(Q33370734)

26 July 2017

title

Identification of chemical inhibitors to human tissue transglutaminase by screening existing drug libraries (English)

1 reference

26 July 2017

0 references

James R Burke

7

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author name string

Thung-S Lai

1

1 reference

26 July 2017

Yusha Liu

2

1 reference

26 July 2017

Tim Tucker

3

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26 July 2017

Kurt R Daniel

4

1 reference

26 July 2017

David C Sane

5

1 reference

26 July 2017

Eric Toone

6

1 reference

26 July 2017

Warren J Strittmatter

8

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26 July 2017

Charles S Greenberg

9

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26 July 2017

publication date

1 September 2008

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26 July 2017

published in

Chemistry and Biology

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26 July 2017

volume

15

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26 July 2017

issue

9

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26 July 2017

page(s)

969-978

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Type 2 transglutaminase in neurodegenerative diseases: the mitochondrial connection

26 July 2017

cites work

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New uses for old drugs

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21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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The specificities of protein kinase inhibitors: an update

21 June 2018

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2-Methyl-1,4-naphthoquinone, vitamin K(3), decreases gap-junctional intercellular communication via activation of the epidermal growth factor receptor/extracellular signal-regulated kinase cascade.

21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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Potentiation of insulin-related signal transduction by a novel protein-tyrosine phosphatase inhibitor, Et-3,4-dephostatin, on cultured 3T3-L1 adipocytes

21 June 2018

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Specificity and mechanism of action of some commonly used protein kinase inhibitors

21 June 2018

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Cdc25 inhibition and cell cycle arrest by a synthetic thioalkyl vitamin K analogue.

21 June 2018

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Interactions of G(h)/transglutaminase with phospholipase Cdelta1 and with GTP

21 June 2018

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Epidermal growth factor receptor signaling cascade as target for tyrphostin (RG 50864) in epithelial cells. Paradoxical effects on mitogen-activated protein kinase kinase and mitogen-activated protein kinase activities

21 June 2018

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21 June 2018

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21 June 2018

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Mechanism and BASIS for Specificity of Transglutaminase-Catalyzed ε-(γ-Glutamyl) Lysine Bond Formation

21 June 2018

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Identification of a guanosine triphosphate-binding site on guinea pig liver transglutaminase. Role of GTP and calcium ions in modulating activity

21 June 2018

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A monoclonal antibody to cellular transglutaminase

21 June 2018

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Rapid uptake of tyrphostin into A431 human epidermoid cells is followed by delayed inhibition of epidermal growth factor (EGF)-stimulated EGF receptor tyrosine kinase activity

21 June 2018

1 reference

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Transglutaminases: multifunctional cross‐linking enzymes that stabilize tissues

21 June 2018

1 reference

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A microtiter plate transglutaminase assay utilizing 5-(biotinamido)pentylamine as substrate

21 June 2018

1 reference

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Protein transduction domain-mediated delivery of QBP1 suppresses polyglutamine-induced neurodegeneration in vivo.

21 June 2018

1 reference

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Covalent blocking of fibril formation and aggregation of intracellular amyloidgenic proteins by transglutaminase-catalyzed intramolecular cross-linking

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Effect of tissue transglutaminase on the solubility of proteins containing expanded polyglutamine repeats.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Tissue transglutaminase catalyzes the formation of alpha-synuclein crosslinks in Parkinson's disease

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Kinetic analysis of the action of tissue transglutaminase on peptide and protein substrates

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Therapeutic effects of cystamine in a murine model of Huntington's disease.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

'Tissue' transglutaminase ablation reduces neuronal death and prolongs survival in a mouse model of Huntington's disease

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Prolonged survival and decreased abnormal movements in transgenic model of Huntington disease, with administration of the transglutaminase inhibitor cystamine

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Fluorescence approaches to study G protein mechanisms.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Tau is modified by tissue transglutaminase in situ: possible functional and metabolic effects of polyamination.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Expanded polyglutamine protein forms nuclear inclusions and causes neural degeneration in Drosophila

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Carboxyl-terminal truncation of recombinant factor XIII A-chains. Characterization of minimum structural requirement for transglutaminase activity.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2637080

Regulation of human tissue transglutaminase function by magnesium-nucleotide complexes. Identification of distinct binding sites for Mg-GTP and Mg-ATP

31 October 2018

1 reference

12 December 2020

Naphthoquinone analogs as inactivators of cdc25 phosphatase

1 reference

12 December 2020

Kinetic analysis of the interaction of tissue transglutaminase with a nonpeptidic slow-binding inhibitor

1 reference

12 December 2020

A toxic monomeric conformer of the polyglutamine protein

1 reference

12 December 2020

The 1,4-naphthoquinone scaffold in the design of cysteine protease inhibitors

1 reference

12 December 2020

Inhibition of GTP-utilizing enzymes by tyrphostins

1 reference

12 December 2020

10.1016/J.CHEMBIOL.2008.07.015

Identifiers

DOI

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26 July 2017

1 reference

26 July 2017

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