the novel thiadiazolidinone NP031115 in mice
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
19 August 2018
First non-ATP competitive glycogen synthase kinase 3 beta (GSK-3beta) inhibitors: thiadiazolidinones (TDZD) as potential drugs for the treatment of Alzheimer's disease
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3285107
retrieved
19 August 2018
Identifiers
DOI
10.1021/ML200263Y
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
PMC publication ID
3285107
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
PubMed publication ID
22368763
1 reference
stated in
Europe PubMed Central
PMC publication ID
3285107
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:22368763%20AND%20SRC:MED&resulttype=core&format=json
retrieved
24 January 2020
ResearchGate publication ID
221865018
0 references
Sitelinks
Wikipedia
(0 entries)
edit
Wikibooks
(0 entries)
edit
Wikinews
(0 entries)
edit
Wikiquote
(0 entries)
edit
Wikisource
(0 entries)
edit
Wikiversity
(0 entries)
edit
Wikivoyage
(0 entries)
edit
Wiktionary
(0 entries)
edit
Multilingual sites
(0 entries)
edit