(Q42232413)

19 October 2017

The DiPPro approach: synthesis, hydrolysis, and antiviral activity of lipophilic d4T diphosphate prodrugs (English)

1 reference

19 October 2017

2

Jan Balzarini

1 reference

19 October 2017

Tilmann Schulz

1

1 reference

PubMed ID

24616176

19 October 2017

Chris Meier

series ordinal

3

1 reference

19 October 2017

11 March 2014

1 reference

19 October 2017

1 reference

19 October 2017

9

1 reference

19 October 2017

4

1 reference

19 October 2017

762-775

1 reference

Metabolism and mechanism of antiretroviral action of purine and pyrimidine derivatives

19 October 2017

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Nucleoside and nucleotide HIV reverse transcriptase inhibitors: 25 years after zidovudine.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

cycloSal-Pronucleotides of 2',3'-dideoxyadenosine and 2', 3'-dideoxy-2',3'-didehydroadenosine: synthesis and antiviral evaluation of a highly efficient nucleotide delivery system

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

CycloSal-BVDUMP pronucleotides: how to convert an antiviral-inactive nucleoside analogue into a bioactive compound against EBV.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Aryloxy phosphoramidate triesters: a technology for delivering monophosphorylated nucleosides and sugars into cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

The application of phosphoramidate protide technology to acyclovir confers anti-HIV inhibition.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Prodrugs of phosphates and phosphonates

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

cycloSal-2',3'-dideoxy-2',3'-didehydrothymidine monophosphate (cycloSal-d4TMP): synthesis and antiviral evaluation of a new d4TMP delivery system

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Intracellular trapping of cycloSal-pronucleotides: modification of prodrugs with amino acid esters

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Doubly loaded cycloSaligenyl-pronucleotides - 5,5'-Bis-(cycloSaligenyl-2',3'-dideoxy-2',3'-didehydrothymidine monophosphates).

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Structure of thymidylate kinase reveals the cause behind the limiting step in AZT activation

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

3'-azido-3'-deoxythymidine (AZT) monophosphate: an inhibitor of exonucleolytic repair of AZT-terminated DNA

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

3'-Azidothymidine (zidovudine) inhibits glycosylation and dramatically alters glycosphingolipid synthesis in whole cells at clinically relevant concentrations

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Greatly enhanced inhibition of human immunodeficiency virus type 1 replication in CEM and HT4-6C cells by 3'-deoxythymidine diphosphate dimyristoylglycerol, a lipid prodrug of 3'-deoxythymidine

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Acyclovir diphosphate dimyristoylglycerol: a phospholipid prodrug with activity against acyclovir-resistant herpes simplex virus

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Comparative study of bis(benzyl)phosphate triesters of 2',3'-dideoxy-2',3'-didehydrothymidine (d4T) and cyclosal-d4TMP--hydrolysis, mechanistic insights and anti-HIV activity

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Enzymatically activated cycloSal-d4T-monophosphates: The third generation of cycloSal-pronucleotides

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Studies on enzyme-cleavable dialkoxymethyl-cyclosaligenyl-2',3'-dideoxy-2',3'-didehydrothymidine monophosphates

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

Diastereoselective synthesis of cyclosaligenyl-nucleosyl-phosphotriesters

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

7 January 2021

The bottleneck in AZT activation

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

7 January 2021

Lipid conjugates of antiretroviral agents: release of antiretroviral nucleoside monophosphates by a nucleoside diphosphate diglyceride hydrolase activity from rat liver mitochondria

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

7 January 2021

Bioreversible protection of nucleoside diphosphates

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

7 January 2021

Synthesis of a lipid/peptide/drug conjugate: N4-(acylpeptidyl)-ara-C

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201300500

7 January 2021

Identifiers

DOI

10.1002/CMDC.201300500

1 reference

19 October 2017

1 reference

PubMed ID

24616176