(Q41888707)

13 October 2017

Acylideneoxoindoles: a new class of reversible inhibitors of human transglutaminase 2. (English)

1 reference

13 October 2017

3

1 reference

13 October 2017

Cornelius Klöck

1

1 reference

13 October 2017

Xi Jin

2

1 reference

13 October 2017

Chaitan Khosla

4

1 reference

13 October 2017

Peter B Madrid

5

1 reference

13 October 2017

Andrew Spencer

6

1 reference

13 October 2017

Brian C Raimundo

7

1 reference

13 October 2017

Paul Boardman

8

1 reference

13 October 2017

Guido Lanza

9

1 reference

13 October 2017

John H Griffin

10

1 reference

13 October 2017

language of work or name

English

0 references

publication date

16 December 2010

1 reference

Bioorganic & Medicinal Chemistry Letters

13 October 2017

1 reference

13 October 2017

21

1 reference

13 October 2017

9

1 reference

13 October 2017

2692-2696

1 reference

A profiling platform for the characterization of transglutaminase 2 (TG2) inhibitors

13 October 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Cytotoxic and anticancer activities of isatin and its derivatives: a comprehensive review from 2000-2008.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Identification of chemical inhibitors to human tissue transglutaminase by screening existing drug libraries

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Tissue transglutaminase contributes to interstitial renal fibrosis by favoring accumulation of fibrillar collagen through TGF-beta activation and cell infiltration.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Tissue transglutaminase activation modulates inflammation in cystic fibrosis via PPARgamma down-regulation.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Tissue transglutaminase-mediated chemoresistance in cancer cells

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Transglutaminase 2 inhibitors and their therapeutic role in disease states

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Noxious compounds activate TRPA1 ion channels through covalent modification of cysteines

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Structure-activity relationship analysis of the selective inhibition of transglutaminase 2 by dihydroisoxazoles

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Transglutaminase 2 in neurodegenerative disorders

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Transglutaminases in neurodegenerative disorders.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

A library of spirooxindoles based on a stereoselective three-component coupling reaction.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Transglutaminase 2: an enigmatic enzyme with diverse functions

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Coeliac disease: dissecting a complex inflammatory disorder

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

High selectivity of human tissue transglutaminase for immunoactive gliadin peptides: implications for celiac sprue

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Potent and selective nonpeptide inhibitors of caspases 3 and 7.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Asymmetric quadruple aminocatalytic domino reactions to fused carbocycles incorporating a spirooxindole motif

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Potent transglutaminase inhibitors, aryl beta-aminoethyl ketones.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Targeting structural and stereochemical complexity by organocascade catalysis: construction of spirocyclic oxindoles having multiple stereocenters

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Cinnamoyl inhibitors of tissue transglutaminase.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Vasodilatory activity of novel carbamate derivatives of isatin

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Design and synthesis of N-alkyl oxindolylidene acetic acids as a new class of potent Cdc25A inhibitors.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Enantioselective construction of spirocyclic oxindolic cyclopentanes by palladium-catalyzed trimethylenemethane-[3+2]-cycloaddition

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

A direct fluorometric assay for tissue transglutaminase

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Biological activities of isatin and its derivatives.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Structure-activity relationship study of novel tissue transglutaminase inhibitors

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Mapping the kinase domain of Janus Kinase 3.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Oxindole-based compounds are selective inhibitors of Plasmodium falciparum cyclin dependent protein kinases.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Design, synthesis, and evaluation of gluten peptide analogs as selective inhibitors of human tissue transglutaminase

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Novel oxindole derivatives and their biological activity

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

Evaluation of novel dipeptide-bound alpha,beta-unsaturated amides and epoxides as irreversible inhibitors of guinea pig liver transglutaminase

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3081996

A highly diastereoselective, catalytic three-component assembly reaction for the synthesis of spiropyrrolidinyloxindoles

18 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21215619

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Transglutaminase inhibition by 2-[(2-oxopropyl)thio]imidazolium derivatives: mechanism of factor XIIIa inactivation

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21215619

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Synthesis of potential anticonvulsants: Condensation of isatins with acetone and related ketones

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21215619

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BMCL.2010.12.037

1 reference

13 October 2017

1 reference

13 October 2017

1 reference